Allosteric interactions within the AT 1 angiotensin receptor homodimer: Role of the conserved DRY motif

Biochemical Pharmacology

Volumn 84, Issue 4, 2012, Pages 477-485

  Szalai, Bence ^a   Barkai, László ^a   Turu, Gábor ^a   Szidonya, László ^a   Várnai, Péter ^a   Hunyady, László ^a  

^a SEMMELWEIS UNIVERSITY   (Hungary)

Author keywords

Allosteric interaction; Angiotensin receptor; BRET; Dimerization; GPCR

Indexed keywords

ANGIOTENSIN 1 RECEPTOR; BETA ARRESTIN 2; GUANINE NUCLEOTIDE BINDING PROTEIN; HOMODIMER; RADIOLIGAND; RENILLA LUCIFERIN 2 MONOOXYGENASE; YELLOW FLUORESCENT PROTEIN;

ALLOSTERISM; ANIMAL CELL; ARTICLE; BIOLUMINESCENCE RESONANCE ENERGY TRANSFER; CARBOXY TERMINAL SEQUENCE; GENETIC CONSERVATION; LIGAND BINDING; NONHUMAN; PRIORITY JOURNAL; PROTEIN BINDING; PROTEIN CONFORMATION; PROTEIN INTERACTION;

ALLOSTERIC REGULATION; AMINO ACID MOTIFS; ANGIOTENSIN II TYPE 1 RECEPTOR BLOCKERS; ANIMALS; ARRESTINS; BACTERIAL PROTEINS; BIOLUMINESCENCE RESONANCE ENERGY TRANSFER TECHNIQUES; CHO CELLS; CONSERVED SEQUENCE; CRICETINAE; CRICETULUS; LUMINESCENT PROTEINS; MUTATION; PROMOTER REGIONS, GENETIC; PROTEIN BINDING; PROTEIN CONFORMATION; PROTEIN MULTIMERIZATION; RATS; RECEPTOR, ANGIOTENSIN, TYPE 1;

EID: 84864117586     PISSN: 00062952     EISSN: 18732968     Source Type: Journal    
DOI: 10.1016/j.bcp.2012.04.014     Document Type: Article

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