Synthesis and in vitro antitubercular activity of 4-aryl/ alkylsulfonylmethylcoumarins as inhibitors of Mycobacterium tuberculosis

Bioorganic and Medicinal Chemistry Letters

Volumn 22, Issue 14, 2012, Pages 4807-4809

  Jeyachandran, Malaichamy ^a   Ramesh, Penugonda ^b   Sriram, Dharmarajan ^c   Senthilkumar, Palaniappan ^c   Yogeeswari, Perumal ^c  

^a SRI PARAMAKALYANI COLLEGE   (India)

^b MADURAI KAMARAJ UNIVERSITY   (India)

^c BIRLA INSTITUTE OF TECHNOLOGY AND SCIENCE   (India)

Author keywords

4 Aryl alkylsulfonylmethylcoumarins; Antitubercular activity; Mycobacterium tuberculosis

Indexed keywords

4 ARYL ALKYLSULFONYLMETHYLCOUMARIN DERIVATIVE; COUMARIN DERIVATIVE; TUBERCULOSTATIC AGENT; UNCLASSIFIED DRUG;

ANTIBACTERIAL ACTIVITY; ARTICLE; DRUG SCREENING; DRUG SYNTHESIS; IN VITRO STUDY; MINIMUM INHIBITORY CONCENTRATION; MYCOBACTERIUM TUBERCULOSIS; NONHUMAN;

ANTITUBERCULAR AGENTS; MOLECULAR STRUCTURE; MYCOBACTERIUM TUBERCULOSIS; STRUCTURE-ACTIVITY RELATIONSHIP;

MYCOBACTERIUM TUBERCULOSIS;

EID: 84863453968     PISSN: 0960894X     EISSN: 14643405     Source Type: Journal    
DOI: 10.1016/j.bmcl.2012.05.054     Document Type: Article

References (26)

1. A.S. Ginsburg, J.H. Grosset, and W.R. Bishai Lancet Infect. Dis. 3 2003 432
2. D.G. Russell, C.E. Barry, and J.L. Flynn Science 328 2010 852
3. D.G. Russell Nat. Rev. Microbiol. 5 2007 39
4. S.H.E. Kaufmann, and A.J. McMichael Nat. Med. 11 2005 578
5. Y.C. Manabe, and W.R. Bishai Nat. Med. 6 2000 1327
6. A.G. Nikalie, and P. Mudassar Asian. J. Biol. Sci. 4 2011 101
7. J.C. Sacchettini, E.J. Rubin, and J.S. Freundlich Nat. Rev. Microbiol. 6 2008 41
8. Global tuberculosis control: a short update to the 2009 report. http://www.who.int/tb/publications/global-report/2009/update/en/index.html.
9. K. Duncan Tuberculosis 83 2003 201
10. W. Jie, L. Yun, and Y. Zhen J. Org. Chem. 66 2001 3642
11. O. Kayser, and H. Kolodziej Planta Med. 63 1997 508
12. S. Vilar, E. Quezada, L. Santana, E. Uriarte, M. Yanez, N. Fraiz, C. Alcaide, E. Cano, and F. Orallo Bioorg. Med. Chem. Lett. 16 2006 257
13. C.J. Wang, Y.J. Hsieh, C.Y. Chu, Y.L. Lin, and T.H. Tseng Cancer Lett. 183 2002 163
14. I. Kostova Curr. Med. Chem. Anti Cancer Agents 5 2005 29
15. M. Bhalla, P.K. Nathani, A. Kumar, T.N. Bhalla, and K. Shanker Indian. J. Chem., Sect. B 31 1992 183
16. S. Kirkiacharian, D.T. Thuy, S. Sicsic, R. Bakhchinian, R. Kurkjian, and T. Tonnaire Il Farmaco 57 9 2002 703
17. R.M. Jaysukhlal, S.G. Arvind, J.S. Paresh, and S.S. Shyam Chem. Ind. (London) 10 1979 351
18. R.M. Jaysukhlal, and J.S. Paresh Chem. Ind. (London) 19 1980 791
19. R.M. Jaysukhlal, M.K. Nirmal, and S.G. Arvind Chem. Ind. (London) 23 1982 955
20. Jie, W.; Zhen, Y.; Reza. F.; Qiang, Z. U.S. Pat. Appl. Publ., 752654, 538, 2004.
21. K. Serge, T.D. Thanh, S. Sames, B. Robert, K. Raffi, and T. Thierry Il Farmaco 57 2002 703
22. Z.M. Nofal, A.H. Mandour, and M.I. Nassar Egypt. J. Chem. 33 1990 509
23. Jeyachandran, M.; Ramesh, P. Organic Chemistry International, 2011, Article ID 360810, doi: http://dx.doi.org/10.1155/2011/360810.
24. P.S. Kumar, M. Dinakaran, D. Banerjee, R.V. Devakaram, P. Yogeeswari, A. China, V. Nagaraja, and D. Sriram Bioorg. Med. Chem. 16 2008 2558
25. M. Dinakaran, P.S. Kumar, P. Yogeeswari, A. China, V. Nagaraja, and D. Sriram Bioorg. Med. Chem. 16 2008 3408
26. M. Dinakaran, P.S. Kumar, P. Yogeeswari, A. China, V. Nagaraja, and D. Sriram Int. J. Antimicrob. Chemother. 31 2008 337