Route selection and process development of a multikilogram route to the inhaled A 2a agonist UK-432,097

Organic Process Research and Development

Volumn 16, Issue 3, 2012, Pages 470-483

  Ashcroft, Christopher P ^a   Dessi, Yann ^a   Entwistle, David A ^a   Hesmondhalgh, Lynsey C ^a   Longstaff, Adrian ^a   Smith, Julian D ^a  

^a PFIZER GLOBAL RESEARCH AND DEVELOPMENT   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

CRYSTALLIZATION PROCESS; ELEVATED TEMPERATURE; GLYCOSIDATIONS; NUCLEOSIDE ANALOGUES; PROCESS DEVELOPMENT; ROUTE SELECTION; SCALE-UP; STEREO-SELECTIVE; SYNTHETIC ROUTES;

EID: 84863341343     PISSN: 10836160     EISSN: 1520586X     Source Type: Journal    
DOI: 10.1021/op200365n     Document Type: Article

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