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Bioorganic and Medicinal Chemistry Letters

Volumn 22, Issue 9, 2012, Pages 3269-3273

New diarylureas and diarylamides possessing acet(benz)amidophenyl scaffold: Design, synthesis, and antiproliferative activity against melanoma cell line

(9) Kim, Hee Jin a Cho, Hye Jung a Kim, Hwan a El Gamal, Mohammed I a,b Oh, Chang Hyun a,b Lee, So Ha a Sim, Taebo a Hah, Jung Mi c Yoo, Kyung Ho a

a Korea Institute of Science and Technology (South Korea)

b University of Science and Technology (UST) (South Korea)

c Hanyang University (South Korea)

Author keywords

A375P; Acet(benz)amidophenyl; Antiproliferative activity; Diarylamide; Diarylurea; Melanoma

Indexed keywords

ANTINEOPLASTIC AGENT; AROMATIC AMIDE; BENZAMIDE DERIVATIVE; SORAFENIB; UREA DERIVATIVE; VEMURAFENIB;

ANTINEOPLASTIC ACTIVITY; ARTICLE; CELL PROLIFERATION; CONTROLLED STUDY; DRUG ABSORPTION; DRUG BIOAVAILABILITY; DRUG DESIGN; DRUG DISTRIBUTION; DRUG EXCRETION; DRUG METABOLISM; DRUG POTENCY; DRUG SOLUBILITY; DRUG SYNTHESIS; HUMAN; HUMAN CELL; IC 50; MELANOMA CELL; PREDICTION; REFRACTOMETRY; STRUCTURE ACTIVITY RELATION;

AMIDES; ANTINEOPLASTIC AGENTS; CELL LINE, TUMOR; CELL PROLIFERATION; DRUG DESIGN; HUMANS; MELANOMA; UREA;

EID: 84862777763 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2012.03.020 Document Type: Article

Times cited : (34)

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