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Volumn 232, Issue 2, 2012, Pages 416-420

Awakening properties of newly discovered highly selective H 3 receptor antagonists in rats

Author keywords

Awakening; EEG; Histamine H 3 receptor; Rats

Indexed keywords

6 (3 CYCLOBUTYL 2,3,4,5 TETRAHYDRO 1H 3 BENZAZEPIN 7 YLOXY) N METHYLNICOTINAMIDE; ABT 0239; ABT 039; AMPHETAMINE; CIPROXIFAN; HISTAMINE H3 RECEPTOR; HISTAMINE H3 RECEPTOR AGONIST; HISTAMINE H3 RECEPTOR ANTAGONIST; MODAFINIL; SAR 110068; SAR 110894; TETRAHYDRO PYRAN 4 CARBOXYLIC ACID [2 METHYL 4 (2 METHYL [1,3']BIPYRROLIDINYL 1' YL)PHENYL]AMIDE; UNCLASSIFIED DRUG;

EID: 84861681383     PISSN: 01664328     EISSN: 18727549     Source Type: Journal    
DOI: 10.1016/j.bbr.2012.04.033     Document Type: Article
Times cited : (18)

References (23)
  • 4
    • 77952351891 scopus 로고    scopus 로고
    • 3 receptor antagonists in dementias
    • 3 receptor antagonists in dementias. Drug News Perspect 2010, 23:99-103.
    • (2010) Drug News Perspect , vol.23 , pp. 99-103
    • Chazot, P.L.1
  • 13
    • 33845904178 scopus 로고    scopus 로고
    • BF2.649 [1-{3-[3-(4-chlorophenyl)propoxy]propyl}piperidine, hydrochloride], a non-imidazole inverse agonist/antagonist at the human histamine H3 receptor: preclinical pharmacology
    • Ligneau X., Perrin D., Landais L., Camelin J.C., Calmels T.P., Berrebi-Bertrand I., et al. BF2.649 [1-{3-[3-(4-chlorophenyl)propoxy]propyl}piperidine, hydrochloride], a non-imidazole inverse agonist/antagonist at the human histamine H3 receptor: preclinical pharmacology. Journal of Pharmacology and Experimental Therapeutics 2007, 320:365-375.
    • (2007) Journal of Pharmacology and Experimental Therapeutics , vol.320 , pp. 365-375
    • Ligneau, X.1    Perrin, D.2    Landais, L.3    Camelin, J.C.4    Calmels, T.P.5    Berrebi-Bertrand, I.6
  • 15
    • 80052912549 scopus 로고    scopus 로고
    • Effect of a novel histamine subtype-3 receptor inverse agonist and modafinil on EEG power spectra during sleep deprivation and recovery sleep in male volunteers
    • James L.M., Iannone R., Palcza J., Renger J.J., Calder N., Cerchio K., et al. Effect of a novel histamine subtype-3 receptor inverse agonist and modafinil on EEG power spectra during sleep deprivation and recovery sleep in male volunteers. Psychopharmacology (Berlin) 2011, 215:643-653.
    • (2011) Psychopharmacology (Berlin) , vol.215 , pp. 643-653
    • James, L.M.1    Iannone, R.2    Palcza, J.3    Renger, J.J.4    Calder, N.5    Cerchio, K.6
  • 16
    • 84861652480 scopus 로고    scopus 로고
    • SAR110894, a novel, potent and selective histamine H3 receptor (H3-R) antagonist: III. Potential activity in positive symptom and cognitive domains of schizophrenia using latent inhibition (LI) models in the rat
    • Program No 160.19. 2008 Neuroscience Meeting Planner Washington, DC: Society for Neuroscience November 15-19.
    • Black M, Pichat P, Weiner S, Barak S, Arad M, Delevie A, Varty GB, Bergis O, Griebel G. SAR110894, a novel, potent and selective histamine H3 receptor (H3-R) antagonist: III. Potential activity in positive symptom and cognitive domains of schizophrenia using latent inhibition (LI) models in the rat. Program No 160.19. 2008 Neuroscience Meeting Planner Washington, DC: Society for Neuroscience November 15-19; 2008.
    • (2008)
    • Black, M.1    Pichat, P.2    Weiner, S.3    Barak, S.4    Arad, M.5    Delevie, A.6    Varty, G.B.7    Bergis, O.8    Griebel, G.9
  • 17
    • 84861652478 scopus 로고    scopus 로고
    • SAR110894, a novel, potent and selective H3-receptor (H3-R) antagonist: II. Effects in models predictive of therapeutic activity against cognitive and attention deficits in schizophrenia and ADHD. Program No 160.20. 2008 Neuroscience Meeting Planner Washington, DC: Society for Neuroscience November 15-19.
    • Pichat P, Boulay D, Terranova JP, Decobert M, Françon D, Guillot E, Bergis O, Alonso R, Avenet P, Griebel G. SAR110894, a novel, potent and selective H3-receptor (H3-R) antagonist: II. Effects in models predictive of therapeutic activity against cognitive and attention deficits in schizophrenia and ADHD. Program No 160.20. 2008 Neuroscience Meeting Planner Washington, DC: Society for Neuroscience November 15-19; 2008.
    • (2008)
    • Pichat, P.1    Boulay, D.2    Terranova, J.P.3    Decobert, M.4    Françon, D.5    Guillot, E.6    Bergis, O.7    Alonso, R.8    Avenet, P.9    Griebel, G.10
  • 19
    • 34248562939 scopus 로고    scopus 로고
    • GSK189254, a novel H3 receptor antagonist that binds to histamine H3 receptors in Alzheimer's disease brain and improves cognitive performance in preclinical models
    • Medhurst A.D., Atkins A.R., Beresford I.J., Brackenborough K., Briggs M.A., Calver A.R., et al. GSK189254, a novel H3 receptor antagonist that binds to histamine H3 receptors in Alzheimer's disease brain and improves cognitive performance in preclinical models. Journal of Pharmacology and Experimental Therapeutics 2007, 321:1032-1045.
    • (2007) Journal of Pharmacology and Experimental Therapeutics , vol.321 , pp. 1032-1045
    • Medhurst, A.D.1    Atkins, A.R.2    Beresford, I.J.3    Brackenborough, K.4    Briggs, M.A.5    Calver, A.R.6
  • 21
    • 33947121092 scopus 로고    scopus 로고
    • 3 receptor antagonists GSK207040 and GSK334429 improve scopolamine-induced memory impairment and capsaicin-induced secondary allodynia in rats
    • 3 receptor antagonists GSK207040 and GSK334429 improve scopolamine-induced memory impairment and capsaicin-induced secondary allodynia in rats. Biochemical Pharmacology 2007, 73:1182-1194.
    • (2007) Biochemical Pharmacology , vol.73 , pp. 1182-1194
    • Medhurst, A.D.1    Briggs, M.A.2    Bruton, G.3    Calver, A.R.4    Chessell, I.5    Crook, B.6
  • 23
    • 3843054587 scopus 로고    scopus 로고
    • Pharmacological and behavioral properties of A-349821, a selective and potent human histamine H3 receptor antagonist
    • Esbenshade T.A., Fox G.B., Krueger K.M., Baranowski J.L., Miller T.R., Kang C.H., et al. Pharmacological and behavioral properties of A-349821, a selective and potent human histamine H3 receptor antagonist. Biochemical Pharmacology 2004, 68:933-945.
    • (2004) Biochemical Pharmacology , vol.68 , pp. 933-945
    • Esbenshade, T.A.1    Fox, G.B.2    Krueger, K.M.3    Baranowski, J.L.4    Miller, T.R.5    Kang, C.H.6


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.