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Volumn 56, Issue 6, 2012, Pages 2814-2818

In Vitro antimalarial activity and drug interactions of fenofibric acid

Author keywords

[No Author keywords available]

Indexed keywords

ABC TRANSPORTER; ATORVASTATIN; CHLOROQUINE; CLOFIBRATE; DIHYDROARTEMISININ; FENOFIBRIC ACID; GEMFIBROZIL; ISOTOPE;

EID: 84861152021     PISSN: 00664804     EISSN: 10986596     Source Type: Journal    
DOI: 10.1128/AAC.05076-11     Document Type: Article
Times cited : (5)

References (37)
  • 1
    • 20144373625 scopus 로고    scopus 로고
    • Fenofibric acid, an active form of fenofibrate, increases apolipoprotein A-I-mediated high-density lipoprotein biogenesis by enhancing transcription of ATP-binding cassette transporter A1 gene in a liver X receptor-dependent manner
    • DOI 10.1161/01.ATV.0000163844.07815.c4
    • Arakawa R, Tamehiro N, Nishimaki-Mogami T, Ueda K, Yokoyama S. 2005. Fenofibric acid, an active form of fenofibrate, increases apolipoprotein A-I-mediated high-density lipoprotein biogenesis by enhancing transcription of ATP-binding cassette transporter A1 gene in a liver X receptor- dependent manner. Arterioscler. Thromb. Vasc. Biol. 25:1193-1197. (Pubitemid 40776608)
    • (2005) Arteriosclerosis, Thrombosis, and Vascular Biology , vol.25 , Issue.6 , pp. 1193-1197
    • Arakawa, R.1    Tamehiro, N.2    Nishimaki-Mogami, T.3    Ueda, K.4    Yokoyama, S.5
  • 2
    • 0017843255 scopus 로고
    • A method for testing for synergy with any number of agents
    • Berenbaum MC. 1978. A method for testing for synergy with any number of agents. J. Infect. Dis. 137:122-130. (Pubitemid 8289152)
    • (1978) Journal of Infectious Diseases , vol.137 , Issue.2 , pp. 122-130
    • Berenbaum, M.C.1
  • 3
    • 70349503854 scopus 로고    scopus 로고
    • Determination of fenofibric acid in human plasma by ultra performance liquid chromatography-electrospray ionization mass spectrometry: Application to a bioequivalence study
    • Bhavesh D, Shah S. 2009. Determination of fenofibric acid in human plasma by ultra performance liquid chromatography-electrospray ionization mass spectrometry: application to a bioequivalence study. Biomed. Chromatogr. 23:922-928.
    • (2009) Biomed. Chromatogr. , vol.23 , pp. 922-928
    • Bhavesh, D.1    Shah, S.2
  • 4
    • 70049086389 scopus 로고    scopus 로고
    • Use of peroxisome proliferator-activated receptor gamma agonists as adjunctive treatment for Plasmodium falciparum malaria: A randomized, double-blind, placebo-controlled trial
    • Boggild AK, et al. 2009. Use of peroxisome proliferator-activated receptor gamma agonists as adjunctive treatment for Plasmodium falciparum malaria: a randomized, double-blind, placebo-controlled trial. Clin. Infect. Dis. 49:841- 849.
    • (2009) Clin. Infect. Dis. , vol.49 , pp. 841-849
    • Boggild, A.K.1
  • 6
    • 0037265207 scopus 로고    scopus 로고
    • Persistence of atovaquone in human sera following treatment: Inhibition of Plasmodium falciparum development in vivo and in vitro
    • Butcher GA, Sinden RE. 2003. Persistence of atovaquone in human sera following treatment: inhibition of Plasmodium falciparum development in vivo and in vitro. Am. J. Trop. Med. Hyg. 68:111-114. (Pubitemid 38234858)
    • (2003) American Journal of Tropical Medicine and Hygiene , vol.68 , Issue.1 , pp. 111-114
    • Butcher, G.A.1    Sinden, R.E.2
  • 7
    • 0029078941 scopus 로고
    • Interactions of atovaquone with other antimalarial drugs against Plasmodium falciparum in vitro
    • Canfield CJ, Pudney M, Gutteridge WE. 1995. Interactions of atovaquone with other antimalarial drugs against Plasmodium falciparum in vitro. Exp. Parasitol. 80:373-381.
    • (1995) Exp. Parasitol. , vol.80 , pp. 373-381
    • Canfield, C.J.1    Pudney, M.2    Gutteridge, W.E.3
  • 8
    • 84858449712 scopus 로고    scopus 로고
    • Changes in the treatment responses to artesunatemefloquine on the northwestern border of Thailand during 13 years of continuous deployment
    • Carrara VI, et al. 2009. Changes in the treatment responses to artesunatemefloquine on the northwestern border of Thailand during 13 years of continuous deployment. PLoS One 4:e4551.
    • (2009) PLoS One , vol.4
    • Carrara, V.I.1
  • 10
    • 67649528611 scopus 로고    scopus 로고
    • Is human malarial coma caused, or merely deepened, by sequestration?
    • Clark IA, Alleva LM. 2009. Is human malarial coma caused, or merely deepened, by sequestration? Trends Parasitol. 25:314-318.
    • (2009) Trends Parasitol. , vol.25 , pp. 314-318
    • Clark, I.A.1    Alleva, L.M.2
  • 11
    • 40649097787 scopus 로고    scopus 로고
    • Understanding the role of inflammatory cytokines in malaria and related diseases
    • Clark IA, Alleva LM, Budd AC, Cowden WB. 2008. Understanding the role of inflammatory cytokines in malaria and related diseases. Travel Med. Infect. Dis. 6:67- 81.
    • (2008) Travel Med. Infect. Dis. , vol.6 , pp. 67-81
    • Clark, I.A.1    Alleva, L.M.2    Budd, A.C.3    Cowden, W.B.4
  • 12
    • 78951474167 scopus 로고    scopus 로고
    • Effects of fenofibrate on renal function in patients with type 2 diabetes mellitus: The Fenofibrate Intervention and Event Lowering in Diabetes (FIELD) Study
    • Davis TM, et al. 2011. Effects of fenofibrate on renal function in patients with type 2 diabetes mellitus: the Fenofibrate Intervention and Event Lowering in Diabetes (FIELD) Study. Diabetologia 54:280-290.
    • (2011) Diabetologia , vol.54 , pp. 280-290
    • Davis, T.M.1
  • 13
    • 67650844186 scopus 로고    scopus 로고
    • Fenofibrate, simvastatin and their combination in the management of dyslipidaemia in type 2 diabetic patients
    • Derosa G, et al. 2009. Fenofibrate, simvastatin and their combination in the management of dyslipidaemia in type 2 diabetic patients. Curr. Med. Res. Opin. 25:1973-1983.
    • (2009) Curr. Med. Res. Opin. , vol.25 , pp. 1973-1983
    • Derosa, G.1
  • 14
    • 0029737127 scopus 로고    scopus 로고
    • Pharmaco-dynamic activity of lipoprotein lipase and hepatic lipase, and pharmacokinetic parameters measured in normolipidaemic subjects receiving ciprofibrate (100 or 200 mg/day) or micronised fenofibrate (200 mg/day) therapy for 23 days
    • Desager JP, Horsmans Y, Vandenplas C, Harvengt C. 1996. Pharmaco-dynamic activity of lipoprotein lipase and hepatic lipase, and pharmacokinetic parameters measured in normolipidaemic subjects receiving ciprofibrate (100 or 200 mg/day) or micronised fenofibrate (200 mg/day) therapy for 23 days. Atherosclerosis 124(Suppl):S65-S73.
    • (1996) Atherosclerosis , vol.124 , Issue.SUPPL.
    • Desager, J.P.1    Horsmans, Y.2    Vandenplas, C.3    Harvengt, C.4
  • 15
    • 0018606732 scopus 로고
    • Quantitative assessment of antimalarial activity in vitro by semiautomated microdilution technique
    • Desjardin RE, Canfield Haynes CJ, Chulay DJD. 1979. Quantitative assessment of antimalarial activity in vitro by semiautomated microdilution technique. Antimicrob. Agents Chemother. 16:710-718.
    • (1979) Antimicrob. Agents Chemother. , vol.16 , pp. 710-718
    • Desjardin, R.E.1    Canfield Haynes, C.J.2    Chulay, D.J.D.3
  • 16
    • 77949568358 scopus 로고    scopus 로고
    • Artemisinin resistance: Current status and scenarios for containment
    • Dondorp AM, et al. 2010. Artemisinin resistance: current status and scenarios for containment. Nat. Rev. Microbiol. 8:272-280.
    • (2010) Nat. Rev. Microbiol. , vol.8 , pp. 272-280
    • Dondorp, A.M.1
  • 17
    • 77649319341 scopus 로고    scopus 로고
    • Rapid, sensitive and validated ultra-performance liquid chromatography/mass spectrometric method for the determination of fenofibric acid and its application to human pharmacokinetic study
    • Dubey S, et al. 2010. Rapid, sensitive and validated ultra-performance liquid chromatography/mass spectrometric method for the determination of fenofibric acid and its application to human pharmacokinetic study. E-J. Chem. 7:25-36.
    • (2010) E-J. Chem. , vol.7 , pp. 25-36
    • Dubey, S.1
  • 20
    • 7244240741 scopus 로고    scopus 로고
    • Modified fixed-ratio isobologram method for studying in vitro interactions between atovaquone and proguanil or dihydroartemisinin against drug-resistant strains of Plasmodium falciparum
    • DOI 10.1128/AAC.48.11.4097-4102.2004
    • Fivelman QL, Adagu IS, Warhurst DC. 2004. Modified fixed-ratio isobologram method for studying in vitro interactions between atovaquone and proguanil or dihydroartemisinin against drug-resistant strains of Plasmodium falciparum. Antimicrob. Agents Chemother. 48: 4097-4102. (Pubitemid 39434861)
    • (2004) Antimicrobial Agents and Chemotherapy , vol.48 , Issue.11 , pp. 4097-4102
    • Fivelman, Q.L.1    Adagu, I.S.2    Warhurst, D.C.3
  • 21
    • 84861117116 scopus 로고    scopus 로고
    • Therapeutic uses of PPAR mediators
    • November U.S. patent 20030220373A1
    • Jaye M, Duverger N, Searfoss G, Minnich A. November 2003. Therapeutic uses of PPAR mediators. U.S. patent 20030220373A1.
    • (2003)
    • Jaye, M.1    Duverger, N.2    Searfoss, G.3    Minnich, A.4
  • 22
    • 74549192880 scopus 로고    scopus 로고
    • A comparative study of a flow-cytometry-based assessment of in vitro Plasmodium falciparum drug sensitivity
    • Karl S, Wong RP, St Pierre TG, Davis TM. 2009. A comparative study of a flow-cytometry-based assessment of in vitro Plasmodium falciparum drug sensitivity. Malar. J. 8:294 -304.
    • (2009) Malar. J. , vol.8 , pp. 294-304
    • Karl, S.1    Wong, R.P.2    St Pierre, T.G.3    Davis, T.M.4
  • 23
    • 0036382889 scopus 로고    scopus 로고
    • Micronised fenofibrate: An updated review of its clinical efficacy in the management of dyslipidaemia
    • Keating GM, Ormrod D. 2002. Micronised fenofibrate: an updated review of its clinical efficacy in the management of dyslipidaemia. Drugs 62:1909 -1944.
    • (2002) Drugs , vol.62 , pp. 1909-1944
    • Keating, G.M.1    Ormrod, D.2
  • 24
    • 28044452217 scopus 로고    scopus 로고
    • Effects of long-term fenofibrate therapy on cardiovascular events in 9795 people with type 2 diabetes mellitus (the FIELD study): Randomised controlled trial
    • Keech A, et al. 2005. Effects of long-term fenofibrate therapy on cardiovascular events in 9795 people with type 2 diabetes mellitus (the FIELD study): randomised controlled trial. Lancet 366:1849 -1861.
    • (2005) Lancet , vol.366 , pp. 1849-1861
    • Keech, A.1
  • 25
    • 0031968706 scopus 로고    scopus 로고
    • Effectiveness and tolerability of 12-week treatment with micronised fenofibrate 200 mg in a drug-monitoring programme involving 9884 patients with dyslipidaemia
    • DOI 10.2165/00044011-199815030-00004
    • Kirchgassler KU, Schmitz H, Bach G. 1998. Effectiveness and tolerability of 12-week treatment with micronised fenofibrate 200 mg in a drug monitoring programme involving 9884 patients with dyslipidaemia. Clin. Drug Invest. 15:197-204. (Pubitemid 28163746)
    • (1998) Clinical Drug Investigation , vol.15 , Issue.3 , pp. 197-204
    • Kirchgassler, K.U.1    Schmitz, H.2    Bach, G.3
  • 26
    • 0018704491 scopus 로고
    • Synchronization of Plasmodium falciparum erythrocytic stages in culture
    • DOI 10.2307/3280287
    • Lambros C, Vanderberg JP. 1979. Synchronization of Plasmodium falciparum erythrocytic stages in culture. J. Parasitol. 65:418-420. (Pubitemid 10222999)
    • (1979) Journal of Parasitology , vol.65 , Issue.3 , pp. 418-420
    • Lambros, C.1    Vanderberg, J.P.2
  • 27
    • 0018378241 scopus 로고
    • Effect of temperature and clofibrate on Plasmodium berghei infection in mice
    • McQuistion TE. 1979. Effect of temperature and clofibrate on Plasmodium berghei infection in mice. Am. J. Trop. Med. Hyg. 28:12-14. (Pubitemid 9111786)
    • (1979) American Journal of Tropical Medicine and Hygiene , vol.28 , Issue.1 , pp. 12-14
    • McQuistion, T.E.1
  • 28
    • 0031909536 scopus 로고    scopus 로고
    • Clinical pharmacokinetics of fibric acid derivatives (Fibrates)
    • DOI 10.2165/00003088-199834020-00003
    • Miller DB, Spence JD. 1998. Clinical pharmacokinetics of fibric acid derivatives (fibrates). Clin. Pharmacokinet. 34:155-162. (Pubitemid 28077673)
    • (1998) Clinical Pharmacokinetics , vol.34 , Issue.2 , pp. 155-162
    • Miller, D.B.1    Spence, J.D.2
  • 29
    • 33846566278 scopus 로고    scopus 로고
    • Activity of azithromycin or erythromycin in combination with antimalarial drugs against multidrug-resistant Plasmodium falciparum in vitro
    • DOI 10.1016/j.actatropica.2006.10.008, PII S0001706X06002087
    • Nakornchai S, Konthiang P. 2006. Activity of azithromycin or erythromycin in combination with antimalarial drugs against multidrugresistant Plasmodium falciparum in vitro. Acta Trop. 100:185-191. (Pubitemid 46176762)
    • (2006) Acta Tropica , vol.100 , Issue.3 , pp. 185-191
    • Nakornchai, S.1    Konthiang, P.2
  • 30
    • 67049107926 scopus 로고    scopus 로고
    • Atorvastatin is a promising partner for antimalarial drugs in treatment of Plasmodium falciparum malaria
    • Parquet V, et al. 2009. Atorvastatin is a promising partner for antimalarial drugs in treatment of Plasmodium falciparum malaria. Antimicrob. Agents Chemother. 53:2248-2252.
    • (2009) Antimicrob. Agents Chemother. , vol.53 , pp. 2248-2252
    • Parquet, V.1
  • 32
    • 0034708162 scopus 로고    scopus 로고
    • Pgh1 modulates sensitivity and resistance to multiple antimalarials in Plasmodium falciparum
    • DOI 10.1038/35002615
    • Reed MB, Saliba KJ, Caruana SR, Kirk K, Cowman AF. 2000. Pgh1 modulates sensitivity and resistance to multiple antimalarials in Plasmodium falciparum. Nature 403:906-909. (Pubitemid 30130994)
    • (2000) Nature , vol.403 , Issue.6772 , pp. 906-909
    • Reed, M.B.1    Sallba, K.J.2    Caruana, S.R.3    Kirk, K.4    Cowman, A.F.5
  • 34
    • 66149139771 scopus 로고    scopus 로고
    • Statins as potential antimalarial drugs: Low relative potency and lack of synergy with conventional antimalarial drugs
    • Wong R, Davis TM. 2009. Statins as potential antimalarial drugs: low relative potency and lack of synergy with conventional antimalarial drugs. Antimicrob. Agents Chemother. 53:2212-2214.
    • (2009) Antimicrob. Agents Chemother. , vol.53 , pp. 2212-2214
    • Wong, R.1    Davis, T.M.2
  • 35
    • 79952339074 scopus 로고    scopus 로고
    • Desbutyl-lumefantrine is a metabolite of lumefantrine with potent in vitro antimalarial activity that may influence artemether-lumefantrine treatment outcome
    • Wong RP, et al. 2011. Desbutyl-lumefantrine is a metabolite of lumefantrine with potent in vitro antimalarial activity that may influence artemether-lumefantrine treatment outcome. Antimicrob. Agents Chemother. 55:1194 -1198.
    • (2011) Antimicrob. Agents Chemother. , vol.55 , pp. 1194-1198
    • Wong, R.P.1
  • 36
    • 45249099771 scopus 로고    scopus 로고
    • Declining artesunatemefloquine efficacy against falciparum malaria on the Cambodia- Thailand border
    • Wongsrichanalai C, Meshnick SR. 2008. Declining artesunatemefloquine efficacy against falciparum malaria on the Cambodia- Thailand border. Emerg. Infect. Dis. 14:716 -719.
    • (2008) Emerg. Infect. Dis. , vol.14 , pp. 716-719
    • Wongsrichanalai, C.1    Meshnick, S.R.2
  • 37
    • 77955780152 scopus 로고    scopus 로고
    • Comparison of the gastrointestinal absorption and bioavailability of fenofibrate and fenofibric acid in humans
    • Zhu T, Ansquer JC, Kelly MT, Sleep DJ, Pradhan RS. 2010. Comparison of the gastrointestinal absorption and bioavailability of fenofibrate and fenofibric acid in humans. J. Clin. Pharmacol. 50:914 -921.
    • (2010) J. Clin. Pharmacol. , vol.50 , pp. 914-921
    • Zhu, T.1    Ansquer, J.C.2    Kelly, M.T.3    Sleep, D.J.4    Pradhan, R.S.5


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