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Bioorganic and Medicinal Chemistry Letters

Volumn 22, Issue 8, 2012, Pages 2948-2950

Synthesis and biological evaluation of novel small non-peptidic HIV-1 PIs: The benzothiophene ring as an effective moiety

(6) Chiummiento, Lucia a Funicello, Maria a Lupattelli, Paolo a Tramutola, Francesco a Berti, Federico b Marino Merlo, Francesca c

a UNIVERSITY OF BASILICATA (Italy)

b UNIVERSITY OF TRIESTE (Italy)

c UNIVERSITY OF MESSINA (Italy)

Author keywords

Heterocycles; HIV protease; Inhibitor; Synthesis

Indexed keywords

BENZOTHIOPHENE DERIVATIVE; HUMAN IMMUNODEFICIENCY VIRUS PROTEINASE; HUMAN IMMUNODEFICIENCY VIRUS PROTEINASE INHIBITOR;

ANTIVIRAL ACTIVITY; ARTICLE; DRUG POTENCY; DRUG STRUCTURE; DRUG SYNTHESIS; HUMAN IMMUNODEFICIENCY VIRUS 1; HYDROPHOBICITY; NONHUMAN; REACTION ANALYSIS; STRUCTURE ANALYSIS;

ANTIVIRAL AGENTS; HETEROCYCLIC COMPOUNDS; HIV PROTEASE INHIBITORS; HIV-1; HUMANS; INHIBITORY CONCENTRATION 50; MOLECULAR STRUCTURE; THIOPHENES;

HUMAN IMMUNODEFICIENCY VIRUS 1;

EID: 84859439361 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2012.02.046 Document Type: Article

Times cited : (23)

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