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Bioorganic and Medicinal Chemistry Letters

Volumn 22, Issue 8, 2012, Pages 2850-2855

Radioiodinated sunitinib as a potential radiotracer for imaging angiogenesis - Radiosynthesis and first radiopharmacological evaluation of 5-[ 125I]Iodo-sunitinib

(5) Kuchar, Manuela a Oliveira, Maria Cristina b Gano, Lurdes b Santos, Isabel b Kniess, Torsten a

a INSTITUTE OF ION BEAM PHYSICS AND MATERIALS RESEARCH (Germany)

b INSTITUTO TECNOLÓGICO E NUCLEAR (Portugal)

Author keywords

Iodine 125; Radiolabeling; RTKs; Sunitinib ; VEGFR

Indexed keywords

5 IODOSUNITINIB I 125; IODINE 125; SUNITINIB; TRACER; UNCLASSIFIED DRUG;

ANGIOGENESIS; ANIMAL EXPERIMENT; ARTICLE; DRUG DISTRIBUTION; DRUG SYNTHESIS; DRUG UPTAKE; FEMALE; HUMAN; KNOEVENAGEL CONDENSATION; MOUSE; NONHUMAN; REACTION ANALYSIS;

ANGIOGENESIS INHIBITORS; ANIMALS; CELL PROLIFERATION; FEMALE; HUMANS; INDOLES; INHIBITORY CONCENTRATION 50; IODINE RADIOISOTOPES; MAGNETIC RESONANCE SPECTROSCOPY; MICE; MOLECULAR STRUCTURE; PYRROLES; RADIOPHARMACEUTICALS;

MUS;

EID: 84859438032 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2012.02.068 Document Type: Article

Times cited : (36)

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