Controlled delivery of nanosuspensions from osmotic pumps: Zero order and non-zero order kinetics

Journal of Controlled Release

Volumn 158, Issue 3, 2012, Pages 403-412

  Hill, Alexandra ^a,b   Geißler, Simon ^b   Weigandt, Markus ^b   Mäder, Karsten ^a  

^a MARTIN LUTHER UNIVERSITY HALLE WITTENBERG   (Germany)

^b MERCK KGAA   (Germany)

Author keywords

Burst release; Nanosuspension; Osmotic pumps; Preclinical development; Pump position; Viscosity

Indexed keywords

BURST RELEASE; NANO-SUSPENSIONS; OSMOTIC PUMPS; PRECLINICAL DEVELOPMENT; PUMP POSITION;

AROMATIC COMPOUNDS; BIOCHEMISTRY; DRUG PRODUCTS; ORGANIC POLYMERS; ORIFICES; OSMOSIS; SALINE WATER; VISCOSITY;

PUMPS;

FENOFIBRATE; FLUORESCEIN SODIUM; METHYLENE BLUE; NANOMATERIAL; NANOSUSPENSION; UNCLASSIFIED DRUG;

ARTICLE; DRUG DELIVERY SYSTEM; DRUG FORMULATION; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; IN VITRO STUDY; OSMOLALITY; OSMOTIC PUMP; PARTICLE SIZE; PRIORITY JOURNAL; SUSPENSION; ULTRAVIOLET RADIATION; VISCOSITY;

ANTIHYPERTENSIVE AGENTS; CAPTOPRIL; COLORING AGENTS; DELAYED-ACTION PREPARATIONS; FENOFIBRATE; FLUORESCEIN; HYPOLIPIDEMIC AGENTS; INFUSION PUMPS, IMPLANTABLE; KINETICS; METHYLENE BLUE; OSMOSIS; PARTICLE SIZE; SUSPENSIONS;

EID: 84859267161     PISSN: 01683659     EISSN: 18734995     Source Type: Journal    
DOI: 10.1016/j.jconrel.2011.12.005     Document Type: Article

References (29)

1. V.B. Patravale, A.A. Date, and R.M. Kulkarni Nanosuspensions: a promising drug delivery strategy J. Pharm. Pharmacol. 56 2004 827 840 (Pubitemid 38885975)
2. B.E. Rabinow Nanosuspensions in drug delivery Nat. Rev. Drug Discov. 3 2004 785 796 (Pubitemid 39242830)
3. P. Kocbek, S. Baumgartner, and J. Kristl Preparation and evaluation of nanosuspensions for enhancing the dissolution of poorly soluble drugs Int. J. Pharm. 312 2006 179 186
4. C.M. Keck, and R.H. Muller Drug nanocrystals of poorly soluble drugs produced by high pressure homogenisation Eur. J. Pharm. Biopharm. 62 2006 3 16 (Pubitemid 41736019)
5. J. Wong, A. Brugger, A. Khare, M. Chaubal, P. Papadopoulos, B. Rabinow, J. Kipp, and J. Ning Suspensions for intravenous (IV) injection: a review of development, preclinical and clinical aspects Adv. Drug Deliv. Rev. 60 2008 939 954
6. S. Rose, and J.F. Nelson A continuous long-term injector Aust. J. Exp. Biol. Med. Sci. 33 1955 415 419
7. T. Higuchi, H. M.Leeper, Improved osmotic dispenser employing magnesium sulfate and magnesium chloride, US patent 3760804 (1973).
8. F. Theeuwes, Osmotically powered agent dispending device with filling means, US patent 3760984 (1973).
9. J.C. Wright, L.S. Tao, C.L. Stevenson, J.C. Beck, G. Chen, R.M. Jao, P.A. Johnson, J. Leonard, and R.J. Skowronski An in vivo/in vitro comparison with a leuprolide osmotic implant for the treatment of prostate cancer J. Control. Release 75 2001 1 10 (Pubitemid 32635192)
10. B. Eckenhoff, and S.I. Yum The osmotic pump: novel research tool for optimizing drug regimens Biomaterials 2 1981 89 97 (Pubitemid 11080763)
11. A.K. Dash, and G.C. Cudworth Therapeutic applications of implantable drug delivery systems J. Pharmacol. Toxicol. Methods 40 1998 1 12 (Pubitemid 29062900)
12. H. Fansa, W. Schneider, G. Wolf, and G. Keilhoff Influence of insulin-like growth factor-I (IGF-I) on nerve autografts and tissue-engineered nerve grafts Muscle Nerve 26 2002 87 93 (Pubitemid 34734400)
13. J. Ambati, E.S. Gragoudas, J.W. Miller, T.T. You, K. Miyamoto, F.C. Delori, and A.P. Adamis Transscleral delivery of bioactive protein to the choroid and retina Invest. Ophthalmol. Vis. Sci. 41 2000 1186 1191 (Pubitemid 30187559)
14. B.R. Pratt, R.L. Butcher, and E.K. Inskeep Effect of continuous intrauterine administration of prostaglandin E2 on life span of corpora lutea of nonpregnant ewes J. Anim. Sci. 48 1979 1441 1446
15. J. Rousseau, J.F. Adam, P. Deman, T.D. Wu, J.L. Guerquin-Kern, B. Gouget, R.F. Barth, F. Esteve, and H. Elleaume Intracerebral delivery of 5-iodo-2′-deoxyuridine in combination with synchrotron stereotactic radiation for the therapy of the F98 glioma J. Synchrotron Radiat. 16 2009 573 581
16. F. Theeuwes, and S.I. Yum Principles of the design and operation of generic osmotic pumps for the delivery of semisolid or liquid drug formulations Ann. Biomed. Eng. 4 1976 343 353
17. B. Eckenhoff Osmotically driven pumps for the rate-controlled delivery of solutions and viscous suspensions AlChE Symp. Ser. 77 1981 1 9 (Pubitemid 11420793)
18. J.R. Zingerman, J.R. Cardinal, R.T. Chern, J. Holste, J.B. Williams, B. Eckenhoff, and J. Wright The in vitro and in vivo performance of an osmotically controlled delivery system-IVOMEC SR-bolus J. Control. Release 47 1997 1 11
19. E. Merisko-Liversidge, P. Sarpotdar, J. Bruno, S. Hajj, L. Wei, N. Peltier, J. Rake, J.M. Shaw, S. Pugh, L. Polin, J. Jones, T. Corbett, E. Cooper, and G.G. Liversidge Formulation and antitumor activity evaluation of nanocrystalline suspensions of poorly soluble anticancer drugs Pharm. Res. 13 1996 272 278 (Pubitemid 26074194)
20. J.W. Mouton, A. van Peer, K. de Beule, V.A. Van, J.P. Donnelly, and P.A. Soons Pharmacokinetics of itraconazole and hydroxyitraconazole in healthy subjects after single and multiple doses of a novel formulation Antimicrob. Agents Chemother. 50 2006 4096 4102 (Pubitemid 44865154)
21. B. Bittner, T. Thelly, H. Isel, and R.J. Mountfield The impact of co-solvents and the composition of experimental formulations on the pump rate of the ALZET osmotic pump Int. J. Pharm. 205 2000 195 198
22. S.Z. Kerenyi, and S.L. Hartgraves Premature excess release from the Alzet osmotic pump Pharmacol. Biochem. Behav. 27 1987 199 201 (Pubitemid 17096860)
23. S.G. Ortiz, T. Ma, N.J. Epstein, R.L. Smith, and S.B. Goodman Validation and quantification of an in vitro model of continuous infusion of submicron-sized particles J. Biomed. Mater. Res. B Appl. Biomater. 84B 2008 328 333
24. T.E. Sweeney, and C.A. Beuchat Limitations of methods of osmometry: measuring the osmolality of biological fluids Am. J. Physiol. 264 1993 R469 R480
25. D.R. Powell, J. Swarbrick, and G.S. Banker Effects of shear processing and thermal exposure on the viscosity-stability of polymer solutions J. Pharm. Sci. 55 1966 601 605
26. O. Mengual, G. Meunier, I. Cayre, K. Puech, and P. Snabre TURBISCAN MA 2000: multiple light scattering measurement for concentrated emulsion and suspension instability analysis Talanta 50 1999 445 456
27. J. Shokri, P. Ahmadi, P. Rashidi, M. Shahsavari, A. Rajabi-Siahboomi, and A. Nokhodchi Swellable elementary osmotic pump (SEOP): an effective device for delivery of poorly water-soluble drugs Eur. J. Pharm. Biopharm. 68 2008 289 297
28. C.C. Miller The Stokes-Einstein law for diffusion in solution Proc. R. Soc. London, Ser. A 106 1924 724 749
29. X. Ye, and P. Tong Transport of probe particles in semidilute polymer solutions Macromolecules 31 1998 5785 5793 (Pubitemid 128563337)