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Bioorganic and Medicinal Chemistry Letters

Volumn 22, Issue 3, 2012, Pages 1330-1334

Evaluation of vitamin D3 A-ring analogues as Hedgehog pathway inhibitors

(3) Banerjee, Upasana a Ghosh, Manuka a Kyle Hadden, M a

a UNIVERSITY OF CONNECTICUT (United States)

Author keywords

Cyp24A1; Gli1; Hedgehog pathway; Vitamin D receptor; Vitamin D3

Indexed keywords

ANTINEOPLASTIC AGENT; CELL PROTEIN; COLECALCIFEROL DERIVATIVE; CYP24A1 PROTEIN; MESSENGER RNA; SONIC HEDGEHOG PROTEIN; TRANSCRIPTION FACTOR GLI1; UNCLASSIFIED DRUG; VITAMIN D RECEPTOR; VITAMIN D3 A RING DERIVATIVE;

ANTINEOPLASTIC ACTIVITY; ANTIPROLIFERATIVE ACTIVITY; ARTICLE; BINDING AFFINITY; CONTROLLED STUDY; DOWN REGULATION; DRUG SCREENING; HUMAN; HUMAN CELL; IC 50; METHYLATION; MITSUNOBU REACTION; SIGNAL TRANSDUCTION; STRUCTURE ACTIVITY RELATION; UPREGULATION;

ANTINEOPLASTIC AGENTS; CELL LINE, TUMOR; CHOLECALCIFEROL; HEDGEHOG PROTEINS; HUMANS; MOLECULAR STRUCTURE; SIGNAL TRANSDUCTION; STRUCTURE-ACTIVITY RELATIONSHIP;

ERINACEIDAE;

EID: 84856208746 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2011.12.081 Document Type: Article

Times cited : (21)

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