5-arylbenzothiadiazine type compounds as positive allosteric modulators of AMPA/kainate receptors

ACS Medicinal Chemistry Letters

Volumn 3, Issue 1, 2012, Pages 25-29

  Battisti, Umberto M ^a   Jozwiak, Krzysztof ^b   Cannazza, Giuseppe ^a   Puia, Giulia ^a   Stocca, Gabriella ^a   Braghiroli, Daniela ^a   Parenti, Carlo ^a   Brasili, Livio ^a   Carrozzo, Marina M ^c   Citti, Cinzia ^c   Troisi, Luigino ^c  

^a UNIVERSITY OF MODENA AND REGGIO EMILIA   (Italy)

^b MEDICAL UNIVERSITY OF LUBLIN   (Poland)

^c UNIVERSITY OF SALENTO   (Italy)

Author keywords

AMPA modulators; benzothiadiazines; cognitive enhancers; IDRA21

Indexed keywords

5 ARYL 2,3 DIHYDROBENZOTHIADIAZINE; 7 CHLORO 3,4 DIHYDRO 3 METHYL 2H 1,2,4 BENZOTHIADIAZINE 1,1 DIOXIDE; AMPA RECEPTOR; BENZOTHIADIAZINE DERIVATIVE; CYCLOTHIAZIDE; KAINIC ACID RECEPTOR; UNCLASSIFIED DRUG;

ALLOSTERISM; ARTICLE; BLOOD BRAIN BARRIER; BRAIN; CRYSTALLOGRAPHY; ELECTROPHYSIOLOGY; MICRODIALYSIS; MOLECULAR DOCKING; NONHUMAN; PRIORITY JOURNAL;

EID: 84855902830     PISSN: None     EISSN: 19485875     Source Type: Journal    
DOI: 10.1021/ml200184w     Document Type: Article

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