Synthesis, characterization and evaluation of antimicrobial activity of a series of 1,2,4-triazoles

Der Pharma Chemica

Volumn 3, Issue 6, 2011, Pages 32-40

  Agrawal, Rajkumar ^a   Pancholi, S S ^b  

^a Govt of Chhattisgarh ^*  (India)

^b Gujarat Technological University   (India)

Author keywords

1,2,4 triazole; Agar diffusion; Hydrazides; Minimum inhibitory concentration (MIC)

Indexed keywords

1,2,4 TRIAZOLE DERIVATIVE; 4 (5 MERCAPTO 4H 1,2,4 TRIAZOL 3 YL)PHENOL; 5 (2,4 DICHLOROPHENYL) 4H 1,2,4 TRIAZOLE 3 THIOL; 5 (4 NITROPHENYL) 4H 1,2,4 TRIAZOLE 3 THIOL; 5 (PHENOXYMETHYL) 4H 1,2,4 TRIAZOLE 3 THIOL; 5 (PYRIDIN 4 YL) 4H 1,2,4 TRIAZOLE 3 THIOL; 5 [(2,4 DICHLOROPHENOXY)METHYL] 4H 1,2,4 TRIAZOLE 3 THIOL; 5 [(4 CHLOROPHENOXY)METHYL] 4H 1,2,4 TRIAZOLE 3 THIOL; 5 PHENYL 4H 1,2,4 TRIAZOLE 3 THIOL; AMPHOTERICIN B; ANTIBIOTIC AGENT; ANTIFUNGAL AGENT; GENTAMICIN; UNCLASSIFIED DRUG;

ANTIBACTERIAL ACTIVITY; ANTIFUNGAL ACTIVITY; ARTICLE; ASPERGILLUS NIGER; BACTERIAL MEMBRANE; BACTERIAL STRAIN; CANDIDA ALBICANS; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG DETERMINATION; DRUG EFFECT; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS; ESCHERICHIA COLI; FUNGAL CELL; FUNGAL STRAIN; INFRARED SPECTROSCOPY; KLEBSIELLA PNEUMONIAE; MINIMUM INHIBITORY CONCENTRATION; NONHUMAN; PROTEUS VULGARIS; PSEUDOMONAS AERUGINOSA; STAPHYLOCOCCUS; STAPHYLOCOCCUS AUREUS; STAPHYLOCOCCUS COHNII;

EID: 84855297200     PISSN: None     EISSN: 0975413X     Source Type: Journal    
DOI: None     Document Type: Article

References (42)

1. E. Akbas, I. Berber, A. Sener, B. Hasanov, Il Farmaco, 2005, 60, 23-26.
2. C.G. Bonde, N.J. Gaikwad, Bioorg. Med. Chem., 2004, 12, 2151-2161.
3. M.A. Weidner-Wells, C.M. Boggs, B.D. Foleno, J. Melton, K. Bush, R.M. Goldschmidt, D.J. Hlasta, Bioorg. Med. Chem., 2002, 10, 2345-2351.
4. S. Castellano, G. Stefancich, A. Chillotti, G. Poni, Il Farmaco, 2003, 58, 563-568.
5. D.J. Prasad, M. Ashok, P. Karegoudar, B. Poojary, B.S. Holla, N.S. Kumari, Eur. J. Med. Chem., 2009, 44, 551-557.
6. A. Foroumadi, S. Mansouri, Z. Kiani, A. Rahamani, Eur. J. Med. Chem., 2003, 38, 851-854.
7. V.J. Ram, L. Mishra, N.H. Pandey, D.S. Kushwaha, L.A.C. Pieters, A.J. Vlietinck, J. Heterocycl. Chem., 1990, 27, 351-355.
8. N. Ergenc, E. Ilhan, G. Otuk, Pharmazie, 1992, 47, 59-60.
9. V.J. Ram, H.N. Pandey, Chem. Pharm. Bull,. 1974, 22,2778-2783.
10. K.R. Reddy, K. Mogilaiah, B. Swamy, Acta Chim. Hung, 1990, 127, 45-50.
11. S.P. Hiremath, V.N. Sonar, K.R. Sekhar, M.G. Purohit, Indian J. Chem., 1989, 28B, 626-630.
12. B.K. Bhattacharya, V.D. Dirk, G. Hoornaert, S. Sawant, Chem. Abstr., 1985, 102, 24441.
13. N. Kalyoncuoglu, S. Rollas, D. Sur-Altiner, Y. Yegenoglu, A. Ong, Pharmazie, 1992, 47, 796-797.
14. S. Rollas, N. Kalyoncuoglu, D. Sur-Altiner, Y. Yegenoglu, Pharmazie, 1973, 48, 308-309.
15. S.C. Bennur, V.B. Jigajinni, V.V. Badiger, Rev. Roum. Chim. 1976, 21, 757-762.
16. C.S. Andotra, S.K. Sharma, Indian J. Pharm. Sci., 1989, 51, 107.
17. Z. Zhang, X. Feng, L. Chen, Q. Meng, D. Gao, Gaodeng Xuexiao Huaxue Xuebao, 1989, 10, 471.
18. W. Rudnicka, H. Foks, M. Janowiec, Z. Zwolska-Kwiek, Acta Pol. Pharm,. 1986, 43, 523-528.
19. W. Rudnicka, J. Sawlewicz, Acta Pol. Pharm., 1978, 35, 135-142.
20. I. Kuçukguzel, S.G. Kuçukguzel, S. Rollas, M. Kiraz, Bioorg. Med. Chem. Lett., 2001, 11, 1703-1707.
21. M. Kritsanida, A. Mouroutsou, P. Marakos, N. Pouli, S. Papakonstantino-Garoufalias, C. Pannecouque, M. Witvouw, E. De Clercq, Il Farmaco, 2002, 57, 253-257.
22. V. Mathew, J. Keshavayya, V.P. Vaidya, D. Giles, Eur. J. Med. Chem., 2007, 42, 823-840.
23. B. Tozkoparan, N. Gokhan, G. Aktay, E. Yesilada, M. Ertan, Eur. J. Med. Chem., 2000, 35, 743-750.
24. B. Tozkoparan, E. Kupeli, E. Yesilada, M. Ertan, Bioorg. Med. Chem. 2007, 15, 1808-1814.
25. M. Amir, S. Kumar, Acta Pharm., 2007, 57, 31-45.
26. M.S. Langley, S.P. Clissold, Drugs, 1988, 35, 104-122.
27. J.L. Kelley, C.S. Koble, R.G. Davis, E.W. McLean, F.E. Soroko, B.R. Cooper, J. Med.Chem., 1995, 38, 4131-4134.
28. E. Przegalinski, A. Lewandowska, J. Neural Transm. 1979, 46, 303-312.
29. N. Demirbas, R. Ugurluoglu, A. Demirbas, Bioorg. Med. Chem., 2002, 10, 3717-3723.
30. A. Howell, J. Cuzick, M. Baum, A. Buzdar, M. Dowsett, J.F. Forbes, G. Hoctin-Boes, J. Houghton, G.Y. Locker, J.S. Tobias, Lancet, 2005, 365, 60-62.
31. A. Czarnocka-Janowicz, H. Foks, A. Nasal, J. Petrusewicz, B. Damasiewicz,A. Radwanska, R. Kaliszan, Pharmazie, 1991, 46, 109-112.
32. G. Turan-Zitouni, Z.A. Kaplancikli, K. Erol, F.S. Killic, Il Farmaco, 1999, 54, 218-223.
33. M. Ghannoum, L.B. Rice, Clin. Microbiol. Rev., 1999, 12, 501-517.
34. M.Y. Mhasalkar, M.H. Shah, S.T. Nikam, K.G. Ananthanarayana, C.V. Deliwala, J. Med. Chem., 1970, 13, 672-674.
35. J.N. Delgado, W.A. Remers, Text Book of Organic Medicinal Pharmaceutical Chemistry, tenth ed.. J.B., Lippincott Company, Philadelphia, 1998, p. 189.
36. M. Moreno-Manas, Y. Arredondo, R. Pleixats, M. Teixido, M.M. Haga, C. Palacin,J.M. Castello, J.A. Oritizz, J. Heterocycl. Chem., 1992, 29, 1557-1560.
37. L. Czollner, G. Sxilagli, J. Janaky, Arch. Pharm. 1990, 323, 225-229.
38. C.H. Chu, X.W. Sun, L. Sun, Z.Y. Zhang, Z.C. Li, R.A. Liao, J. Chin. Chem. Soc., 1999, 46, 229-235.
39. A. Er-Rhaimini, R. Mornet, Indian J. Heterocycl. Chem., 1992, 29, 1561.
40. H.L. EIbe, K.H. Buechel, W. Brandes, S. Dutzmann, K. Luerssen, Ger. Offen, 1996, 4, 803-883.
41. B. Wolfgan, R. Wolfgan, P. Arbold, S. Bartel, Ger. Offen DE. 4,425,660, Chem.Abstr., 1996, 124, 261076.
42. Y. Liu, A. Gangguly, F. Bennet, Chem. Abstr., 1998 129, 260464.