Release behaviour of propranolol HCl from hydrophilic matrix tablets containing psyllium powder in combination with hydrophilic polymers

AAPS PharmSciTech

Volumn 12, Issue 4, 2011, Pages 1176-1182

  Siahi Shadbad, Mohammad R ^a   Asare Addo, Kofi ^b   Azizian, Kakali ^a   Hassanzadeh, Davoud ^a   Nokhodchi, Ali ^b  

^a TABRIZ UNIVERSITY OF MEDICAL SCIENCES   (Iran)

^b MEDWAY SCHOOL OF PHARMACY   (United Kingdom)

Author keywords

drug release; hydroxypropyl methylcellulose; ionic polymers; psyllium husk; synergistic effect

Indexed keywords

ALGINIC ACID; CELLULOSE; HYDROXYPROPYLMETHYLCELLULOSE; ISPAGULA; POLYMER; PROPRANOLOL; SODIUM CARBOXY METHYL CELLULOSE; UNCLASSIFIED DRUG;

ARTICLE; CONCENTRATION (PARAMETERS); DRUG FORMULATION; DRUG RELEASE; DRUG SOLUBILITY; HYDROPHILICITY; PH MEASUREMENT; PRIORITY JOURNAL; TABLET;

ADRENERGIC BETA-ANTAGONISTS; ALGINATES; CARBOXYMETHYLCELLULOSE SODIUM; CHEMISTRY, PHARMACEUTICAL; DELAYED-ACTION PREPARATIONS; DRUG CARRIERS; DRUG COMPOUNDING; GLUCURONIC ACID; HEXURONIC ACIDS; HYDROGEN-ION CONCENTRATION; HYDROPHOBIC AND HYDROPHILIC INTERACTIONS; KINETICS; METHYLCELLULOSE; POLYMERS; POWDERS; PROPRANOLOL; PSYLLIUM; SOLUBILITY; TABLETS; TECHNOLOGY, PHARMACEUTICAL;

EID: 83555176131     PISSN: None     EISSN: 15309932     Source Type: Journal    
DOI: 10.1208/s12249-011-9687-x     Document Type: Article

References (33)

1. VF Naggar M El-Khawas FA Ismail NA Boraie 1992 Pectin, a possible matrix for oral sustained-release preparations of water-soluble drugs STP Pharma Sci 2 227 34 1:CAS:528:DyaK38XkvFOjuro%3D
2. MC Bonferoni S Rossi M Tamayo JL Pedraz A Dominguez-Gil C Caramella 1993 On the employment of lcarrageenan in a matrix system. I. Sensitivity to dissolution medium and comparison with Na carboxymethylcellulose and xanthan gum J Control Release 26 119 27 10.1016/0168-3659(93)90111-H 1:CAS:528: DyaK3sXmtlersL4%3D (Pubitemid 23226017)
3. T Kristmundsdóttir K Ingvarsdottir G Sæmundsdottir 1995 Chitosan matrix tablets: the influence of excipients on drug release Drug Dev Ind Pharm 21 1591 8 10.3109/03639049509069249
4. P Khullar RK Khar SP Agarwal 1998 Evaluation of guar gum in the preparation of sustained-release matrix tablets Drug Dev Ind Pharm 24 1095 9 9876566 10.3109/03639049809089955 1:CAS:528:DyaK1cXmsVamsLo%3D (Pubitemid 28460250)
5. L Vervoort G Van den Mooter P Augustijns R Kinget 1998 Inulin hydrogels. I. Dynamic and equilibrium swelling properties Int J Pharm 172 127 35 10.1016/S0378-5173(98)00200-2 1:CAS:528:DyaK1cXls1equ70%3D (Pubitemid 28430250)
6. A Nokhodchi H Nazemiyeh A Khodaparast T Sorkh-Shahan H Valizadeh JL Ford 2008 An in vitro evaluation of fenugreek mucilage as a potential excipient for oral controlled-release matrix tablet Drug Dev Ind Pharm 34 323 9 18363148 10.1080/03639040701662594 1:CAS:528:DC%2BD1cXjs1Wgsbc%3D (Pubitemid 351431205)
7. P Colombo U Conte C Caramella A Gazzaniga A La Manna 1985 Compressed polymeric mini-matrices for drug release control J Control Release 1 283 9 10.1016/0168-3659(85)90004-5 1:CAS:528:DyaL2MXkvFaktbg%3D (Pubitemid 15057115)
8. P Colombo R Bettini G Massimo PL Catellani P Santi NA Peppas 1995 Drug diffusion front movement is important in drug release control from swellable matrix tablets J Pharm Sci 84 991 7 7500286 10.1002/jps.2600840816 1:CAS:528:DyaK2MXmvVeisrY%3D
9. JE Mockel BC Lippold 1993 Zero-order drug release from hydrocolloid matrices Pharm Res 10 1066 70 8378249 10.1023/A:1018931210396 1:STN:280:DyaK3szptFartg%3D%3D (Pubitemid 23211433)
10. AS Hussain RD Johnson P Shivanand MA Zoglio 1994 Effects of blending a nonionic and an anionic cellulose ether polymer on drug release from hydrophilic matrix capsules Drug Dev Ind Pharm 20 2645 57 10.3109/03639049409042668 1:CAS:528:DyaK2cXlvVOjt70%3D (Pubitemid 24288826)
11. DL Munday PJ Cox 2000 Compressed xanthan and karaya gum matrices: hydration, erosion and drug release mechanism Int J Pharm 203 179 92 10967440 10.1016/S0378-5173(00)00444-0 1:CAS:528:DC%2BD3cXmtValsLs%3D (Pubitemid 30627638)
12. TD Reynolds SH Gehrke AS Hussain LS Shenouda 1998 Polymer erosion and drug release characterisation of hydroxypropylmethylcellulose matrices J Pharm Sci 87 1115 23 9724564 10.1021/js980004q 1:CAS:528:DyaK1cXltV2rt7Y%3D (Pubitemid 28452113)
13. F Ughini IF Andreazza JLMS Ganter TMB Bresolin 2004 Evaluation of xanthan and highly substituted galactomannan from M. scabrella as a sustained release matrix Int J Pharm 271 197 205 15129986 10.1016/j.ijpharm.2003.11.011 1:CAS:528:DC%2BD2cXhtVekurc%3D (Pubitemid 38210097)
14. M Nakano A Ogata 1984 Examination of natural gums as matrices for sustained release of theophylline Chem Pharm Bull 32 782 5 6733818 1:CAS:528:DyaL2cXitFGgurc%3D (Pubitemid 14125926)
15. JW McRorie BP Daggy JG Morel PS Diersing PB Miner M Robinson 1998 Psyllium is superior to docusate sodium for treatment of chronic conspitation Aliment Pharmacol Ther 12 491 7 9663731 10.1046/j.1365-2036.1998.00336.x 1:CAS:528:DyaK1cXjslGksrs%3D (Pubitemid 28247523)
16. D Belknap LJ Davidson CR Smith 1997 The effects of psyllium hydrophilic mucilliod on diarrhea in enterally fed patients Heart Lung 26 229 37 9176691 10.1016/S0147-9563(97)90060-1 1:STN:280:DyaK2szhvFyjsQ%3D%3D (Pubitemid 27232968)
17. M Juarranz ME Calle-Puron A Gonzalez-Navarro E Regidor-Poyatos T Soriano D Martinez-Hernandez VD Rojas VF Guinee 2002 Physical exercise, use of Plantago ovata and aspirin, and reduced risk of colon cancer Eur J Cancer Prev 11 465 72 12394244 10.1097/00008469-200210000-00009 1:STN:280:DC%2BD38njsV2lsg%3D%3D (Pubitemid 35265848)
18. DJ Jenkinz CW Kendall M Axelsen LAS Augustin V Vuksa 2000 Viscous and nonviscous fibres, nonabsorbable and low glycaemic index carbohydrates, blood lipids and coronary heart disease Curr Opin Lippidol 11 49 56 10.1097/00041433-200002000-00008 (Pubitemid 30148198)
19. B Singh S Kumar N Chauhan 2008 Radiation crosslinked psyllium and polyacrylic acid based hydrogels for use in colon specific drug delivery Carbohydr Polym 73 445 6
20. M Chavanpatil P Jain S Chaudhari R Shear P Vavia 2006 Novel sustained release, swellable and bioadhesive gastroretentive drug delivery system for ofloxacin Int J Pharm 316 86 92 16567072 10.1016/j.ijpharm.2006.02.038 1:CAS:528:DC%2BD28XkvVWrtL0%3D (Pubitemid 43765689)
21. M Gohel M Patel A Amin 2003 Development of modified release diltiazem HCl tablets using composite index to identify optimal formulation Drug Dev Ind Pharm 29 565 74 12779286 10.1081/DDC-120018645 1:CAS:528:DC%2BD3sXkt1Ont7c%3D (Pubitemid 36597397)
22. B Kaith K Kumar 2008 In vacuum synthesis of psyllium and acrylic acid based hydrogels for selective water absorption from different oil-water emulsions Desalination 229 331 41 10.1016/j.desal.2007.08.020 1:CAS:528:DC%2BD1cXosVajtLs%3D (Pubitemid 351940562)
23. Korsemeyer RW, Peppas NA. Macromolecular and modelling aspects of swelling-controlled systems. In: Mansdorf SZ, Roseman TJ, editors. Controlled release delivery systems. New York: Marcel Dekker; 1983. p. 77.
24. J Siepmann H Kranz R Bodmeier NA Peppas 1999 HPMC-matrices for controlled drug delivery: a new model combining diffusion, swelling, and dissolution mechanisms and predicting the release kinetics Pharm Res 16 1748 56 10571282 10.1023/A:1018914301328 1:CAS:528:DyaK1MXnt1GgsLo%3D (Pubitemid 29530409)
25. PL Ritger NA Peppas 1987 A simple equation for description of solute release. I. Fickian and non-Fickian release from non-swellable devices in the form of slabs, spheres, cylinders or discs J Control Release 5 23 36 10.1016/0168-3659(87)90034-4 1:CAS:528:DyaL2sXkvVeku7o%3D (Pubitemid 17106643)
26. FO Costa JJS Sousa AACC Pais SJ Formosinho 2003 Comparison of dissolution profiles of ibuprofen pellets J Control Rel 89 199 212 10.1016/S0168-3659(03) 00033-6 1:CAS:528:DC%2BD3sXjtVegur4%3D (Pubitemid 36507015)
27. KA Khan 1975 Concept of dissolution efficiency J Pharm Pharmacol 27 48 9 235616 10.1111/j.2042-7158.1975.tb09378.x 1:CAS:528:DyaE2MXhsVCru7o%3D
28. AK Bajpai A Mishra 2004 Ionizable interpenetrating polymer networks of carboxymethyl cellulose and polyacrylic acid: evaluation of water uptake J Appl Polym Sci 93 5 2054 65 10.1002/app.20674 1:CAS:528:DC%2BD2cXmtlGiuro%3D (Pubitemid 39075277)
29. D Cohn M Aronhime B Azdo 1992 Poly(urethane)-crosslinked poly(HEMA) hydrogels J Macromol Sci Pure Appl Chem A29 10 841 51 1:CAS:528: DyaK38Xlslyht7k%3D (Pubitemid 23589570)
30. AK Bajpai A Giri 2003 Water sorption behaviour of highly swelling (carboxy methylcellulose-g-polyacrylamide) hydrogels and release of potassium nitrate as agrochemical Carbohydr Polym 53 271 2790 10.1016/S0144-8617(03)00071- 7 1:CAS:528:DC%2BD3sXks1Wgt78%3D
31. KV Ranga Rao P Padmalatha Devi P Buri 1990 Influence of molecular size and water solubility of the solute on its release from swelling and erosion controlled polymeric matrices J Control Release 12 133 41 10.1016/0168-3659(90) 90089-C (Pubitemid 20123878)
32. JL Ford MH Rubinstein F McCaul JE Hogan PJ Edgar 1987 Importance of drug type, tablet shape and added diluents on drug release kinetics from hydroxypropylmethylcellulose matrix tablets Int J Pharm 40 223 34 10.1016/0378-5173(87)90172-4 1:CAS:528:DyaL1cXktl2mtg%3D%3D (Pubitemid 18025827)
33. SK Baveja KV Ranga Rao 1986 Sustained release tablet formulations of centperazine Int J Pharm 31 169 74 10.1016/0378-5173(86)90228-0 1:CAS:528:DyaL1cXotF2gsg%3D%3D (Pubitemid 16057429)