Formulation and evaluation of fenoprofen calcium compressed coated tablets for colon specific drug delivery

Asian Journal of Pharmaceutical and Clinical Research

Volumn 4, Issue SUPPL. 2, 2011, Pages 88-95

  Potu, Apparao ^a   Pasunooti, Sandeep ^a   Veerareddy, Prabhakarreddy ^a   Burra, Shashidher ^a  

^a ST PETER'S INSTITUTE OF PHARMACEUTICAL SCIENCES   (India)

Author keywords

Colon specific drug delivery; Compression coating; Guar gum; Rat caecal contents caecal contents

Indexed keywords

FENOPROFEN CALCIUM; GUAR GUM; HYDROXYPROPYLMETHYLCELLULOSE;

ABDOMINAL RADIOGRAPHY; ADULT; ANIMAL TISSUE; ARTICLE; CONTROLLED STUDY; DRUG COATING; DRUG DELIVERY SYSTEM; DRUG DETERMINATION; DRUG DISTRIBUTION; DRUG MONITORING; DRUG RELEASE; DRUG SOLUBILITY; EX VIVO STUDY; HUMAN; HUMAN EXPERIMENT; INFRARED SPECTROSCOPY; NONHUMAN; NORMAL HUMAN; PH MEASUREMENT; PROCESS OPTIMIZATION; RAT; TABLET COMPRESSION; TABLET DISINTEGRATION TIME; TABLET FORMULATION;

EID: 83455249893     PISSN: 09742441     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

References (44)

1. Antonin, K.H., Rak, R., Beick, P.R., Schenker, U., Hastewell, J., Fox, R., Mackay, M., The absorption of human calcitonin from the transverse colon of man. Int. J. Pharm.(1996), 130, 33-39.
2. Tozaki, H., Komoike, J., Tada, C., Maruyama, T., Terabe, A., Suzuki, T., Yamamoto, A., Muranishi, S. Chitosan capsules for colon-specific drug delivery: Improvement of insulin absorption from the rat colon. J. Pharm. Sci. (1997), 86, 1016-1021.
3. Davis S, Overcoming barriers to the oral administration of peptide drugs. Trends Pharm Sci, (1990), 11: 353-355.
4. Van den Mooter G. V., Kinget R, Oral colon-specific drug delivery: a review. DrugDeliv, (1995), 2: 81-93.
5. Singh BN, Kim, KH. In: Swarbrick J, Boylan JC (Eds.), Encyclopedia of Pharmaceutical Technology, New York, Marcel Dekker, Inc., (2002), 886-909.
6. Ashford M, Fell J T. Targeting drugs to the colon: delivery systems for oral administration. JDrug Target, (1994), 2: 241-258.
7. Ashford, M., Fell, J., Attwood, D., Sharma, H., Woodhead, P. An evaluation of pectin as a carrier for drug targeting to the colon. J. Control. Release. (1993b), 26, 213-220.
8. Fukui E, Miyamura N, Uemura K, Kobayashi M. Preparation of enteric coated timed release press-coated tablets and evaluation of their function by in vitro and in vivo tests for colon targeting. Int J Pharm (2000) 204:7-15.
9. Ishibashi T, Hatano H, Kobayashi M, Mizobe M, Yoshino H. Design and evaluation of a new capsule-type dosage form for colon-targeted delivery of drugs. Int J Pharm (1998) 168:31-40.
10. Tomlin J, Read NW. The relation between bacterial degradation of viscous polysaccharides and stool output in human beings. Brit J Nutr. (1988), 60:476.
11. Krishnaiah YSR, Satyanarayana S. Colonspecific drug delivery systems. In: Jain NK, ed. Advances in Controlled and Novel Drug Delivery. New Delhi, India: CBS Publishers and Distributors (2000),89-119.
12. Lee VHL, Mukherjee SK. Drug Delivery:Oral Colon-Specific. Ency Pharm Tech. Dekker Encyclopedia: (2002),871-885.
13. Rao SSC, Read NW, Bruce C, Brown C, Holdsworth CD. Studies on the mechanismof bowel disturbance in ulcerative colitis. Gastroenterol.(1987),93: 934-940
14. Friend, D.R., Philips, S., Tozer, T.N. Colon-specific drug delivery from a glucoside prodrug in the guinea pig.Efficacy study. J. Control. Release.(1991), 15, 47-54.
15. Cummings JH, Southgate DA, Branch WJ, Wiggins HS, Houston H, Jenkins DJ, et al. The digestion of pectin in human gut and its effect on calcium absorption and large bowel function. Br J Nutr (1979) 41: 477-85.
16. Sinha VR, Kumria R. Polysaccharides in colon specific drug delivery. Int J Pharm (2001) 224:19-38.
17. Munjeri, O., Collett, J.H., Fell, J.T. Hydrogel beads based on amidated pectins for colon-specific drug delivery:the role of chitosan in modifying drug release. J. Control. Release. (1997) 46, 273-278.
18. Englyst HN, MacFarlane GT. Breakdown of resistant and readily digestible starch of human gut bacteria. J Sci Food Agric (1986)37:699-706.
19. Chaurasia M, Chourasia MK, Jain NK, Jain A, Soni V, Gupta Y, et al. Cross-linked guar gum microspheres: A viable approach for improved delivery of anticancer drugs for the treatment of colorectal cancer. AAPS Pharm Sci Tech (2006) 7:74.
20. Chourasia MK, Jain SK. Design and development of multiparticulate system for targeted drug delivery to colon. J Drug Deliv. (2004)11:201-7.
21. Chourasia MK, Jain SK. Potential of guar gum microspheres for target specific drug release to colon. J Drug Target.(2004)2: 1-8.
22. Cummings JH, Milojevic S, Harding M, Coward WA, Gibson GR, Botham RL, et al. In-vivo studies of amylose and ethylcellulose coated 13 C glucose microspheres as a model for drug delivery to the colon. J Control Release (1996)40:123-31.
23. Jain A, Gupta Y, Jain SK. Perspectives of biodegradable natural polysaccharides for Site-Specific drug delivery to the colon. J Pharm Pharmaceut Sci (2007)10:86-128.
24. Krogars K, Heinamaki J, Vesalahti J, Marvola M. Antikainen O, Yliruusi J, et al. Extrusion spheronization of pH-sensitive polymeric matrix pellets for possible colonic drug delivery. Int J Pharm (2000)199:187-94.
25. Rodriguez M, Vila-Jato JL, Torres D. Design of a new multiparticulate system for potential site-specific and controlled drug delivery to the colonic region. J Control Rel (1998); 55:67-77.
26. Jain SK, Jain A, Gupta Y, Ahirwar M. Design and development of hydrogel beads for targeted drug delivery to Colon. AAPS Pharm Sci Tech (2007); 8:1-8.
27. Takeuchi H, Yasuji T, Yamamoto H, Kawashima Y. Spray-dried lactose composite particles containing an ion complex of alginate-chitosan for designing a dry coated tablet having a time-controlled releasing function. Pharm Res. (2000); 17:94-99.
28. Wong, D., Larrabee, S., Clifford, K., Tremblay, J., Friend, D.R., USP dissolution apparatus III (reciprocating cylinder) for screening of guar-based colonic delivery formulations. J. Control. Release. (1997), 47, 173-179.
29. Kopecek, J., Kopecekova, P., Bronsted, H., Rathi, R., Rihova, B., Yeh, P.Y., Ikesue, K. Polymers for colon specific drug delivery. J. Control. Release,(1992). 19, 121-130.
30. Van den Mooter, G., Samyn, C., Kinget, R., Azo polymers for colon-specific drug delivery. II. Influence of the type of azo polymer on the degradation by intestinal microflora. Int. J. Pharm. (1993), 97, 133-135
31. Kalala, W., Kinget, R., Van den Mooter, G., Samyn, C., Colonic drug targeting: in vitro release of ibuprofen from capsules coated with poly (ether-ester) azopolymers. Int. J.Pharm. (1996), 139,187-195.
32. Krishnaiah, Y.S.R S. Satyanarayana, Y.V. Rama Prasad a, S. Narasimha Rao Evaluation of guar gum as a compression coat for drug targeting to colon. International Journal of Pharmaceutics. 171 (1998) 137-146.
33. Krishnaiah, Y.S.R S. Satyanarayana, Y.V. Rama Prasad a, S. Narasimha Rao bEvaluation of guar gum as a compression coat for drug targeting to colon. International Journal of Pharmaceutics 171 (1998) 137-146
34. Davis, S.S., Hardy, J.G., Taylor, M.J., Stockwell, A., Whalley, D.R., Wilson, C.G.,. The in vivo evaluation of an osmotic device (Osmet) using g-scintigraphy. J. Pharm.Pharmacol. (1984), 36, 740-742.
35. Van den Mooter, G., Kinget, R. Oral colon-specific drug delivery: A review. Drug Delivery. (1995) 2, 81-93.
36. Rubinstein, A., Nakar, D., Sintov, A. Chondroitin sulfate: A potential biodegradable carrier for colon-specific drug delivery. Int. J. Pharm.(1992b), 84, 141-150.
37. Vervoort, L., Kinget, R. In vitro degradation by colonic bacteria of inulinHP incorporated in Eudragit RS films. Int. J. Pharm. (1996), 129, 185-190.
38. Rubinstein, A., Radai, R., Ezra, M., Pathak, S., Rokea, J.S. In vitro evaluation of calcium pectinate: A potential colon-specific drug delivery carrier. Pharm. Res.(1993) 10, 258-263.
39. Rubinstein, A., Nakar, D., Sintov, A. Colonic drug delivery: Enhanced release of indomethacin from crosslinked chondroitin matrix in rat caecal content. Pharm.Res. (1992)9, 276-278.
40. Wakerly, Z., Fell, J.T., Attwood, D., Parkins, D.A. In vitro evaluation of pectin-based colonic drug delivery systems. Int. J. Pharm. (1996a) 129, 73-77.
41. Wakerly, Z., Fell, J.T., Attwood, D., Parkins, D.A. Pectin:ethyl cellulose film coating formulations for colonic drug delivery. Pharm. Res. (1996b)13, 1210-1212.
42. Rama Prasad, Y.V., Krishnaiah, Y.S.R., Satyanarayana, S., In vitro evaluation of guar gum as a carrier for colon-specific drug delivery. J. Control. Release, (1998)51, 281-287.
43. McLeod, A.D., Friend, D.R., Tozer, T.N.,. Glucocorticoid-dextran conjugates as potential prodrugs for colonspecificdelivery: Hydrolysis in rat gastrointestinal tract contents. J. Pharm. Sci. (1994), 83, 1284-1288.
44. Khosla, R., Davis, S.S.,.Gastric emptying time and small and large bowel transit of non-disintegrating tablets in fasted subjects. Int. J. Pharm. (1989)52, 1-10.