Kinase inhibitor selectivity profiling using differential scanning fluorimetry

Methods in Molecular Biology

Volumn 795, Issue , 2012, Pages 109-118

  Fedorov, Oleg ^a   Niesen, Frank H ^a   Knapp, Stefan ^a  

^a UNIVERSITY OF OXFORD   (United Kingdom)

Author keywords

Compound screening; Differential scanning fluorimetry; Inhibitor selectivity; Kinase; Protein stability

Indexed keywords

LIGAND; PROTEIN KINASE INHIBITOR;

ARTICLE; DRUG EFFECT; ENZYME ASSAY; ENZYME SPECIFICITY; FLUOROMETRY; HIGH THROUGHPUT SCREENING; METHODOLOGY; PROTEIN BINDING; PROTEIN STABILITY;

ENZYME ASSAYS; FLUOROMETRY; HIGH-THROUGHPUT SCREENING ASSAYS; LIGANDS; PROTEIN BINDING; PROTEIN KINASE INHIBITORS; PROTEIN STABILITY; SUBSTRATE SPECIFICITY;

EID: 80555135984     PISSN: 10643745     EISSN: None     Source Type: Book Series    
DOI: 10.1007/978-1-61779-337-0_7     Document Type: Article

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