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ChemMedChem

Volumn 6, Issue 11, 2011, Pages 1971-1976

Discovery of α,β- and α,γ-diamino acid scaffolds for the inhibition of M1 family aminopeptidases

(4) Gumpena, Rajesh a Kishor, Chandan a Ganji, Roopa Jones a Addlagatta, Anthony a

a INDIAN INSTITUTE OF CHEMICAL TECHNOLOGY (India)

Author keywords

Aminopeptidases; Drug discovery; Modeling; Structural biology

Indexed keywords

2,3 DIAMINOPROPIONIC ACID; 2,4 DIAMINOBUTYRIC ACID; AMINOPEPTIDASE; AMINOPEPTIDASE INHIBITOR; BESTATIN; BETA ALANINE; DIAMINO ACID; ENZYME INHIBITOR; LYSINE; ORNITHINE; UNCLASSIFIED DRUG;

ARTICLE; DRUG ACTIVITY; DRUG EFFICACY; DRUG PROTEIN BINDING; DRUG SPECIFICITY; DRUG SYNTHESIS; ENZYME INHIBITION; ENZYME INHIBITOR INTERACTION; HUMAN; NONHUMAN; PRIORITY JOURNAL;

AMINO ACIDS, DIAMINO; AMINOBUTYRIC ACIDS; AMINOPEPTIDASES; BACTERIAL PROTEINS; BETA-ALANINE; BINDING SITES; CATALYTIC DOMAIN; CRYSTALLOGRAPHY, X-RAY; DRUG DESIGN; HUMANS; METHIONINE; MODELS, MOLECULAR; PROTEASE INHIBITORS; SERINE;

EID: 80054980238 PISSN: 18607179 EISSN: 18607187 Source Type: Journal
DOI: 10.1002/cmdc.201100298 Document Type: Article

Times cited : (14)

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