Erratum: Synthesis and evaluation of anti-inflammatory, analgesic, ulcerogenic and lipid peroxidation properties of new 2-(4-isobutylphenyl) propanoic acid derivatives (Journal of Enzyme Inhibition and Medicinal Chemistry (2012) 27: 1 (110-116) DOI: 10.3109/14756366.2011.578743);Synthesis and evaluation of anti-inflammatory, analgesic, ulcerogenic and lipid peroxidation properties of new 2-(4-isobutylphenyl)propanoic acid derivatives

Journal of Enzyme Inhibition and Medicinal Chemistry

Volumn 27, Issue 1, 2012, Pages 110-116

  Raval, Jignesh Priyakant ^a   Gandhi, Ankur Navinchandra ^a   Akhaja, Tarunkumar Nanjibhai ^a   Myangar, Kruti Navinbhai ^a   Patel, Nilesh Hasmukhbhai ^b  

^a Ashok & Rita Patel Institute of Integrated Study and Research in Biotechnology and Allied Sciences   (India)

^b EMCURE Pharmaceuticals USA INC   (United States)

Author keywords

2 (4 isobutylphenyl)propanoic acid; Analgesic; Anti inflammatory; Lipid peroxidation activities; Thiadiazolo 3; 2 a 1; 3; 5 triazine 5 thione; Ulcerogenic

Indexed keywords

2 (4 ISOBUTYLPHENYL)PROPANOIC ACID DERIVATIVE; 2 [1 (4 ISOBUTYLPHENYL)ETHYL] 7 (4 NITRO PHENYL) 6,7 DIHYDRO 5H [1,3,4]THIADIAZOLO[3,2 A][1,3,5]TRIAZINE 5 THIONE; 2 [1 (4 ISOBUTYLPHENYL)ETHYL] 7 PHENYL 6,7 DIHYDRO 5H [1,3,4]THIADIAZOLO[3,2 A][1,3,5]TRIAZINE 5 THIONE; ANALGESIC AGENT; ANTIINFLAMMATORY AGENT; IBUPROFEN; MALONALDEHYDE; N (4 CHLOROBENZYLIDENE) 5 [1 (4 ISOBUTYLPHENYL)ETHYL] 1,3,4 THIADIAZOL 2 AMINE; N (4 FLUORO BENZYLIDENE) 5 [1 (4 ISOBUTYLPHENYL)ETHYL] 1,3,4 THIADIAZOL 2 AMINE; N BENZYLIDINE 5 [1 (4 ISOBUTYLPHENYL)ETHYL] 1,3,4 THIADIAZOL 2 AMINE; PROPIONIC ACID DERIVATIVE; UNCLASSIFIED DRUG;

ANALGESIC ACTIVITY; ANIMAL EXPERIMENT; ANIMAL TISSUE; ANTIINFLAMMATORY ACTIVITY; ARTICLE; CARBON NUCLEAR MAGNETIC RESONANCE; CONTROLLED STUDY; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS; INFRARED SPECTROSCOPY; LIPID PEROXIDATION; MALE; MOUSE; NONHUMAN; PAW EDEMA; PRIORITY JOURNAL; PROTON NUCLEAR MAGNETIC RESONANCE; RAT; STOMACH MUCOSA; ULCEROGENESIS;

EID: 80054897224     PISSN: 14756366     EISSN: 14756374     Source Type: Journal    
DOI: 10.3109/14756366.2012.682431     Document Type: Erratum

References (20)

1. Kimmey MB. NSAID, ulcers, and prostaglandins. J Rheumatol Suppl 1992;36:68-73.
2. Smith CJ, Zhang Y, Koboldt CM, Muhammad J, Zweifel BS, Shaffer A et al. Pharmacological analysis of cyclooxygenase-1 in inflammation. Proc Natl Acad Sci USA 1998;95:13313-13318. (Pubitemid 28509568)
3. Hawkey C, Laine L, Simon T, Beaulieu A, Maldonado-Cocco J, Acevedo E et al. Comparison of the effect of rofecoxib (a cyclooxygenase 2 inhibitor), ibuprofen, and placebo on the gastroduodenal mucosa of patients with osteoarthritis: a randomized, double-blind, placebo-controlled trial. The Rofecoxib Osteoarthritis Endoscopy Multinational Study Group. Arthritis Rheum 2000;43:370-377. (Pubitemid 30395746)
4. Warner TD, Giuliano F, Vojnovic I, Bukasa A, Mitchell JA, Vane JR. Nonsteroid drug selectivities for cyclo-oxygenase-1 rather than cyclo-oxygenase-2 are associated with human gastrointestinal toxicity: a full in vitro analysis. Proc Natl Acad Sci USA 1999;96:7563-7568. (Pubitemid 29299702)
5. Lanza FL. A guideline for the treatment and prevention of NSAIDinduced ulcers. Members of the Ad Hoc Committee on Practice Parameters of the American College of Gastroenterology. Am J Gastroenterol 1998;93:2037-2046. (Pubitemid 29076848)
6. Kalgutkar AS, Marnett AB, Crews BC, Remmel RP, Marnett LJ. Ester and amide derivatives of the nonsteroidal antiinflammatory drug, indomethacin, as selective cyclooxygenase-2 inhibitors. J Med Chem 2000;43:2860-2870. (Pubitemid 30599644)
7. Duflos M, Nourrisson MR, Brelet J, Courant J, LeBaut G, Grimaud N et al. N-pyridinyl-indole-3-(alkyl)carboxamides and derivatives as potential systemic and topical inflammation inhibitors. Eur J Med Chem 2001;36:545-553. (Pubitemid 32781718)
8. Palaska E, Sahin G, Kelicen P, Durlu NT, Altinok G. Synthesis and anti-inflammatory activity of 1-acylthiosemicarbazides, 1,3,4-oxadiazoles, 1,3,4-thiadiazoles and 1,2,4-triazole-3-thiones. Farmaco 2002;57:101-107. (Pubitemid 34175107)
9. Sainy J, Mishra GP, Sharma R, Chaturvedi SC. 2-Amino-5-sulfanyl-1,3,4- thiadiazoles: a novel series of anti-inflammatory and analgesic agents. Pharm Chem Jr 2009; 43:19-24.
10. Geronikaki A, Hadjipavlou-Litina D, Amourgianou M. Novel thiazolyl, thiazolinyl and benzothiazolyl Schiff bases as possible lipoxygenase's inhibitors and anti-inflammatory agents. Farmaco 2003;58:489-495. (Pubitemid 36765349)
11. Kim SH. Anti-inflammatory 7-phenyl pyrazolo-[1,5a]-1,3,5-triazine derivatives. 1987; EP0207651 A2. Appl. No. EP19860304353.
12. Brown DE. Analgesic 6-acylaminotetrahydro-1,3,5-triazine-2,4-dione derivatives, pharmaceutical compositions thereof, and process for their manufacture. 1982; EP0005911 B1. Appl. No. EP19790300756.
13. Raval JP, Desai KR. Synthesis and antimicrobial activity of new triazolopyridinyl phenothiazines. Arkivoc 2005;xiii:21-28. (Pubitemid 40397771)
14. Raval JP, Desai KG, Desai KR. Neat reaction technology for the synthesis of 4-oxothiazolidines derived from 2-SH-Benzothiazole and antimicrobial screening of some synthesized 4-thiazolidinones. J Iran Chem Soc 2006; 3:233-241.
15. Raval JP, Desai JT, Desai CK, Desai KR. A comparative study of microwave assisted and conventional synthesis of 2,3-dihydro-2-aryl-4-[4-(2-oxo-2H- chromen-3-yl)-1,3-thiazol-2-ylamino]-1,5-benzothiazepines and its antimicrobial activity. Arkivoc 2008; xii:233-244.
16. Rahman MA, Omar FA, Mahfouz NM. Design, synthesis and antiinflammatory activity of some 1,3,4-oxadiazole derivatives. Eur J Med Chem 1996; 31:819-825. (Pubitemid 26341447)
17. Winter CA, Risley EA, Nuss GW. Carrageenin-induced edema in hind paw of the rat as an assay for antiiflammatory drugs. Proc Soc Exp Biol Med 1962;111:544-547.
18. Siegmund E, Cadmus R, Lu G. A method for evaluating both non-narcotic and narcotic analgesics. Proc Soc Exp Biol Med 1957;95:729-731.
19. Cioli V, Putzolu S, Rossi V, Scorza Barcellona P, Corradino C. The role of direct tissue contact in the production of gastrointestinal ulcers by anti-inflammatory drugs in rats. Toxicol Appl Pharmacol 1979;50:283-289. (Pubitemid 10233388)
20. Ohkawa H, Ohishi N, Yagi K. Assay for lipid peroxides in animal tissues by thiobarbituric acid reaction. Anal Biochem 1979;95:351-358. (Pubitemid 9194347)