Isolation of modulators of the liver-specific Organic Anion-Transporting Polypeptides (OATPs) 1B1 and 1B3 from Rollinia emarginata Schlecht (Annonaceae)

Journal of Pharmacology and Experimental Therapeutics

Volumn 339, Issue 2, 2011, Pages 624-632

  Roth, Megan ^a   Araya, Juan J ^b   Timmermann, Barbara N ^b   Hagenbuch, Bruno ^a,c  

^a UNIVERSITY OF KANSAS SCHOOL OF MEDICINE   (United States)

^b UNIVERSITY OF KANSAS   (United States)

^c UNIVERSITY OF KANSAS CANCER CENTER   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

8 TRANS 4 COUMAROYLOXY ALPHA TERPINEOL; ESTRADIOL 17 GLUCURONIDE; ESTRONE SULFATE; OLEANOLIC ACID; ORGANIC ANION TRANSPORTER 1; ORGANIC ANION TRANSPORTING POLYPEPTIDE 1B1; ORGANIC ANION TRANSPORTING POLYPEPTIDE 1B3; PLANT EXTRACT; QUERCETIN 3 O ALPHA LEVO ARABINOPYRANOSYL (1-2) ALPHA LEVO RHAMNOPYRANOSIDE; RIFAMPICIN; ROLLINIA EMARGINATA EXTRACT; TERPINEOL; UNCLASSIFIED DRUG; URSOLIC ACID;

ANIMAL CELL; ANIMAL TISSUE; ANNONACEAE; ARTICLE; BINDING AFFINITY; CONTROLLED STUDY; DRUG ACTIVITY; DRUG BINDING; DRUG EFFICACY; DRUG ISOLATION; DRUG SCREENING; DRUG TRANSPORT; FEMALE; LIVER CELL; NONHUMAN; PRIORITY JOURNAL; ROLLINIA EMARGINATA; TRANSPORT KINETICS;

ANIMALS; CHO CELLS; CRICETINAE; CRICETULUS; DRUG DISCOVERY; ESTRADIOL; ESTRONE; HEPATOCYTES; KINETICS; LIVER; MOLECULAR TARGETED THERAPY; OLEANOLIC ACID; ORGANIC ANION TRANSPORTERS; ORGANIC ANION TRANSPORTERS, SODIUM-INDEPENDENT; PLANT BARK; PLANT EXTRACTS; ROLLINIA; TERPENES; TRITERPENES;

EID: 80054778404     PISSN: 00223565     EISSN: 15210103     Source Type: Journal    
DOI: 10.1124/jpet.111.184564     Document Type: Article

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