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Volumn 130, Issue 1-2, 2011, Pages 361-366

Stabilized amorphous glibenclamide nanoparticles by high-gravity technique

Author keywords

Amorphous materials; Nanostructures; Precipitation; Recrystallisation

Indexed keywords

ANTI-SOLVENTS; CRYSTALLINE FORM; DISSOLUTION RATES; DISSOLUTION TESTS; FOURIER TRANSFORM INFRARED; GLIBENCLAMIDE; HIGH-GRAVITY; MEAN SIZE; NARROW DISTRIBUTION; OPERATING VARIABLES; PHYSICAL STABILITY; RECRYSTALLISATION;

EID: 80052604859     PISSN: 02540584     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.matchemphys.2011.06.049     Document Type: Article
Times cited : (27)

References (32)
  • 1
    • 2642572791 scopus 로고    scopus 로고
    • Glibenclamide transdermal patches: Physicochemical, pharmacodynamic, and pharmacokinetic evaluations
    • DOI 10.1002/jps.20058
    • S. Mutalik, and N. Udupa Glibenclamide transdermal patches: physicochemical, pharmacodynamic, and pharmacokinetic evaluations J. Pharm. Sci. 93 6 2004 1577 1594 (Pubitemid 38725029)
    • (2004) Journal of Pharmaceutical Sciences , vol.93 , Issue.6 , pp. 1577-1594
    • Mutalik, S.1    Udupa, N.2
  • 2
    • 0020967084 scopus 로고
    • Pharmacokinetics and effects of glibenclamide in two formulations, HB 419 and HB 420, in type 2 diabetes
    • H.J. Arnqvist, B.E. Karlberg, and A. Melander Pharmacokinetics and effects of glibenclamide in two formulations, HB 419 and HB 420, in type 2 diabetes Ann. Clin. Res. 37 1983 21 25 (Pubitemid 14124718)
    • (1983) Annals of Clinical Research , vol.15 , Issue.SUPPL. 37 , pp. 21-25
    • Arnqvist, H.J.1    Karlberg, B.E.2    Melander, A.3
  • 3
    • 0022909293 scopus 로고
    • Correlations between in vitro dissolution, in vivo bioavailability and hypoglycaemic effect of oral glibenclamide
    • DOI 10.1007/BF00606655
    • J.B. Chalk, M. Patterson, M.T. Smith, and M.J. Eadie Correlation between in vitro dissolution, in vivo bioavailability and hypoglycaemic effect of oral glibenclamide Eur. J. Clin. Pharmacol. 31 1986 177 182 (Pubitemid 17014586)
    • (1986) European Journal of Clinical Pharmacology , vol.31 , Issue.2 , pp. 177-182
    • Chalk, J.B.1    Patterson, M.2    Smith, M.T.3    Eadie, M.J.4
  • 4
    • 10644275105 scopus 로고    scopus 로고
    • Enhancement of dissolution rate of poorly-soluble active ingredients by supercritical fluid processes: Part I: Micronization of neat particles
    • DOI 10.1016/j.ijpharm.2004.09.007, PII S0378517304005411
    • M. Perrut, J. Jung, and F. Leboeuf Enhancement of dissolution rate of poorly-soluble active ingredients by supercritical fluid processes. Part I: micronization of neat particles Int. J. Pharm. 288 2005 3 10 (Pubitemid 39656449)
    • (2005) International Journal of Pharmaceutics , vol.288 , Issue.1 , pp. 3-10
    • Perrut, M.1    Jung, J.2    Leboeuf, F.3
  • 6
    • 0035895236 scopus 로고    scopus 로고
    • Crystallization of hydrocortisone acetate: Influence of polymers
    • S.L. Raghavan, A. Trividic, A.F. Davis, and J. Hadgraft Crystallization of hydrocortisone acetate: influence of polymers Int. J. Pharm. 212 2003 213 221
    • (2003) Int. J. Pharm. , vol.212 , pp. 213-221
    • Raghavan, S.L.1    Trividic, A.2    Davis, A.F.3    Hadgraft, J.4
  • 7
    • 0022608689 scopus 로고
    • Effect of sodium lauryl sulphate and tween(R)80 on the therapeutic efficacy of glibenclamide tablet formulations in terms of BSL lowering in rabbits and diabetic human volunteers
    • J. Singh Effect of sodium lauryl sulfate and Tween 80 on the therapeutic efficacy of glibenclamide tablet formulations in terms of BSL lowering in rabbits and diabetic human volunteers Drug Dev. Ind. Pharm. 12 1986 851 866 (Pubitemid 16120824)
    • (1986) Drug Development and Industrial Pharmacy , vol.12 , Issue.6 , pp. 851-866
    • Singh, J.1
  • 8
    • 0021218129 scopus 로고
    • The effect of in-vivo dispersion and gastric emptying on glibenclamide absorption from a novel, rapidly dissolving capsule formulation
    • J.A. Ganley, J. McEven, R.T. Calvert, and C.J. Barker The effect of in vivo dispension and gastric emptying on glibenclamide absorption from a novel, rapidly dissolving capsule formulation J. Pharm. Pharmacol. 36 1984 734 739 (Pubitemid 14021953)
    • (1984) Journal of Pharmacy and Pharmacology , vol.36 , Issue.11 , pp. 734-739
    • Ganley, J.A.1    Mcewen, J.2    Calvert, R.T.3    Barker, M.C.J.4
  • 10
    • 47249130261 scopus 로고    scopus 로고
    • Formulation of fast disintegrating tablets of ternary solid dispersions consisting of TPGS 1000 and HPMC 2910 or PVPVA 64 to improve the dissolution of the anti-HIV drug UC 871
    • C. Goddeeris, T. Willems, and G.V.D. Mooter Formulation of fast disintegrating tablets of ternary solid dispersions consisting of TPGS 1000 and HPMC 2910 or PVPVA 64 to improve the dissolution of the anti-HIV drug UC 871 Eur. J. Pharm. Sci. 34 2008 293 302
    • (2008) Eur. J. Pharm. Sci. , vol.34 , pp. 293-302
    • Goddeeris, C.1    Willems, T.2    Mooter, G.V.D.3
  • 11
    • 1142303337 scopus 로고    scopus 로고
    • What is the true solubility advantage for amorphous pharmaceuticals?
    • DOI 10.1023/A:1007516718048
    • B.C. Hancock, and M. Parks What is the true solubility advantage for amorphous pharmaceuticals? Pharm. Res. 17 2000 397 404 (Pubitemid 30395293)
    • (2000) Pharmaceutical Research , vol.17 , Issue.4 , pp. 397-404
    • Hancock, B.C.1    Parks, M.2
  • 12
    • 0030638567 scopus 로고    scopus 로고
    • Characteristics and significance of the amorphous state in pharmaceutical systems
    • B.C. Hancock, and G. Zografi Characteristics and significance of the amorphous state in pharmaceutical systems J. Pharm. Sci. 86 1997 1 12
    • (1997) J. Pharm. Sci. , vol.86 , pp. 1-12
    • Hancock, B.C.1    Zografi, G.2
  • 13
    • 0026089175 scopus 로고
    • Characterization of glibenclamide glassy state
    • M.A. Hassan, N.M. Najib, and M.S. Suleiman Characterization of glibenclamide glassy state Int. J. Pharm. 67 1991 131 137
    • (1991) Int. J. Pharm. , vol.67 , pp. 131-137
    • Hassan, M.A.1    Najib, N.M.2    Suleiman, M.S.3
  • 14
    • 77956431273 scopus 로고    scopus 로고
    • Study of the amorphous glibenclamide drug: Analysis of the molecular dynamics of quenched and cryomilled material
    • Z. Wojnarowska, K. Grzybowska, K. Adrjanowicz, and K. Kaminski Study of the amorphous glibenclamide drug: analysis of the molecular dynamics of quenched and cryomilled material Mol. Pharm. 7 2010 1692 1707
    • (2010) Mol. Pharm. , vol.7 , pp. 1692-1707
    • Wojnarowska, Z.1    Grzybowska, K.2    Adrjanowicz, K.3    Kaminski, K.4
  • 15
    • 4143055826 scopus 로고    scopus 로고
    • Preparation of microcrystals by in situ micronization
    • DOI 10.1016/j.powtec.2004.04.021, PII S0032591004001792
    • N. Rasenack, H. Steckel, and B.W. Müller Preparation of microcrystals by in situ micronization Powder Technol. 143-144 2004 291 296 (Pubitemid 39091949)
    • (2004) Powder Technology , vol.143-144 , pp. 291-296
    • Rasenack, N.1    Steckel, H.2    Muller, B.W.3
  • 16
    • 33750089277 scopus 로고    scopus 로고
    • Preparation and in vitro/in vivo evaluation of nano-sized crystals for dissolution rate enhancement of ucb-35440-3, a highly dosed poorly water-soluble weak base
    • DOI 10.1016/j.ejpb.2006.05.008, PII S0939641106001408
    • J. Hecq, M. Deleers, D. Franara, H. Vranckx, P. Boulanger, S.L. Lamer, and K. Amighi Preparation and in vitro/in vivo evaluation of nano-sized crystals for dissolution rate enchancement of ucb-35440-3, a highly dosed poorly water-soluble weak base Eur. J. Pharm. Biopharm. 64 2006 360 368 (Pubitemid 44585201)
    • (2006) European Journal of Pharmaceutics and Biopharmaceutics , vol.64 , Issue.3 , pp. 360-368
    • Hecq, J.1    Deleers, M.2    Fanara, D.3    Vranckx, H.4    Boulanger, P.5    Le Lamer, S.6    Amighi, K.7
  • 17
    • 0036375657 scopus 로고    scopus 로고
    • Mixing and characterization of nanosized powders: An assessment of different techniques
    • DOI 10.1023/A:1020184524538
    • D. Wei, H.R. Dave, and R. Pfeffer Mixing and characterization of nanosized powders: an assessment of different techniques J. Nanopart. Res. 42 2002 21 41 (Pubitemid 135713399)
    • (2002) Journal of Nanoparticle Research , vol.4 , Issue.1-2 , pp. 21-41
    • Wei, D.1    Dave, R.2    Pfeffer, R.3
  • 20
    • 33748701219 scopus 로고    scopus 로고
    • Preparation of amorphous cefuroxime axetil nanoparticles by controlled nanoprecipitation method without surfactants
    • DOI 10.1016/j.ijpharm.2006.05.048, PII S0378517306004315
    • J.Y. Zhang, Z.G. Shen, J. Zhong, T.T. Hu, J.F. Chen, Z.Q. Ma, and J. Yun Preparation of amorphous cefuroxime axetil nanoparticles by controlled nanoprecipitation method without surfactants Int. J. Pharm. 323 2006 153 160 (Pubitemid 44397363)
    • (2006) International Journal of Pharmaceutics , vol.323 , Issue.1-2 , pp. 153-160
    • Zhang, J.-Y.1    Shen, Z.-G.2    Zhong, J.3    Hu, T.-T.4    Chen, J.-F.5    Ma, Z.-Q.6    Yun, J.7
  • 21
    • 0034042048 scopus 로고    scopus 로고
    • Rapid expansion from supercritical to aqueous solution to produce submicron suspensions of water-insoluble drugs
    • DOI 10.1021/bp000032q
    • T.J. Young, S.M. Mawson, K.P. Johnston, I.B. Henriksen, G.W. Pace, and A.K. Mishra Rapid expansion from supercritical to aqueous solution to produce submicron suspensions of water-insoluble drugs Biotechnol. Prog. 16 2000 402 407 (Pubitemid 30369011)
    • (2000) Biotechnology Progress , vol.16 , Issue.3 , pp. 402-407
    • Young, T.J.1    Mawson, S.2    Johnston, K.P.3    Henriksen, I.B.4    Pace, G.W.5    Mishra, A.K.6
  • 24
    • 33750325780 scopus 로고    scopus 로고
    • Drug nanoparticles by antisolvent precipitation: Mixing energy versus surfactant stabilization
    • DOI 10.1021/la061122t
    • M.E. Matteucci, M.A. Hotze, K.P. Johnston, and R.O. Williams III Drug nanoparticles by antisolvent precipitation: mixing energy versus surfactant stabilization Langmuir 22 2006 8951 8959 (Pubitemid 44626160)
    • (2006) Langmuir , vol.22 , Issue.21 , pp. 8951-8959
    • Matteucci, M.E.1    Hotze, M.A.2    Johnston, K.P.3    Williams III, R.O.4
  • 25
    • 67349131897 scopus 로고    scopus 로고
    • Combination chemotherapeutic dry powder aerosols via controlled nanoparticle agglomeration
    • N. EI-Gendy, and C. Berkland Combination chemotherapeutic dry powder aerosols via controlled nanoparticle agglomeration Pharm. Res. 26 2009 1752 1763
    • (2009) Pharm. Res. , vol.26 , pp. 1752-1763
    • Ei-Gendy, N.1    Berkland, C.2
  • 27
    • 67349118498 scopus 로고    scopus 로고
    • Micronization of atorvastatin calcium by antisolvent precipitation process
    • H.X. Zhang, J.X. Wanga, Z.B. Zhang, Y. Le, Z.G. Shen, and J.F. Chen Micronization of atorvastatin calcium by antisolvent precipitation process Int. J. Pharm. 374 2009 106 113
    • (2009) Int. J. Pharm. , vol.374 , pp. 106-113
    • Zhang, H.X.1    Wanga, J.X.2    Zhang, Z.B.3    Le, Y.4    Shen, Z.G.5    Chen, J.F.6
  • 28
    • 0031750464 scopus 로고    scopus 로고
    • Crystalline properties of carbamazepine in sustained release hydrophilic matrix tablets based on hydroxypropyl methylcellulose
    • I. Katzhendlera, R. Azouryb, and M. Friedmana Crystalline properties of carbamazepine in sustained release hydrophilic matrix tablets based on hydroxypropyl methylcellulose J. Controll. Release 54 1998 69 85
    • (1998) J. Controll. Release , vol.54 , pp. 69-85
    • Katzhendlera, I.1    Azouryb, R.2    Friedmana, M.3
  • 29
    • 64649088132 scopus 로고    scopus 로고
    • Amorphous compositions using concentration enhancing polymers for improved bioavailability of itraconazole
    • J.C. Dinunzio, D.A. Miller, W. Yang, G.W. Mcginity, and R.O. Williams Amorphous compositions using concentration enhancing polymers for improved bioavailability of itraconazole Mol. Pharm. 5 2008 968 980
    • (2008) Mol. Pharm. , vol.5 , pp. 968-980
    • Dinunzio, J.C.1    Miller, D.A.2    Yang, W.3    McGinity, G.W.4    Williams, R.O.5
  • 31
    • 4344604026 scopus 로고    scopus 로고
    • Physicochemical parameters associated with nanoparticle formation in the salting-out, emulsification-diffusion, and nanoprecipitation methods
    • DOI 10.1023/B:PHAM.0000036917.75634.be
    • S. Galindo-Rodriguez, S.E. Allemann, H. Fessi, and E. Doelker Physicochemical parameters associated with nanoparticle formation in the tsaltingout, emulsification-diffusion, and nanoprecipitation methods Pharm. Res. 21 2004 1428 1439 (Pubitemid 39149658)
    • (2004) Pharmaceutical Research , vol.21 , Issue.8 , pp. 1428-1439
    • Galindo-Rodriguez, S.1    Allemann, E.2    Fessi, H.3    Doelker, E.4
  • 32
    • 34548023425 scopus 로고    scopus 로고
    • Crystal engineering of active pharmaceutical ingredients to improve solubility and dissolution rates
    • DOI 10.1016/j.addr.2007.05.011, PII S0169409X07000828
    • N. Blagden, M. de Matas, P.T. Gavan, and P. York Crystal engineering of active pharmaceutical ingredients to improve solubility and dissolution rates Adv. Drug Deliv. Rev. 59 2007 617 630 (Pubitemid 47285407)
    • (2007) Advanced Drug Delivery Reviews , vol.59 , Issue.7 , pp. 617-630
    • Blagden, N.1    De Matas, M.2    Gavan, P.T.3    York, P.4


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.