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Volumn 28, Issue 1, 2011, Pages 284-290
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Label-free electrochemical measurement of protein tyrosine kinase activity and inhibition based on electro-catalyzed tyrosine signaling
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Author keywords
Electrochemical; Indium tin oxide; Kinase activity; Phosphorylation; Tyrosine
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Indexed keywords
2 ,2'-BIPYRIDINE;
DIAGNOSTIC APPLICATIONS;
DRUG DISCOVERY;
ELECTROCHEMICAL;
ELECTROCHEMICAL BIOSENSOR;
ELECTROCHEMICAL CURRENTS;
ELECTROCHEMICAL MEASUREMENTS;
ELECTROCHEMICAL METHODS;
ELECTROCHEMICAL SIGNALS;
ELECTRON MEDIATOR;
EPIDERMAL GROWTH FACTOR RECEPTORS;
EXPERIMENTAL CONDITIONS;
HIGH SENSITIVITY;
HIGH-THROUGHPUT ASSAYS;
IN-VITRO;
INDIUM TIN OXIDE;
INDIUM TIN OXIDE ELECTRODES;
INHIBITION CONSTANTS;
INHIBITOR CONCENTRATION;
KINASE ACTIVITY;
KINASE ASSAYS;
KINASE INHIBITION;
LABEL FREE;
LIMIT OF DETECTION;
PROTEIN TYROSINE KINASE;
SENSING MECHANISM;
SILANIZATIONS;
SOLID TUMORS;
TYROSINE;
VOLTAMMETRIC CURRENTS;
BIOASSAY;
BIOSENSORS;
CATALYSIS;
ENZYME INHIBITION;
INDIUM;
INDIUM COMPOUNDS;
OSMIUM;
PEPTIDES;
PHOSPHORYLATION;
TIN;
TIN OXIDES;
AMINO ACIDS;
2,2' BIPYRIDINE DERIVATIVE;
4 (3 BROMOANILINO) 6,7 DIMETHOXYQUINAZOLINE;
CYCLIC AMP DEPENDENT PROTEIN KINASE;
EPIDERMAL GROWTH FACTOR RECEPTOR;
ERLOTINIB;
GEFITINIB;
INDIUM TIN OXIDE;
PROTEIN TYROSINE KINASE;
SILANE;
TYROSINE;
ARTICLE;
CATALYSIS;
CHEMICAL REACTION;
CHEMICAL STRUCTURE;
CONCENTRATION RESPONSE;
CONTROLLED STUDY;
CYCLIC POTENTIOMETRY;
ELECTRIC CURRENT;
ELECTROCHEMICAL ANALYSIS;
ENZYME ACTIVITY;
ENZYME ASSAY;
ENZYME INHIBITION;
ENZYME STABILITY;
ENZYMIC BIOSENSOR;
HIGH THROUGHPUT SCREENING;
HUMAN;
IC 50;
IN VITRO STUDY;
LIMIT OF DETECTION;
NONHUMAN;
OXIDATION;
PROTEIN IMMOBILIZATION;
PROTEIN PHOSPHORYLATION;
QUANTITATIVE ANALYSIS;
SIGNAL PROCESSING;
SIGNAL TRANSDUCTION;
BIOSENSING TECHNIQUES;
CATALYSIS;
ELECTROCHEMICAL TECHNIQUES;
ELECTRODES;
PHOSPHORYLATION;
PROTEIN-TYROSINE KINASES;
RECEPTOR, EPIDERMAL GROWTH FACTOR;
TYROSINE;
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EID: 80052366404
PISSN: 09565663
EISSN: 18734235
Source Type: Journal
DOI: 10.1016/j.bios.2011.07.033 Document Type: Article |
Times cited : (34)
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References (37)
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