-
1
-
-
0029836953
-
Discovering high-affinity ligands for proteins: SAR by NMR
-
DOI 10.1126/science.274.5292.1531
-
SB Shuker PJ Hajduk RP Meadows SW Fesik 1996 Science 274 1531 1534 10.1126/science.274.5292.1531 1:CAS:528:DyaK28Xnt1ansLs%3D (Pubitemid 26403929)
-
(1996)
Science
, vol.274
, Issue.5292
, pp. 1531-1534
-
-
Shuker, S.B.1
Hajduk, P.J.2
Meadows, R.P.3
Fesik, S.W.4
-
4
-
-
36549033318
-
Integration of fragment screening and library design
-
DOI 10.1016/j.drudis.2007.08.005, PII S1359644607003108
-
G Siegal E Ab J Schultz 2007 Drug Discov Today 12 1032 1039 10.1016/j.drudis.2007.08.005 1:CAS:528:DC%2BD2sXhsVSmurnI (Pubitemid 350180558)
-
(2007)
Drug Discovery Today
, vol.12
, Issue.23-24
, pp. 1032-1039
-
-
Siegal, G.1
Ab, E.2
Schultz, J.3
-
5
-
-
36248944181
-
An integrated approach to fragment-based lead generation: Philosophy, strategy and case studies from AstraZeneca's drug discovery programmes
-
DOI 10.2174/156802607782341091
-
JS Albert N Blomberg AL Breeze AJ Brown JN Burrows PD Edwards RH Folmer S Geschwindner EJ Griffen PW Kenny T Nowak LL Olsson H Sanganee AB Shapiro 2007 Curr Top Med Chem 7 1600 1629 10.2174/156802607782341091 1:CAS:528: DC%2BD2sXhsVOrur%2FM (Pubitemid 350131017)
-
(2007)
Current Topics in Medicinal Chemistry
, vol.7
, Issue.16
, pp. 1600-1629
-
-
Albert, J.S.1
Blomberg, N.2
Breeze, A.L.3
Brown, A.J.H.4
Burrows, J.N.5
Edwards, P.D.6
Folmer, R.H.A.7
Geschwindner, S.8
Griffen, E.J.9
Kenny, P.W.10
Nowak, T.11
Olsson, L.-L.12
Sanganee, H.13
Shapiro, A.B.14
-
6
-
-
33751204422
-
Fragment-based lead discovery: A chemical update
-
DOI 10.1016/j.copbio.2006.10.007, PII S0958166906001510
-
DA Erlanson 2006 Curr Opin Biotechnol 17 643 652 10.1016/j.copbio.2006. 10.007 1:CAS:528:DC%2BD28Xht1eqs7zF (Pubitemid 44791912)
-
(2006)
Current Opinion in Biotechnology
, vol.17
, Issue.6
, pp. 643-652
-
-
Erlanson, D.A.1
-
7
-
-
33751112979
-
Puzzling through fragment-based drug design
-
DOI 10.1038/nchembio1206-658, PII NCHEMBIO1206658
-
PJ Hajduk 2006 Nat Chem Biol 2 658 659 10.1038/nchembio1206-658 1:CAS:528:DC%2BD28Xht1SrtLbI (Pubitemid 44764204)
-
(2006)
Nature Chemical Biology
, vol.2
, Issue.12
, pp. 658-659
-
-
Hajduk, P.J.1
-
8
-
-
33845364148
-
Fragment-based drug design: How big is too big?
-
DOI 10.1021/jm060511h
-
PJ Hajduk 2006 J Med Chem 49 6972 6976 10.1021/jm060511h 1:CAS:528:DC%2BD28XhtFOmtLbJ (Pubitemid 44885985)
-
(2006)
Journal of Medicinal Chemistry
, vol.49
, Issue.24
, pp. 6972-6976
-
-
Hajduk, P.J.1
-
10
-
-
33847381100
-
A decade of fragment-based drug design: Strategic advances and lessons learned
-
DOI 10.1038/nrd2220, PII NRD2220
-
PJ Hajduk J Greer 2007 Nat Rev Drug Discov 6 211 219 10.1038/nrd2220 1:CAS:528:DC%2BD2sXit12rtr4%3D (Pubitemid 46344625)
-
(2007)
Nature Reviews Drug Discovery
, vol.6
, Issue.3
, pp. 211-219
-
-
Hajduk, P.J.1
Greer, J.2
-
11
-
-
67649341990
-
-
10.1016/j.drudis.2009.04.007 1:CAS:528:DC%2BD1MXotFyktLo%3D
-
G Chessari AJ Woodhead 2009 Drug Discov Today 14 668 675 10.1016/j.drudis.2009.04.007 1:CAS:528:DC%2BD1MXotFyktLo%3D
-
(2009)
Drug Discov Today
, vol.14
, pp. 668-675
-
-
Chessari, G.1
Woodhead, A.J.2
-
13
-
-
0242291985
-
Why is big Pharma getting out of antibacterial drug discovery?
-
DOI 10.1016/j.mib.2003.08.003
-
SJ Projan 2003 Curr Opin Microbiol 6 427 430 10.1016/j.mib.2003.08.003 (Pubitemid 37345405)
-
(2003)
Current Opinion in Microbiology
, vol.6
, Issue.5
, pp. 427-430
-
-
Projan, S.J.1
-
14
-
-
23044491214
-
Optimizing the discovery organization for innovation
-
DOI 10.1016/S1359-6446(05)03539-7, PII S1359644605035397
-
F Sams-Dodd 2005 Drug Discov Today 10 1049 1056 10.1016/S1359-6446(05) 03539-7 (Pubitemid 41074143)
-
(2005)
Drug Discovery Today
, vol.10
, Issue.15
, pp. 1049-1056
-
-
Sams-Dodd, F.1
-
15
-
-
13844276627
-
Target-based drug discovery: Is something wrong?
-
DOI 10.1016/S1359-6446(04)03316-1, PII S1359644604033161
-
F Sams-Dodd 2005 Drug Discov Today 10 139 147 10.1016/S1359-6446(04) 03316-1 1:CAS:528:DC%2BD2MXhsFarsbk%3D (Pubitemid 40247812)
-
(2005)
Drug Discovery Today
, vol.10
, Issue.2
, pp. 139-147
-
-
Sams-Dodd, F.1
-
16
-
-
33646504430
-
-
10.1016/j.drudis.2006.04.014 1:CAS:528:DC%2BD28XkvVGjt7g%3D
-
SE Hall 2006 Drug Discov Today 11 495 502 10.1016/j.drudis.2006.04.014 1:CAS:528:DC%2BD28XkvVGjt7g%3D
-
(2006)
Drug Discov Today
, vol.11
, pp. 495-502
-
-
Hall, S.E.1
-
19
-
-
77949370572
-
-
10.1111/j.1476-5381.2009.00476.x 1:CAS:528:DC%2BC3cXjs1ektro%3D
-
M Congreve F Marshall 2010 Br J Pharmacol 159 986 996 10.1111/j.1476-5381.2009.00476.x 1:CAS:528:DC%2BC3cXjs1ektro%3D
-
(2010)
Br J Pharmacol
, vol.159
, pp. 986-996
-
-
Congreve, M.1
Marshall, F.2
-
20
-
-
78149501220
-
-
10.1016/j.neuropharm.2010.07.016
-
RE Hubbard 2010 Neuropharmacology 60 7 23 10.1016/j.neuropharm.2010.07. 016
-
(2010)
Neuropharmacology
, vol.60
, pp. 7-23
-
-
Hubbard, R.E.1
-
22
-
-
70449726880
-
-
10.1038/nrd3040 1:CAS:528:DC%2BD1MXhtlCjtr3F
-
M Goodman 2009 Nat Rev Drug Discov 8 837 10.1038/nrd3040 1:CAS:528:DC%2BD1MXhtlCjtr3F
-
(2009)
Nat Rev Drug Discov
, vol.8
, pp. 837
-
-
Goodman, M.1
-
23
-
-
34447336944
-
-
10.1002/biot.200790064 1:CAS:528:DC%2BD2sXnsVGjtrs%3D
-
NS Wong HP Kocher MG Yap 2007 Biotechnol J 2 657 658 10.1002/biot. 200790064 1:CAS:528:DC%2BD2sXnsVGjtrs%3D
-
(2007)
Biotechnol J
, vol.2
, pp. 657-658
-
-
Wong, N.S.1
Kocher, H.P.2
Yap, M.G.3
-
24
-
-
34447297884
-
Discovery and design of novel HSP90 inhibitors using multiple fragment-based design strategies
-
DOI 10.1111/j.1747-0285.2007.00535.x
-
JR Huth C Park AM Petros AR Kunzer MD Wendt X Wang CL Lynch JC Mack KM Swift RA Judge J Chen PL Richardson S Jin SK Tahir ED Matayoshi SA Dorwin US Ladror JM Severin KA Walter DM Bartley SW Fesik SW Elmore PJ Hajduk 2007 Chem Biol Drug Des 70 1 12 10.1111/j.1747-0285.2007.00535.x 1:CAS:528: DC%2BD2sXovFCktrY%3D (Pubitemid 47057425)
-
(2007)
Chemical Biology and Drug Design
, vol.70
, Issue.1
, pp. 1-12
-
-
Huth, J.R.1
Park, C.2
Petros, A.M.3
Kunzer, A.R.4
Wendt, M.D.5
Wang, X.6
Lynch, C.L.7
Mack, J.C.8
Swift, K.M.9
Judge, R.A.10
Chen, J.11
Richardson, P.L.12
Jin, S.13
Tahir, S.K.14
Matayoshi, E.D.15
Dorwin, S.A.16
Ladror, U.S.17
Severin, J.M.18
Walter, K.A.19
Bartley, D.M.20
Fesik, S.W.21
Elmore, S.W.22
Hajduk, P.J.23
more..
|