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Volumn 681, Issue , 2010, Pages 126-132

Development of α-melanocortin analogs for melanoma prevention and targeting

Author keywords

[No Author keywords available]

Indexed keywords

1,4,7,10 TETRAAZACYCLODODECANE 1,4,7,10 TETRAACETIC ACID ACETYL 4 NORLEUCINE 7 DEXTRO PHENYLALANINE ALPHA INTERMEDIN; 1,4,7,10 TETRAAZACYCLODODECANE 1,4,7,10 TETRAACETIC ACID ACETYL 4 NORLEUCINE 7 DEXTRO PHENYLALANINE ALPHA INTERMEDIN IN 111; 1,4,7,10 TETRAAZACYCLODODECANE 1,4,7,10 TETRAACETIC ACID BETA ALANYLNORLEUCYLASPARTYL DEXTRO PHENYLALANYLLYSINE ALPHA INTERMEDIN; 1,4,7,10 TETRAAZACYCLODODECANE 1,4,7,10 TETRAACETIC ACID BETA ALANYLNORLEUCYLASPARTYL DEXTRO PHENYLALANYLLYSINE ALPHA INTERMEDIN IN 111; 1,4,7,10 TETRAAZACYCLODODECANE 1,4,7,10 TETRAACETIC ACID NORLEUCYLASPARTYL DEXTRO PHENYLALANINE ALPHA INTERMEDIN; 1,4,7,10 TETRAAZACYCLODODECANE 1,4,7,10 TETRAACETIC ACID NORLEUCYLASPARTYL DEXTRO PHENYLALANINE ALPHA INTERMEDIN IN 111; 5 PHENYLBUTYRYL DERIVATIVE; ACETYL 4 NORLEUCINE 7 DEXTRO PHENYLALANINE ALPHA INTERMEDIN; ACETYL 4 NORLEUCINE [ASPARTYLHISTIDYL DEXTRO PHENYLALANYLARGINYLTRYPTOPHANYLLYSINE] AMIDE; ACETYLCYSTEINYLCYSTEINE ALPHA INTERMEDIN; ALPHA INTERMEDIN; ALPHA INTERMEDIN DERIVATIVE; BETA ALANYLNORLEUCYLASPARTYL DEXTRO PHENYLALANYLLYSINE ALPHA INTERMEDIN; BETA ALANYLNORLEUCYLASPARTYLHISTIDYL DEXTRO PHENYLALANYLARGINYLTRYPTOPHANYLLYSINE AMIDE TC 99M; COSMETIC; EUMELANIN; LK 184; MELANOCORTIN RECEPTOR AGONIST; MELANOTAN II; MELANOTAN II TC 99M; N ACETYL ALPHA INTERMEDIN[4-10]CYCLO[4 NORLEUCINE 5 ASPARTIC ACID 7 [3 (2 NAPHTHYL)ALANINE] 10 LYSINAMIDE]; N PENTADECANOYLHISTIDYL DEXTRO PHENYLALANYLARGINYLTRYPTOPHAN AMIDE; N PHENYLBUTYRYLHISTIDYL DEXTRO PHENYLALANYLARGINYLTRYPTOPHAN AMIDE; NORLEUCYLASPARTYL DEXTRO PHENYLALANINE ALPHA INTERMEDIN; PHEOMELANIN; RADIOISOTOPE; UNCLASSIFIED DRUG;

EID: 79959561922     PISSN: 00652598     EISSN: None     Source Type: Book Series    
DOI: 10.1007/978-1-4419-6354-3_10     Document Type: Article
Times cited : (9)

References (49)
  • 1
    • 0000550995 scopus 로고
    • α-Melanocyte stimulating hormone: Chemical nature and mechanism of action
    • Sawyer TK, Hruby VJ, Hadley ME et al. α-Melanocyte stimulating hormone: Chemical nature and mechanism of action. Am Zool 1983; 23:529-540.
    • (1983) Am Zool , vol.23 , pp. 529-540
    • Sawyer, T.K.1    Hruby, V.J.2    Hadley, M.E.3
  • 2
    • 0023218035 scopus 로고
    • Stimulation of follicular melanogenesis in the mouse by topical and injected melanotropins
    • Levine N, Lemus-Wilson AL, Wood SH et al. Stimulation of follicular melanogenesis in the mouse by topical and injected melanotropins. J Invest Dermatol 1987; 89:269-273. (Pubitemid 17126579)
    • (1987) Journal of Investigative Dermatology , vol.89 , Issue.3 , pp. 269-273
    • Levine, N.1    Lemus-Wilson, A.2    Wood, S.H.3
  • 3
    • 0021206553 scopus 로고
    • Action of the e locus of mice in the response of phaeomelanic hair follicles to α-melanocyte-stimulating hormone in vitro
    • Tamate HB, Takeuchi T. Action of the e locus of mice in the response of phaeomelanic hair follicles to α-melanocyte-stimulating hormone in vitro. Science 1984; 224:1241-1242. (Pubitemid 14109461)
    • (1984) Science , vol.224 , Issue.4654 , pp. 1241-1242
    • Tamate, H.B.1    Takeuchi, T.2
  • 4
    • 36949078628 scopus 로고
    • Effect of alpha- and beta-melanocyte stimulating hormones on the skin colour of man
    • Lerner AB, McGuire JS. Effect of alpha- and beta-melanocyte stimulating hormones on the skin colour of man. Nature 1961; 189:176-179.
    • (1961) Nature , vol.189 , pp. 176-179
    • Lerner, A.B.1    McGuire, J.S.2
  • 5
    • 0026800892 scopus 로고
    • The cloning of a family of genes that encode the melanocortin receptors
    • Mountjoy KG, Robbins LS, Mortrud MT et al. The cloning of a family of genes that encode the melanocortin receptors. Science 1992; 257:1248-1251.
    • (1992) Science , vol.257 , pp. 1248-1251
    • Mountjoy, K.G.1    Robbins, L.S.2    Mortrud, M.T.3
  • 6
    • 0026731363 scopus 로고
    • Molecular cloning and expression of the human melanocyte stimulating hormone receptor cDNA
    • Chhajlani V, Wikberg JES. Molecular cloning and expression of the human melanocyte stimulating hormone receptor cDNA. FEBS Lett 1992; 309:417-420.
    • (1992) FEBS Lett , vol.309 , pp. 417-420
    • Chhajlani, V.1    Wikberg, J.E.S.2
  • 7
    • 0028920049 scopus 로고
    • Mitogenic and melanogenic stimulation of normal human melanocytes by melanotropic peptides
    • Abdel-Malek Z, Swope VB, Suzuki I et al. Mitogenic and melanogenic stimulation of normal human melanocytes by melanotropic peptides. Proc Natl Acad Sci USA 1995; 92:1789-1793.
    • (1995) Proc Natl Acad Sci USA , vol.92 , pp. 1789-1793
    • Abdel-Malek, Z.1    Swope, V.B.2    Suzuki, I.3
  • 8
    • 0028493031 scopus 로고
    • Cultured human melanocytes respond to MSH peptides and ACTH
    • Hunt G, Donatien PD, Lunec J et al. Cultured human melanocytes respond to MSH peptides and ACTH. Pigment Cell Res 1994; 7:217-221.
    • (1994) Pigment Cell Res , vol.7 , pp. 217-221
    • Hunt, G.1    Donatien, P.D.2    Lunec, J.3
  • 9
    • 0029863304 scopus 로고    scopus 로고
    • Binding of melanotropic hormones to the melanocortin receptor MC1R on human melanocytes stimulates proliferation and melanogenesis
    • DOI 10.1210/en.137.5.1627
    • Suzuki I, Cone R, Im S et al. Binding of melanotropic hormones to the melanocortin receptor MC1R on human melanocytes stimulates proliferation and melanogenesis. Endocrinology 1996; 137:1627-1633. (Pubitemid 26133934)
    • (1996) Endocrinology , vol.137 , Issue.5 , pp. 1627-1633
    • Suzuki, I.1    Cone, R.D.2    Im, S.3    Nordlund, J.4    Abdel-Malek, Z.A.5
  • 11
    • 0004188831 scopus 로고    scopus 로고
    • 4th ed. Upper Saddle River, NJ: Prentice-Hall, Inc.
    • Hadley ME. Endocrinology. 4th ed. Upper Saddle River, NJ: Prentice-Hall, Inc., 1996.
    • (1996) Endocrinology
    • Hadley, M.E.1
  • 12
    • 0002148605 scopus 로고
    • The role of natural photoprotective agents in human skin
    • In: Fitzpatrick TB, Pathak MA, Haber LC et al, eds., Tokyo: University of Tokyo Press
    • Pathak MA, Fitzpatrick TB. The role of natural photoprotective agents in human skin. In: Fitzpatrick TB, Pathak MA, Haber LC et al, eds. Sunlight and Man. Tokyo: University of Tokyo Press, 1974; 725-750.
    • (1974) Sunlight and Man , pp. 725-750
    • Pathak, M.A.1    Fitzpatrick, T.B.2
  • 15
    • 0021881908 scopus 로고
    • Stimulation of S91 melanoma tyrosinase activity by superpotent α-melanotropins
    • DOI 10.1016/0303-7207(85)90020-6
    • Marwan MM, Abdel-Malek ZA, Kreutzfeld KL et al. Stimulation of S91 melanoma tyrosinase activity by superpotent α-melanotropins. Mol Cell Endocrinol 1985; 41:171-177. (Pubitemid 15022741)
    • (1985) Molecular and Cellular Endocrinology , vol.41 , Issue.2-3 , pp. 171-177
    • Marwan, M.M.1    Abdel Malek, A.A.2    Kreutzfeldt, K.L.3
  • 16
    • 0022272665 scopus 로고
    • 7]-α-MSH: A superpotent melanotropin that 'irreversibly' activates melanoma tyrosinase
    • 7]-α-MSH: A superpotent melanotropin that "irreversibly" activates melanoma tyrosinase. Endocr Res 1985; 11:157-170. (Pubitemid 16126188)
    • (1985) Endocrine Research , vol.11 , Issue.3-4 , pp. 157-170
    • Hadley, M.E.1    Abdel Malek, Z.A.2    Marwan, M.M.3
  • 18
    • 33845698356 scopus 로고    scopus 로고
    • Melanoma prevention strategy based on using tetrapeptide alpha-MSH analogs that protect human melanocytes from UV-induced damage and cytotoxicity
    • Abdel-Malek ZA, Kadekaro AL, Kavanagh RJ et al. Melanoma prevention strategy based on using tetrapeptide alpha-MSH analogs that protect human melanocytes from UV-induced damage and cytotoxicity. FASEB J 2006; 20:1561-1563.
    • (2006) FASEB J , vol.20 , pp. 1561-1563
    • Abdel-Malek, Z.A.1    Kadekaro, A.L.2    Kavanagh, R.J.3
  • 19
    • 0025791976 scopus 로고
    • Induction of skin tanning by the subcutaneous administration of a potent synthetic melanotropin
    • Levine N, Sheftel SN, Eytan T et al. Induction of skin tanning by the subcutaneous administration of a potent synthetic melanotropin. JAMA 1991; 266:2730-2736.
    • (1991) JAMA , vol.266 , pp. 2730-2736
    • Levine, N.1    Sheftel, S.N.2    Eytan, T.3
  • 21
    • 33645407840 scopus 로고    scopus 로고
    • Melanocortin peptide therapeutics: Historical milestones, clinical studies and commercialization
    • Hadley ME, Dorr RT. Melanocortin peptide therapeutics: Historical milestones, clinical studies and commercialization. Peptides 2006; 27(4):921-930.
    • (2006) Peptides , vol.27 , Issue.4 , pp. 921-930
    • Hadley, M.E.1    Dorr, R.T.2
  • 22
    • 0026952043 scopus 로고
    • Effects of a melanotropic peptide on melanoma cell growth, metastasis and invasion
    • Gehlsen KR, Hadley ME, Levine N et al. Effects of a melanotropic peptide on melanoma cell growth, metastasis and invasion. Pigment Cell Res 1992; 5:219-223.
    • (1992) Pigment Cell Res , vol.5 , pp. 219-223
    • Gehlsen, K.R.1    Hadley, M.E.2    Levine, N.3
  • 24
    • 0029450765 scopus 로고
    • 7] alpha-MSH, stimulates human melanoma tyrosinase activity and inhibits cell proliferation
    • 7] alpha-MSH, stimulates human melanoma tyrosinase activity and inhibits cell proliferation. Pigment Cell Res 1995; 8(6):314-323.
    • (1995) Pigment Cell Res , vol.8 , Issue.6 , pp. 314-323
    • Jiang, J.1    Sharma, S.D.2    Nakamura, S.3
  • 25
    • 0020378771 scopus 로고
    • Comparative biological activities of highly potent active-site analogues of α-melanotropin
    • DOI 10.1021/jm00351a004
    • Sawyer TK, Hruby VJ, Wilkes BC et al. Comparative biological activities of highly potent active-site analogues of α-melanotropin. J Med Chem 1982; 25:1022-1027. (Pubitemid 13233571)
    • (1982) Journal of Medicinal Chemistry , vol.25 , Issue.9 , pp. 1022-1027
    • Sawyer, T.K.1    Hruby, V.J.2    Wilkes, B.C.3
  • 26
    • 0024310869 scopus 로고
    • Potent and prolonged acting cyclic lactam analogues of α-melanotropin: Design based on molecular dynamics
    • DOI 10.1021/jm00132a010
    • Al-Obeidi F, Castrucci AM, Hadley ME et al. Potent and prolonged acting cyclic lactam analogues of alpha-melanotropin: Design based on molecular dynamics. J Med Chem 1989; 32(12):2555-2561. (Pubitemid 20002805)
    • (1989) Journal of Medicinal Chemistry , vol.32 , Issue.12 , pp. 2555-2561
    • Al-Obeidi, F.1    De Castrucci, A.M.L.2    Hadley, M.E.3    Hruby, V.J.4
  • 27
    • 0029154516 scopus 로고
    • 7,Lys10]-α-MSH(4-10)-NH-2 with bulky aromatic amino acids at position 7 show high antagonist potency and selectivity at specific melanocortin receptors
    • 7,Lys10]-α- MSH(4-10)-NH-2 with bulky aromatic amino acids at position 7 show high antagonist potency and selectivity at specific melanocortin receptors. J Med Chem 1995; 38:3454-3461.
    • (1995) J Med Chem , vol.38 , pp. 3454-3461
    • Hruby, V.J.1    Lu, D.2    Sharma, S.D.3
  • 28
    • 0344495976 scopus 로고    scopus 로고
    • Design and pharmacology of peptoids and peptide-peptoid hybrids based on the melanocortin agonists core tetrapeptide sequence
    • DOI 10.1016/j.bmcl.2003.08.078
    • Holder JR, Bauzo RM, Xiang Z et al. Design and pharmacology of peptoids and peptide-peptoid hybrids based on the melanocortin agonists core tetrapeptide sequence. Bioorg Med Chem Lett 2003; 13(24):4505-4509. (Pubitemid 37490846)
    • (2003) Bioorganic and Medicinal Chemistry Letters , vol.13 , Issue.24 , pp. 4505-4509
    • Holder, J.R.1    Bauzo, R.M.2    Xiang, Z.3    Scott, J.4    Haskell-Luevano, C.5
  • 30
    • 70350102180 scopus 로고    scopus 로고
    • Alpha-MSH activates immediate defense responses to UV-induced oxidative stress in human melanocytes
    • In press
    • Song X, Mosbi N, Yang J et al. Alpha-MSH activates immediate defense responses to UV-induced oxidative stress in human melanocytes. Pigment Cell Mel Res 2009, In press.
    • (2009) Pigment Cell Mel Res
    • Song, X.1    Mosbi, N.2    Yang, J.3
  • 32
    • 45549108249 scopus 로고    scopus 로고
    • Melanocortin-1 receptor signaling markedly induces the expression of the NR4A nuclear receptor subgroup in melanocytic cells
    • Smith AG, Luk N, Newton RA et al. Melanocortin-1 receptor signaling markedly induces the expression of the NR4A nuclear receptor subgroup in melanocytic cells. J Biol Chem 2008; 283(18):12564-12570.
    • (2008) J Biol Chem , vol.283 , Issue.18 , pp. 12564-12570
    • Smith, A.G.1    Luk, N.2    Newton, R.A.3
  • 35
    • 69449092097 scopus 로고    scopus 로고
    • α-MSH tripeptide analogs activate the melanocortin 1 receptor and reduce UV-induced DNA damage in human melanocytes
    • In press
    • Abdel-Malek ZA, Ruwe AR, Kavanagh-Starner R et al. α-MSH tripeptide analogs activate the melanocortin 1 receptor and reduce UV-induced DNA damage in human melanocytes. Pigment Cell Mel Res 2009, In press.
    • (2009) Pigment Cell Mel Res
    • Abdel-Malek, Z.A.1    Ruwe, A.R.2    Kavanagh-Starner, R.3
  • 36
    • 0030782275 scopus 로고    scopus 로고
    • Characterization of melanocyte stimulating hormone receptor variant alleles in twins with red hair
    • DOI 10.1093/hmg/6.11.1891
    • Box NF, Wyeth JR, O'Gorman LE et al. Characterization of melanocyte stimulating hormone receptor variant alleles in twins with red hair. Hum Mol Genet 1997; 6:1891-1897. (Pubitemid 27460365)
    • (1997) Human Molecular Genetics , vol.6 , Issue.11 , pp. 1891-1897
    • Box, N.F.1    Wyeth, J.R.2    O'Gorman, L.E.3    Martin, N.G.4    Sturm, R.A.5
  • 44
    • 66149184413 scopus 로고    scopus 로고
    • Glycosylated DOTA-alpha-melanocyte-stimulating hormone analogues for melanoma targeting: Influence of the site of glycosylation on in vivo biodistribution
    • Bapst JP, Calame M, Tanner H et al. Glycosylated DOTA-alpha-melanocyte- stimulating hormone analogues for melanoma targeting: Influence of the site of glycosylation on in vivo biodistribution. Bioconjug Chem 2009.
    • (2009) Bioconjug Chem
    • Bapst, J.P.1    Calame, M.2    Tanner, H.3
  • 46
    • 48949095565 scopus 로고    scopus 로고
    • Peptide-targeted radionuclide therapy for melanoma
    • Miao Y, Quinn TP. Peptide-targeted radionuclide therapy for melanoma. Crit Rev Oncol Hematol 2008; 67(3):213-228.
    • (2008) Crit Rev Oncol Hematol , vol.67 , Issue.3 , pp. 213-228
    • Miao, Y.1    Quinn, T.P.2
  • 48
    • 0033770092 scopus 로고    scopus 로고
    • The melanocortin 5 receptor is expressed in human sebaceous glands and rat preputial cells
    • Thiboutot D, Sivarajah A, Gilliland K et al. The melanocortin 5 receptor is expressed in human sebaceous glands and rat preputial cells. J Invest Dermatol 2000; 115(4):614-619.
    • (2000) J Invest Dermatol , vol.115 , Issue.4 , pp. 614-619
    • Thiboutot, D.1    Sivarajah, A.2    Gilliland, K.3
  • 49
    • 33645074690 scopus 로고    scopus 로고
    • Quantitative analysis of MC1R gene expression in human skin cell cultures
    • Roberts DW, Newton RA, Beaumont KA et al. Quantitative analysis of MC1R gene expression in human skin cell cultures. Pigment Cell Res 2006; 19(1):76-89.
    • (2006) Pigment Cell Res , vol.19 , Issue.1 , pp. 76-89
    • Roberts, D.W.1    Newton, R.A.2    Beaumont, K.A.3


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