Synthesis of a [18F]fluoroethyltriazolylthymidine radiotracer from [18F]2-fluoroethyl azide and 5-ethynyl-2′-deoxyuridine

Journal of Labelled Compounds and Radiopharmaceuticals

Volumn 54, Issue 5, 2011, Pages 260-266

  Ackermann, U ^a,b   O'Keefe, G ^a   Lee, S T ^a,b,c   Rigopoulos, A ^c   Cartwright, G ^c   Sachinidis, J I ^a   Scott, A M ^a,b,c   Tochon Danguy, H J ^a,b  

^a AUSTIN HEALTH   (Australia)

^b UNIVERSITY OF MELBOURNE   (Australia)

^c LUDWIG INSTITUTE FOR CANCER RESEARCH   (Australia)

Author keywords

A431 tumors; click chemistry; thymidine analogue; tumor cell proliferation

Indexed keywords

CELL PROLIFERATION; COPPER COMPOUNDS; POSITRON EMISSION TOMOGRAPHY; RADIOACTIVE TRACERS; SYNTHESIS (CHEMICAL);

A431 TUMOR; CLICK CHEMISTRY; DEOXYURIDINE; ETHYNYL; RADIOCHEMICAL YIELD; SPECIFIC ACTIVITY; SYNTHESIS TIME; THYMIDINE ANALOG; TUMOR CELL PROLIFERATION; TUMOUR CELLS;

TUMORS;

2 FLUOROETHYL AZIDE F 18; 5 ETHYNYLDEOXYURIDINE; AZIDE; COPPER; DEOXYURIDINE DERIVATIVE; FLUOROETHYLTRIAZOLYLTHYMIDINE F 18; TRACER; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ANIMAL MODEL; ARTICLE; BLOOD SAMPLING; CELL PROLIFERATION; CHEMICAL REACTION; COMPUTER ASSISTED EMISSION TOMOGRAPHY; CONTROLLED STUDY; DRUG SYNTHESIS; FEMALE; HUMAN; HUMAN TISSUE; MOUSE; NONHUMAN; RADIOACTIVITY; RADIOCHEMISTRY;

ANIMALIA; MUS MUSCULUS;

EID: 79958242704     PISSN: 03624803     EISSN: 10991344     Source Type: Journal    
DOI: 10.1002/jlcr.1863     Document Type: Article

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