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ChemMedChem

Volumn 6, Issue 6, 2011, Pages 996-1000

Psoralenquinones as a novel class of proteasome inhibitors: Design, synthesis and biological evaluation

(5) Marzaro, Giovanni a Gandin, Valentina a Marzano, Christine a Guiotto, Adriano a Chilin, Adriana a

a UNIVERSITY OF PADOVA (Italy)

Author keywords

Cytotoxicity; Molecular docking; Proteasome activity; Psoralenquinones

Indexed keywords

BORTEZOMIB; CALPASTATIN; FUROCHROMONE DERIVATIVE; LACTACYSTIN; PROTEASOME INHIBITOR; PSORALENQUINONE DERIVATIVE; QUINONE DERIVATIVE; TMC 95 A; UNCLASSIFIED DRUG;

ANTINEOPLASTIC ACTIVITY; ARTICLE; CANCER CELL CULTURE; CHEMICAL REACTION; CYTOPATHOGENIC EFFECT; DRUG DESIGN; DRUG IDENTIFICATION; DRUG SCREENING; DRUG SELECTIVITY; DRUG SYNTHESIS; ENZYME ACTIVE SITE; ENZYME ACTIVITY; ENZYME ASSAY; ENZYME INHIBITION; ENZYME SPECIFICITY; HUMAN; HUMAN CELL; IC 50; MOLECULAR DOCKING; PRIORITY JOURNAL; STRUCTURE ACTIVITY RELATION;

ANTINEOPLASTIC AGENTS; CELL LINE, TUMOR; DRUG SCREENING ASSAYS, ANTITUMOR; ENZYME INHIBITORS; FICUSIN; HUMANS; MODELS, MOLECULAR; NEOPLASMS; PROTEASOME ENDOPEPTIDASE COMPLEX; PROTEIN BINDING; QUINONES;

EID: 79957619498 PISSN: 18607179 EISSN: 18607187 Source Type: Journal
DOI: 10.1002/cmdc.201100041 Document Type: Article

Times cited : (3)

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