Synthesis of 3-amino-4-fluoropyrazoles

Journal of Organic Chemistry

Volumn 76, Issue 10, 2011, Pages 4105-4111

  Surmont, Riccardo ^a   Verniest, Guido ^a   De Schrijver, Mathias ^a   Thuring, Jan Willem ^b   Ten Holte, Peter ^b   Deroose, Frederik ^b   De Kimpe, Norbert ^a  

^a GHENT UNIVERSITY   (Belgium)

^b JANSSEN RESEARCH AND DEVELOPMENT   (Belgium)

Author keywords

[No Author keywords available]

Indexed keywords

BUILDING BLOCKES; CHLOROMETHYL; ENAMINOKETONES; FLUORINATED PYRAZOLES; FUNCTIONALIZATIONS; MEDICINAL CHEMISTRY; SELECTFLUOR; SYNTHETIC STRATEGIES; TETRAFLUOROBORATES;

FUNCTIONAL GROUPS;

AMINOKETONE; BORIC ACID; HYDRAZINE DERIVATIVE; PYRAZOLE DERIVATIVE; SELECTFLUOR; UNCLASSIFIED DRUG;

ARTICLE; FLUORINATION; POLYMERIZATION; SYNTHESIS;

HALOGENATION; PYRAZOLES;

EID: 79956087435     PISSN: 00223263     EISSN: 15206904     Source Type: Journal    
DOI: 10.1021/jo2000989     Document Type: Article

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