Amorphous trehalose dihydrate by cryogenic milling

Carbohydrate Research

Volumn 346, Issue 8, 2011, Pages 1061-1064

  Megarry, A J ^a   Booth, J ^b   Burley, J ^a  

^a UNIVERSITY OF NOTTINGHAM   (United Kingdom)

^b ASTRAZENECA   (United Kingdom)

Author keywords

Amorphous; Cryomilling; DSC; Hydrates; Raman spectroscopy; XRPD

Indexed keywords

AMORPHOUS; CRYOGENIC MILLING; CRYOGENIC TEMPERATURES; CRYOMILLING; DIHYDRATES; DSC; FOOD INGREDIENTS; GLASS TRANSFORMATIONS; NATURALLY OCCURRING; PHARMACEUTICAL EXCIPIENT; ROOM TEMPERATURE; XRPD;

CRYOGENICS; HYDRATES; HYDRATION; RAMAN SCATTERING; RAMAN SPECTROSCOPY;

MILLING (MACHINING);

DISACCHARIDE; EXCIPIENT; TREHALOSE;

ARTICLE; CRYOMILLING; DIFFERENTIAL SCANNING CALORIMETRY; DRUG FORMULATION; DRUG INDUSTRY; FOOD INDUSTRY; PRIORITY JOURNAL; PROCESS TECHNOLOGY; RAMAN SPECTROMETRY; TEMPERATURE; X RAY POWDER DIFFRACTION;

CHEMISTRY, PHARMACEUTICAL; COLD TEMPERATURE; TREHALOSE; WATER;

EID: 79955682577     PISSN: 00086215     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.carres.2011.03.011     Document Type: Article

References (33)

1. Pifferi, G.; Santoro, P.; Pedrani, M. Il Farmaco 1999, 54, 1-14.
2. Listiohadi, Y.; Hourigan, J.; Sleigh, R.; Steele, R. Int. J. Pharm. 2008, 359, 123-134.
3. Lipinski, C. A. J. Pharmacol. Toxicol. Methods 2000, 44, 235-249.
4. Hancock, B. C.; Parks, M. Pharm. Res. 2000, 17, 397-404.
5. Ediger, M. D.; Angell, C. A.; Nagel, S. R. J. Phys. Chem. 1996, 100, 13200-13212.
6. Vehring, R. Pharm. Res. 2008, 25, 999-1022.
7. Willart, J. F.; Descamps, M. Mol. Pharm. 2008, 5, 905-920.
8. Martin, G., Bellon, P., Eds.Solid State Physics; Academic Press, 1996; Vol. 50, pp 189-331.
9. Serajuddin, A. T. M. J. Pharm. Sci. 1999, 88, 1058-1066.
10. Ye, J.; Schoenung, J. Adv. Eng. Mater. 2004, 6, 656-664.
11. Colombo, I.; Grassi, G.; Grassi, M. J. Pharm. Sci. 2009, 98, 3961-3986.
12. Fecht, H. J. Nature 1992, 356, 133-135.
13. Sundararaman, D. Mater. Sci. Eng., B 1995, 32, 307-313.
14. Descamps, M.; Willart, J.; Dudognon, E.; Caron, V. J. Pharm. Sci. 2007, 96, 1398-1407.
15. Khankari, R. K.; Grant, D. J. W. Thermochim. Acta 1995, 248, 61-79.
16. Rodríguez-Hornedo, N.; Lechuga-Ballesteros, D.; Wu, H. J. Int. J. Pharm. 1992, 85, 149-162.
17. Authelin, J. Int. J. Pharm. 2005, 303, 37-53.
18. Devlin, J.; Buch, V.; Mohamed, F.; Parrinello, M. Chem. Phys. Lett. 2006, 432, 462-467.
19. Parthasaradhi Reddy, B.; Rathnakar Reddy, K.; Raji Reddy, R.; Muralidhara Reddy, D. Amorphous Esomeprazole Hydrate, United States Patent, 7638634, 2009.
20. Desphande, P. B.; Khadangale, B. P.; Ramasubbu, C. Amorphous Hydrate of a Cephalosporin Antibiotic, United States Patent, 7244842, 2007.
21. Center for Food Safety and Applied Nutrition GRAS Notice Inventory-Agency Response Letter GRAS Notice No. GRN 000045. http://www.fda.gov/Food/ FoodIngredientsPackaging/GenerallyRecognizedasSafeGRAS/GRASListings/ ucm154119.htm.
22. Willart, J. F.; De Gusseme, A.; Hemon, S.; Descamps, M.; Leveiller, F.; Rameau, A. J. Phys. Chem. B 2002, 106, 3365-3370.
23. Willart, J. F.; Danede, F.; De Gusseme, A.; Descamps, M.; Neves, C. J. Phys. Chem. B 2003, 107, 11158-11162.
24. Willart, J. F.; Descamps, M.; Caron, V. AIP Conf. Proc. 2008, 982, 108-113.
25. Willart, J. F.; Dujardin, N.; Dudognon, E.; Danède, F.; Descamps, M. Carbohydr. Res. 2010, 345, 1613-1616.
26. Taylor, L. S.; York, P. J. Pharm. Sci. 1998, 87, 347-355.
27. Furuki, T.; Kishi, A.; Sakurai, M. Carbohydr. Res. 2005, 340, 429-438.
28. Miller, D. P.; de Pablo, J. J. J. Phys. Chem. B 2000, 104, 8876-8883.
29. Brittain, H. G. J. Pharm. Sci. 2002, 91, 1573-1580.
30. Brown, G. M.; Rohrer, D. C.; Berking, B.; Beevers, C. A.; Gould, R. O.; Simpson, R. Acta Crystallogr., B Struct. Crystallogr. Cryst. Chem. 1972, 28, 3145-3158.
31. Hédoux, A.; Paccou, L.; Guinet, Y.; Willart, J.; Descamps, M. Eur. J. Pharm. Sci. 2009, 38, 156-164.
32. Courtens, E.; Foret, M.; Hehlen, B.; Vacher, R. Solid State Commun. 2001, 117, 187-200.
33. Gordon, M.; Taylor, J. S. J. Appl. Chem. 1952, 2, 493-500.