Fluorescence investigation of a specific structure formed by aggregation of transglycosylated stevias: Solubilizing effect of poorly water-soluble drugs

European Journal of Pharmaceutical Sciences

Volumn 43, Issue 1-2, 2011, Pages 71-77

  Uchiyama, Hiromasa ^a   Tozuka, Yuichi ^a   Asamoto, Fusatoshi ^a   Takeuchi, Hirofumi ^a  

^a GIFU PHARMACEUTICAL UNIVERSITY   (Japan)

Author keywords

Glycosyl transferase treated stevia; Dissolution; Fluorescence spectroscopy; Pyrene; Solubilization

Indexed keywords

ALPHA GLYCOSYL TRANSFERASE TREATED STEVIA; DRUG ADDITIVE; INDOMETACIN; PYRENE; STEVIOL; UNCLASSIFIED DRUG;

ARTICLE; CONTROLLED STUDY; DISSOLUTION; FLUORESCENCE SPECTROSCOPY; GLYCOSYLATION; HUMAN; HUMAN CELL; HYDROPHOBICITY; MICELLE; MOLECULAR PROBE; PRIORITY JOURNAL; SOLUBILIZATION; SPRAY DRYING; STEVIA; X RAY POWDER DIFFRACTION;

CARBOXYLIC ACIDS; DRUG CARRIERS; GLYCOSYLATION; HYDROPHOBIC AND HYDROPHILIC INTERACTIONS; INDOMETHACIN; MICELLES; MICROSCOPY, ELECTRON, SCANNING; MOLECULAR STRUCTURE; NAPHTHALENES; PARTICLE SIZE; PHARMACEUTICAL PREPARATIONS; POWDERS; PYRENES; SOLUBILITY; SPECTROMETRY, FLUORESCENCE; STEVIA; SURFACE PROPERTIES; WATER; X-RAY DIFFRACTION;

EID: 79955680567     PISSN: 09280987     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.ejps.2011.03.014     Document Type: Article

References (27)

1. J. Aguiar, J.A. Molina-Boĺivar, J.M. Peula-Garćia, and R.C. Carnero Thermodynamics and micellar properties of tetradecyltrimethylammonium bromide in formamide-water mixtures J. Colloid Interf. Sci. 255 2002 382 390 (Pubitemid 36027022)
2. J. Aguiar, P. Carpenaa, J.A. Molina-Bolívara, and R.C. Carnero On the determination of the critical micelle concentration by the pyrene 1:3 ratio method J. Colloid Interf. Sci. 258 2003 116 122 (Pubitemid 36228364)
3. D.E. Alonzo, G.G. Zhang, D. Zhou, Y. Gao, and L.S. Taylor Understanding the behavior of amorphous pharmaceutical systems during dissolution Pharm. Res. 27 2010 608 618
4. O. Anthony, and R. Zana Fluorescence investigation of the binding of pyrene to hydrophobic microdomains in aqueous solutions of polysoaps Macromolecules 27 1994 3885 3891
5. T.J. Burkey, D. Griller, D.A. Lindsay, and J.C. Scaiano Simple method for quantifying the distribution of organic substrates between the micellar and aqueous phases of sodium dodecyl sulfate solution J. Am. Chem. Soc. 106 1984 1983 1985 (Pubitemid 14568833)
6. W.L. Chiou, S.J. Chen, and N. Athanikar Enhancement of dissolution rates of poorly water-soluble drugs by crystallization in aqueous surfactant solutions I: Sulfathiazole, prednisone, and chloramphenicol J. Pharm. Sci. 65 1976 1702 1704
7. J.C. DiNunzio, C. Brough, D.A. Miller, R.O. Williams 3rd, and J.W. McGinity Applications of KinetiSol dispersing for the production of plasticizer free amorphous solid dispersions Eur. J. Pharm. Sci. 40 2010 179 187
8. H.A. Garekani, F. Sadeghi, and A. Ghazi Increasing the aqueous solubility of acetaminophen in the presence of polyvinylpyrrolidone and investigation of the mechanisms involved Drug Dev. Ind. Pharm. 29 2003 173 179 (Pubitemid 36292940)
9. V. Glushko, M.S. Thaler, and C.D. Karp Pyrene fluorescence fine structure as a polarity probe of hydrophobic regions: behavior in model solvents Arch. Biochem. Biophys. 210 1981 33 42
10. K. Kalyanasundaram, and J.K. Thomas Environmental effects on vibronic band intensities in pyrene monomer fluorescence and their application in studies of micellar systems J. Am. Chem. Soc. 99 1976 2039 2044
11. D.S. Karpovich, and G.J. Blanchard Relating the polarity-dependent fluorescence response of pyrene to vibronic coupling. Achieving a fundamental understanding of the py polarity scale J. Phys. Chem. 99 1995 3951 3958
12. K. Lee, S.C. Shin, and I. Oh Fluorescence spectroscopy studies on micellization of poloxamer 407 solution Arch. Pharm. Res. 26 2003 653 658 (Pubitemid 43080199)
13. M. Maghsoodi, and F. Sadeghpoor Preparation and evaluation of solid dispersions of piroxicam and Eudragit S100 by spherical crystallization technique Drug Dev. Ind. Pharm. 36 2010 917 925
14. S. Miyagishi, W. Akasohu, T. Hashimoto, and T. Asakawa Effect of NaCl on aggregation number, microviscosity, and Cmc of N-dodecanoyl amino acid surfactant micelles J. Colloid Interf. Sci. 184 1996 527 534 (Pubitemid 27061986)
15. G. Muhrer, U. Meier, F. Fusaro, S. Albano, and M. Mazzotti Use of compressed gas precipitation to enhance the dissolution behavior of a poorly water-soluble drug: generation of drug microparticles and drug-polymer solid dispersions Int. J. Pharm. 308 2006 69 83 (Pubitemid 43097237)
16. O. Regeva, and R. Zana Aggregation behavior of tyloxapol, a nonionic surfactant oligomer, in aqueous solution J. Colloid Interf. Sci. 210 1999 8 17 (Pubitemid 29394475)
17. H. Sekikawa, J. Fujiwara, T. Naganuma, M. Nakano, and T. Arita Dissolution behaviors and gastrointestinal absorption of phenytoin in phenytoin-polyvinylpyrrolidone coprecipitate Chem. Pharm. Bull. 10 1978 3033 3039 (Pubitemid 9050291)
18. M. Tachiya, and A. Mozumder Kinetics of geminate-ion recombination by electron tunneling Chem. Phys. Lett. 34 1975 77 79
19. L.S. Taylor, and G. Zografi Spectroscopic characterization of interactions between PVP and indomethacin in amorphous molecular dispersions Pharm. Res. 14 1997 1691 1698 (Pubitemid 28062912)
20. Y. Tozuka, C. Yokohama, K. Higashi, K. Moribe, and K. Yamamoto Adsorption state of naphthoic acids on folded sheets mesoporous materials with different pore sizes J. Drug Del. Sci. Tech. 19 2009 401 404
21. K. Tsubonea, and S. Ghoshb Micellization of an anionic gemini surfactant having N, N-dialkylamide, carboxyl, and carboxylate groups in aqueous NaCl solutions J. Surfact Deterg. 7 2004 47 52
22. N.J. Turro, and A. Yekta Luminescent probes for detergent solutions. A simple procedure for determination of the mean aggregation number of micelles J. Am. Chem. Soc. 100 1978 5951 5952
23. H. Uchiyama, Y. Tozuka, M. Imono, and H. Takeuchi Transglycosylated stevia and hesperidin as pharmaceutical excipients: dramatic improvement in drug dissolution and bioavailability Eur. J. Pharm. Sci. 76 2010 238 244
24. M. Ueno, Y. Kimoto, Y. Ikeda, H. Momosea, and R. Zana Study on the aggregation number of mixed micelles in aqueous binary mixtures of the bile salts and nonionic surfactant J. Colloid Interf. Sci. 117 1986 179 186
25. K. Wu, J. Li, W. Wang, and D.A. Winstead Formation and characterization of solid dispersions of piroxicam and polyvinylpyrrolidone using spray drying and precipitation with compressed antisolvent J. Pharm. Sci. 98 2009 2422 2431
26. M. Yang, P. Wang, C.Y. Huang, M.S. Ku, H. Liu, and C. Gogos Solid dispersion of acetaminophen and poly(ethylene oxide) prepared by hot-melt mixing Int. J. Pharm. 395 2010 53 61
27. M. Yoshioka, B.C. Hancock, and G. Zografi Inhibition of indomethacin crystallization in poly (vinylpyrrolidone) coprecipitates J. Pharm. Sci. 84 1995 983 986