Development of anti-EGF receptor peptidomimetics (AERP) as tumor imaging agent

Bioorganic and Medicinal Chemistry Letters

Volumn 21, Issue 8, 2011, Pages 2550-2553

  Ponde, Datta E ^a,c   Su, Zifen ^b   Berezov, Alan ^a   Zhang, Hongtao ^a   Alavi, Abbas ^a   Greene, Mark I ^a   Murali, Ramachandran ^a,c  

^a UNIVERSITY OF PENNSYLVANIA   (United States)

^b SICHUAN UNIVERSITY   (China)

^c CEDARS SINAI MEDICAL CENTER   (United States)

Author keywords

AERP 2; c erbB2; EGFR; EGFR specific radiotracer; Radiolabeled peptidomimetics and peptide; Technetium 99m; Tyrosine kinase receptors

Indexed keywords

CONTRAST MEDIUM; EPIDERMAL GROWTH FACTOR RECEPTOR; EPIDERMAL GROWTH FACTOR RECEPTOR KINASE INHIBITOR; EPIDERMAL GROWTH FACTOR RECEPTOR PEPTIDOMIMETIC INHIBITOR; PENTETATE TECHNETIUM TC 99M; PENTETIC ACID; PEPTIDOMIMETIC AGENT; TECHNETIUM 99M; TRACER; UNCLASSIFIED DRUG;

ARTICLE; BREAST CANCER; CELL LYSATE; DRUG BINDING; DRUG SPECIFICITY; DRUG TARGETING; HUMAN; HUMAN CELL; LUNG CANCER; METASTASIS; NONHUMAN; PANCREAS CANCER; PROSTATE CANCER; PROTEIN EXPRESSION; RECEPTOR BINDING; SOLID TUMOR;

ANIMALS; CELL LINE, TUMOR; ENZYME INHIBITORS; HUMANS; MICE; MICE, NUDE; NEOPLASMS; PENTETIC ACID; PEPTIDOMIMETICS; RADIOPHARMACEUTICALS; RECEPTOR, EPIDERMAL GROWTH FACTOR; TECHNETIUM; TISSUE DISTRIBUTION; TRANSPLANTATION, HETEROLOGOUS;

EID: 79953285347     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2011.02.013     Document Type: Article

References (36)

1. G. Pines, W.J. Kostler, and Y. Yarden FEBS Lett. 584 2010 2699
2. Y. Yarden, and M.X. Sliwkowski Nat. Rev. Mol. Cell Biol. 2 2001 127
3. C.M. Warren, and R. Landgraf Cell. Signalling 18 2006 923
4. Z. Suo, B. Risberg, M.G. Karlsson, K. Villman, E. Skovlund, and J.M. Nesland Int. J. Surg. Pathol. 10 2002 91
5. I.K. Mellinghoff, C. Tran, and C.L. Sawyers Cancer Res. 62 2002 5254
6. V. Smith, S. Hobbs, W. Court, S. Eccles, P. Workman, and L.R. Kelland Anticancer Res. 22 2002 1993
7. M. Korc Surg. Oncol. Clin. N. Am. 7 1998 25
8. B.H. Brandt, A. Roetger, T. Dittma, G. Nikolai, M. Seeling, A. Merschjann, J.R. Nofer, G. Dehmer-Moller, R. Junker, G. Assmann, and K.S. Zaenker FASEB J. 13 1999 1939
9. R.S. Herbst, and D.M. Shin Cancer 94 2002 1593
10. R.M. Reilly, R. Kiarash, J. Sandhu, Y.W. Lee, R.G. Cameron, A. Hendler, K. Vallis, and J. Gariepy J. Nucl. Med. 41 2000 903
11. R.S. Herbst, and M.S. Kies Clin. Adv. Hematol. Oncol. 1 2003 466
12. E. Laack, G. Sauter, and C. Bokemeyer Lung Cancer 69 2010 259
13. E.A. Saukville, Y. El-Sayed, M. Monga, and G. Kim Annu. Pharmacol. Toxicol. 43 2003 199
14. J. Tol, and C.J. Punt Clin. Ther. 32 2010 437
15. B. Liu, and Z. Fan Oncogene 20 2001 3726
16. R.S. Herbst, and W.K. Hong Semin. Oncol. 5 2002 18
17. A. Cuartero-Plaza, E. Martinex-Miralles, R. Rosell, C. Vadell-Nadal, M. Farre, and F.X. Real Clin. Cancer Res. 2 1996 13
18. J. Capala, R.F. Barth, M.Q. Bailey, R.A. Fenstermaker, M.J. Marek, and B.A. Rhodes Bioconjugate Chem. 8 1997 289
19. N. Xu, G. Cai, W. Ye, X. Wang, Y. Li, P. Zhao, A. Zhang, R. Zhang, and B. Cao Anticancer Res. 29 2009 4005
20. L.O.T. Gainkam, L. Huang, V. Caveliers, M. Keyaerts, S. Hernot, I. Vaneycken, C. Vanhove, H. Revets, P. De Baetselier, and T. Lahoutte J. Nucl. Med. 49 2008 788
21. A. Bell, Z.J. Wang, M. Arbabi-Ghahroudi, T.A. Chang, Y. Durocher, U. Trojahn, J. Baardsnes, M.L. Jaramillo, S. Li, T.N. Baral, M. O'Connor-McCourt, R. MacKenzie, and J. Zhang Cancer Lett. 289 2010 81
22. E. Nordberg, M. Friedman, L. Gostring, G.P. Adams, H. Brismar, F.Y. Nilsson, S. Stahl, B. Glimelius, and J. Carlsson Nucl. Med. Biol. 34 2007 609
23. D. Blok, R.I. Feitsma, P. Vermeij, and E.J. Pauwels Eur. J. Nucl. Med. 26 1999 1511
24. J.C. Reubi, and H.R. Maecke J. Nucl. Med. 49 2008 1735
25. F. Buchegger, F. Bonvin, M. Kosinski, A.O. Schaffland, J. Prior, J.C. Reubi, P. Blauenstein, D. Tourwe, E. Garcia Garayoa, and A. Bischof Delaloye J. Nucl. Med. 44 2003 1649
26. K.S. Lin, A. Luu, K.E. Baidoo, H. Hashemzadeh-Gargari, M.K. Chen, K. Brenneman, R. Pili, M. Pomper, M.A. Carducci, and H.N. Wagner Jr. Bioconjugate Chem. 16 2005 43
27. X. Chen, Y. Hou, M. Tohme, R. Park, V. Khankaldyyan, I. Gonzales-Gomez, J.R. Bading, W.E. Laug, and P.S. Conti J. Nucl. Med. 45 2004 1776
28. A.T. Brunger, P.D. Adams, G.M. Clore, W.L. DeLano, P. Gros, R.W. Grosse-Kunstleve, J.S. Jiang, J. Kuszewski, M. Nilges, N.S. Pannu, R.J. Read, L.M. Rice, T. Simonson, and G.L. Warren Acta Crystallogr., Sect. D 54 1998 905
29. A. Berezov, H.T. Zhang, M.I. Greene, and R. Murali J. Med. Chem. 44 2001 2565
30. B.W. Park, H.T. Zhang, C. Wu, A. Berezov, X. Zhang, R. Dua, Q. Wang, G. Kao, D.M. O'Rourke, M.I. Greene, and R. Murali Nat. Biotechnol. 18 2001 194
31. Z.M. Bhujwalla, D. Artemov, E. Aboagye, E. Ackerstaff, R.J. Gillies, K. Natarajan, and M. Solaiyappan Novartis Found. Symp. 240 2001 23 discussion 38, 152
32. D.M. Brizel, T. Schroeder, R.L. Scher, S. Walenta, R.W. Clough, M.W. Dewhirst, and W. Mueller-Klieser Int. J. Radiat. Oncol. Biol. Phys. 51 2001 349
33. S.W. Tsai, Y. Sun, L.E. Williams, A.A. Raubitschek, A.M. Wu, and J.E. Shively Bioconjugate Chem. 11 2000 327
34. A.M. Wu, P.J. Yazaki, S. Tsai, K. Nguyen, A.L. Anderson, D.W. McCarthy, M.J. Welch, J.E. Shively, L.E. Williams, A.A. Raubitschek, J.Y. Wong, T. Toyokuni, M.E. Phelps, and S.S. Gambhir Proc. Natl. Acad. Sci. U.S.A. 97 2000 8495
35. K. Nakamura, C. Fan, G. Liu, S. Gupta, J. He, S. Dou, A. Kubo, M. Rusckowski, and D. Hnatowich Bioconjugate Chem. 15 2004 1475
36. S.F. Rosebrough, Z.D. Grossman, J.G. McAfee, B.J. Kudryk, G. Subramanian, C.A. Ritter-Hrncirik, L.S. Witanowski, G. Tillapaugh-Fay, E. Urrutia, and C. Zapf-Longo J. Med. Chem. 29 1988 1212