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Volumn 65, Issue 6, 2011, Pages 467-478

In vitro and in vivo comparison of [ 3H](+)-PHNO and [ 3H]raclopride binding to rat striatum and lobes 9 and 10 of the cerebellum: A method to distinguish dopamine D 3 from D 2 receptor sites: A method to distinguish dopamine D 3 from D 2 receptor sites

Author keywords

3H (+) PHNO; DA D 3 receptor; In vitro binding; In vivo binding; Rat cerebellum

Indexed keywords

DOPAMINE 2 RECEPTOR; DOPAMINE 2 RECEPTOR BLOCKING AGENT; DOPAMINE 3 RECEPTOR; NAXAGOLIDE; NAXAGOLIDE H 3; RACLOPRIDE; RACLOPRIDE H 3; SV 156; UNCLASSIFIED DRUG;

EID: 79953266808     PISSN: 08874476     EISSN: 10982396     Source Type: Journal    
DOI: 10.1002/syn.20867     Document Type: Article
Times cited : (28)

References (43)
  • 1
    • 0028307196 scopus 로고
    • Dopamine receptor distribution in the rat CNS: Elucidation using anti-peptide antisera directed against D1A and D3 subtypes
    • Ariano MA, Sibley DR. 1994. Dopamine receptor distribution in the rat CNS: Elucidation using anti-peptide antisera directed against D1A and D3 subtypes. Brain Res 649: 95-110.
    • (1994) Brain Res , vol.649 , pp. 95-110
    • Ariano, M.A.1    Sibley, D.R.2
  • 2
    • 0031594426 scopus 로고    scopus 로고
    • 3H]PD 128907, a putatively selective ligand for the D3 dopamine receptor, in rat brain: A receptor binding and quantitative autoradiographic study
    • 3H]PD 128907, a putatively selective ligand for the D3 dopamine receptor, in rat brain: A receptor binding and quantitative autoradiographic study. Neuropsychopharmacology 18: 305-316.
    • (1998) Neuropsychopharmacology , vol.18 , pp. 305-316
    • Bancroft, G.N.1    Morgan, K.A.2    Flietstra, R.J.3    Levant, B.4
  • 3
    • 0030597183 scopus 로고    scopus 로고
    • Evidence for a functional role of the dopamine D3 receptors in the cerebellum
    • Barik S, de Beaurepaire R. 1996. Evidence for a functional role of the dopamine D3 receptors in the cerebellum. Brain Res 737: 347-350.
    • (1996) Brain Res , vol.737 , pp. 347-350
    • Barik, S.1    de Beaurepaire, R.2
  • 4
    • 0033955419 scopus 로고    scopus 로고
    • Microanatomical localization of dopamine receptor protein immunoreactivity in the rat cerebellar cortex
    • Barili P, Bronzetti E, Ricci A, Zaccheo D, Amenta F. 2000. Microanatomical localization of dopamine receptor protein immunoreactivity in the rat cerebellar cortex. Brain Res 854: 130-138.
    • (2000) Brain Res , vol.854 , pp. 130-138
    • Barili, P.1    Bronzetti, E.2    Ricci, A.3    Zaccheo, D.4    Amenta, F.5
  • 7
    • 0015861774 scopus 로고
    • Relationship between the inhibition constant (Ki) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction
    • Cheng Y, Prusoff WH. 1973. Relationship between the inhibition constant (Ki) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction. Biochem Pharmacol 22: 3099-3108.
    • (1973) Biochem Pharmacol , vol.22 , pp. 3099-3108
    • Cheng, Y.1    Prusoff, W.H.2
  • 10
    • 0032502365 scopus 로고    scopus 로고
    • 3 dopamine receptor affinity of dopaminergic compounds in rat brain
    • 3 dopamine receptor affinity of dopaminergic compounds in rat brain. Life Sci 62: 1825-1831.
    • (1998) Life Sci , vol.62 , pp. 1825-1831
    • Flietstra, R.J.1    Levant, B.2
  • 13
    • 0034747210 scopus 로고    scopus 로고
    • 3H]R(+)-7-OH-DPAT binding in the rat caudate-putamen
    • 3H]R(+)-7-OH-DPAT binding in the rat caudate-putamen. Neurochem Int 38: 31-42.
    • (2001) Neurochem Int , vol.38 , pp. 31-42
    • Hillefors, M.1    von Euler, G.2
  • 15
    • 0021844076 scopus 로고
    • Specific in vitro and in vivo binding of 3H-raclopride. A potent substituted benzamide drug with high affinity for dopamine D-2 receptors in the rat brain
    • Kohler C, Hall H, Ogren SO, Gawell L. 1985. Specific in vitro and in vivo binding of 3H-raclopride. A potent substituted benzamide drug with high affinity for dopamine D-2 receptors in the rat brain. Biochem Pharmacol 34: 2251-2259.
    • (1985) Biochem Pharmacol , vol.34 , pp. 2251-2259
    • Kohler, C.1    Hall, H.2    Ogren, S.O.3    Gawell, L.4
  • 16
    • 44749090396 scopus 로고    scopus 로고
    • The involvement of cerebellar dopamine D3 receptors in locomotor activity of rats
    • Kolasiewicz W, Maj J, Ossowska K. 2008. The involvement of cerebellar dopamine D3 receptors in locomotor activity of rats. J Neural Transm 115: 677-681.
    • (2008) J Neural Transm , vol.115 , pp. 677-681
    • Kolasiewicz, W.1    Maj, J.2    Ossowska, K.3
  • 17
    • 0030610305 scopus 로고    scopus 로고
    • 3 dopamine receptor: Neurobiology and potential clinical relevance
    • 3 dopamine receptor: Neurobiology and potential clinical relevance. Pharmacol Rev 49: 231-252.
    • (1997) Pharmacol Rev , vol.49 , pp. 231-252
    • Levant, B.1
  • 18
    • 0032479595 scopus 로고    scopus 로고
    • Differential distribution of D3 dopamine receptors in the brains of several mammalian species
    • Levant B. 1998. Differential distribution of D3 dopamine receptors in the brains of several mammalian species. Brain Res 800: 269-274.
    • (1998) Brain Res , vol.800 , pp. 269-274
    • Levant, B.1
  • 19
    • 0027223078 scopus 로고
    • 3H]quinpirole: Identification of a discrete population of putative D3 receptors
    • 3H]quinpirole: Identification of a discrete population of putative D3 receptors. Synapse 14: 90-95.
    • (1993) Synapse , vol.14 , pp. 90-95
    • Levant, B.1    DeSouza, E.B.2
  • 31
    • 0028989321 scopus 로고
    • Localisation of dopamine D3 receptor in the rat cerebellar cortex: A light microscope autoradiographic study
    • Ricci A, Vega JA, Mammola CL, Amenta F. 1995. Localisation of dopamine D3 receptor in the rat cerebellar cortex: A light microscope autoradiographic study. Neurosci Lett 190: 163-166.
    • (1995) Neurosci Lett , vol.190 , pp. 163-166
    • Ricci, A.1    Vega, J.A.2    Mammola, C.L.3    Amenta, F.4
  • 33
    • 0029802407 scopus 로고    scopus 로고
    • Endogenous dopamine limits the binding of antipsychotic drugs to D3 receptors in the rat brain: a quantitative autoradiography study
    • Schotte A, Janssen PF, Bonaventure P, Leysen J. 1996. Endogenous dopamine limits the binding of antipsychotic drugs to D3 receptors in the rat brain: a quantitative autoradiography study. J Histochem 28: 791-799.
    • (1996) J Histochem , vol.28 , pp. 791-799
    • Schotte, A.1    Janssen, P.F.2    Bonaventure, P.3    Leysen, J.4
  • 35
    • 63049115144 scopus 로고    scopus 로고
    • High receptors measured ex vivo are elevated in amphetamine-sensitized animals
    • High receptors measured ex vivo are elevated in amphetamine-sensitized animals. Synapse 63: 186-192.
    • (2009) Synapse , vol.63 , pp. 186-192
    • Seeman, P.1
  • 42
    • 0034783501 scopus 로고    scopus 로고
    • 2 receptor occupancy is a common mechanism underlying animal models of antipsychotics and their clinical effects
    • 2 receptor occupancy is a common mechanism underlying animal models of antipsychotics and their clinical effects. Neuropsychopharmacology 25: 633-641.
    • (2001) Neuropsychopharmacology , vol.25 , pp. 633-641
    • Wadenberg, M.L.1    Soliman, A.2    VanderSpek, S.C.3    Kapur, S.4
  • 43
    • 0028980498 scopus 로고
    • 3H]propyl-2-aminotetralin and carbetapentane
    • 3H]propyl-2-aminotetralin and carbetapentane. J Neurochem 64: 700-710.
    • (1995) J Neurochem , vol.64 , pp. 700-710
    • Wallace, D.R.1    Booze, R.M.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.