SCOPUS 정보 검색 플랫폼

Volumn 46, Issue 5, 2011, Pages 1841-1848

Preparation and evaluation of tetrabenazine enantiomers and all eight stereoisomers of dihydrotetrabenazine as VMAT2 inhibitors

(7) Yao, Zhangyu a Wei, Xueying a Wu, Xiaoming a Katz, Jonathan L b Kopajtic, Theresa b Greig, Nigel H c Sun, Hongbin a

a CHINA PHARMACEUTICAL UNIVERSITY (China)

b NATIONAL INSTITUTE ON DRUG ABUSE (United States)

c NATIONAL INSTITUTE ON AGING (United States)

Author keywords

Dihydrotetrabenazine stereoisomers; Huntington's chorea; Hyperkinetic disorders; Resolution; Tetrabenazine enantiomers; VMAT2

Indexed keywords

3 ISOBUTYL 9,10 DIMETHOXY 1,3,4,6,7,11B HEXAHYDRO 2H PYRIDO[2,1 A]ISOQUINOLIN 2 OL; DIHYDROTETRABENAZINE; TETRABENAZINE; UNCLASSIFIED DRUG; VESICULAR MONOAMINE TRANSPORTER 2;

ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; BINDING ASSAY; DRUG PROTEIN BINDING; DRUG STRUCTURE; DRUG SYNTHESIS; ENANTIOMER; MALE; NONHUMAN; RAT; STEREOCHEMISTRY; STEREOISOMERISM; STRUCTURE ACTIVITY RELATION;

ANIMALS; MALE; MOLECULAR CONFORMATION; RATS; RATS, SPRAGUE-DAWLEY; STEREOISOMERISM; STRUCTURE-ACTIVITY RELATIONSHIP; TETRABENAZINE; VESICULAR MONOAMINE TRANSPORT PROTEINS;

EID: 79953189647 PISSN: 02235234 EISSN: 17683254 Source Type: Journal
DOI: 10.1016/j.ejmech.2011.02.046 Document Type: Article

Times cited : (46)

References (23)

1
- 84981836927
- A. Brossi, H. Lindlar, M. Walter, and O. Schnider Helv. Chim. Acta 41 1958 119 139
- (1958) Helv. Chim. Acta , vol.41 , pp. 119-139
- Brossi, A.¹ Lindlar, H.² Walter, M.³ Schnider, O.⁴

2
- 68249146267
- J. Jankovic Lancet Neurol. 8 2009 844 856
- (2009) Lancet Neurol. , vol.8 , pp. 844-856
- Jankovic, J.¹

3
- 18944378746
- Y.S. Silay, and J. Jankovic Expert Opin. Emerg. Drugs 10 2005 365 380
- (2005) Expert Opin. Emerg. Drugs , vol.10 , pp. 365-380
- Silay, Y.S.¹ Jankovic, J.²

4
- 0013904103
- D.E. Schwartz, H. Bruderer, J. Rieder, and A. Brossi Biochem. Pharmacol. 15 1966 645 655
- (1966) Biochem. Pharmacol. , vol.15 , pp. 645-655
- Schwartz, D.E.¹ Bruderer, H.² Rieder, J.³ Brossi, A.⁴

5
- 0022647428
- M.S. Roberts, S. McLean, K.S. Millingen, and H.M. Galloway Eur. J. Clin. Pharmacol. 29 1986 703 708
- (1986) Eur. J. Clin. Pharmacol. , vol.29 , pp. 703-708
- Roberts, M.S.¹ McLean, S.² Millingen, K.S.³ Galloway, H.M.⁴

6
- 73149122141
- A. Fasano, and A.R. Bentivoglio Expert Opin. Pharmacother. 10 2009 2883 2896
- (2009) Expert Opin. Pharmacother. , vol.10 , pp. 2883-2896
- Fasano, A.¹ Bentivoglio, A.R.²

7
- 0023856687
- D. Scherman, B. Gasnier, P. Jaudon, and J.P. Henry Mol. Pharmacol. 33 1988 72 77
- (1988) Mol. Pharmacol. , vol.33 , pp. 72-77
- Scherman, D.¹ Gasnier, B.² Jaudon, P.³ Henry, J.P.⁴

8
- 0000431640
- A. Pletscher, A. Brossi, and K.F. Gey Int. Rev. Neurobiol. 4 1962 275 306
- (1962) Int. Rev. Neurobiol. , vol.4 , pp. 275-306
- Pletscher, A.¹ Brossi, A.² Gey, K.F.³

9
- 72249105289
- A.P. Vartak, J.R. Nickell, J. Chagkutip, L.P. Dwoskin, and P.A. Crooks J. Med. Chem. 52 2009 7878 7882
- (2009) J. Med. Chem. , vol.52 , pp. 7878-7882
- Vartak, A.P.¹ Nickell, J.R.² Chagkutip, J.³ Dwoskin, L.P.⁴ Crooks, P.A.⁵

10
- 0028990225
- M. Kilbourn, L. Lee, T.V. Borght, D.M. Jewett, and K. Frey Eur. J. Pharmacol. 278 1995 249 252
- (1995) Eur. J. Pharmacol. , vol.278 , pp. 249-252
- Kilbourn, M.¹ Lee, L.² Borght, T.V.³ Jewett, D.M.⁴ Frey, K.⁵

11
- 0030969697
- M.R. Kilbourn, L.C. Lee, M.J. Heeg, and D.M. Jewett Chirality 9 1997 59 62
- (1997) Chirality , vol.9 , pp. 59-62
- Kilbourn, M.R.¹ Lee, L.C.² Heeg, M.J.³ Jewett, D.M.⁴

12
- 6744226921
- M.R. Kilbourn, L.C. Lee, D.M. Jewett, R.A. Koeppe, and K.A. Frey J. Cereb. Blood Flow Metab. 15 1995 S650
- (1995) J. Cereb. Blood Flow Metab. , vol.15 , pp. 650
- Kilbourn, M.R.¹ Lee, L.C.² Jewett, D.M.³ Koeppe, R.A.⁴ Frey, K.A.⁵

13
- 79953188429
- K.W. Gano PCT patent application: WO2008058261 2008
- (2008) PCT Patent Application: WO2008058261
- Gano, K.W.¹

14
- 79953196948
- I. Clarke, R. Turtle, and G. Johnston PCT patent application: WO2005077946 2005
- (2005) PCT Patent Application: WO2005077946
- Clarke, I.¹ Turtle, R.² Johnston, G.³

15
- 65949095007
- M.J. Rishel, K.K.D. Amarasinghe, S.R. Dinn, and B.F. Johnson J. Org. Chem. 74 2009 4001 4004
- (2009) J. Org. Chem. , vol.74 , pp. 4001-4004
- Rishel, M.J.¹ Amarasinghe, K.K.D.² Dinn, S.R.³ Johnson, B.F.⁴

16
- 70349195185
- K.G. Boldt, M.S. Biggers, S.S. Phifer, G.A. Brine, and K.S. Rehder Synth. Commun. 39 2009 3574 3585
- (2009) Synth. Commun. , vol.39 , pp. 3574-3585
- Boldt, K.G.¹ Biggers, M.S.² Phifer, S.S.³ Brine, G.A.⁴ Rehder, K.S.⁵

17
- 77956639647
- Q.S. Yu, W.M. Luo, J. Deschamps, H.W. Holloway, T. Kopajtic, J.L. Katz, A. Brossi, and N.H. Greig Med. Chem. Lett. 1 2010 105 109
- (2010) Med. Chem. Lett. , vol.1 , pp. 105-109
- Yu, Q.S.¹ Luo, W.M.² Deschamps, J.³ Holloway, H.W.⁴ Kopajtic, T.⁵ Katz, J.L.⁶ Brossi, A.⁷ Greig, N.H.⁸

18
- 79953229291
- H.B. Sun, and Z.Y. Yao Chinese patent application: 2009100318475 2009
- (2009) Chinese Patent Application: 2009100318475
- Sun, H.B.¹ Yao, Z.Y.²

19
- 55549125242
- H.T. Openshaw, and N. Whittaker J. Chem. Soc. 1963 1449 1460
- (1963) J. Chem. Soc. , pp. 1449-1460
- Openshaw, H.T.¹ Whittaker, N.²

20
- 12344278391
- H.T. Openshaw, and N. Whittaker J. Chem. Soc. 1963 1461 1471
- (1963) J. Chem. Soc. , pp. 1461-1471
- Openshaw, H.T.¹ Whittaker, N.²

21
- 0030029369
- L.C. Lee, T.V. Borght, P.S. Sherman, K.A. Frey, and M.R. Kilbourn J. Med. Chem. 39 1996 191 196
- (1996) J. Med. Chem. , vol.39 , pp. 191-196
- Lee, L.C.¹ Borght, T.V.² Sherman, P.S.³ Frey, K.A.⁴ Kilbourn, M.R.⁵

22
- 0000995704
- H.C. Brown, and N.M. Moon J. Am. Chem. Soc. 90 1968 2686 2688
- (1968) J. Am. Chem. Soc. , vol.90 , pp. 2686-2688
- Brown, H.C.¹ Moon, N.M.²

23
- 0001254173
- W.B. Smith J. Org. Chem. 49 1984 3219 3220
- (1984) J. Org. Chem. , vol.49 , pp. 3219-3220
- Smith, W.B.¹

* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.