Microwave assisted one-pot synthesis of highly potent novel isoniazid analogues

Bioorganic and Medicinal Chemistry Letters

Volumn 21, Issue 7, 2011, Pages 2125-2128

  Manjashetty, Thimmappa H ^a   Yogeeswari, Perumal ^a   Sriram, Dharmarajan ^a  

^a BIRLA INSTITUTE OF TECHNOLOGY AND SCIENCE   (India)

Author keywords

Anti TB activity; Antimycobacterial activity; Isoniazid derivative; MDR TB

Indexed keywords

ISONIAZID DERIVATIVE; N [9 [2 (BENZYLOXY)PHENYL] 3,3,6,6 TETRAMETHYL 1,8 DIOXO 2,3,4,5,6,7,8,9 OCTAHYDRO 10[1H]ACRIDINYL]ISONICOTINAMIDE; UNCLASSIFIED DRUG;

ANTIBACTERIAL ACTIVITY; ARTICLE; BACTERIAL STRAIN; CATALYSIS; CYTOTOXICITY; DRUG DETERMINATION; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS; MICROWAVE IRRADIATION; MINIMUM INHIBITORY CONCENTRATION; MYCOBACTERIUM TUBERCULOSIS; NONHUMAN; ONE POT SYNTHESIS;

ANIMALS; ANTITUBERCULAR AGENTS; CERCOPITHECUS AETHIOPS; ISONIAZID; MICROBIAL SENSITIVITY TESTS; MICROWAVES; MYCOBACTERIUM TUBERCULOSIS; VERO CELLS;

MYCOBACTERIUM TUBERCULOSIS;

EID: 79952488137     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2011.01.122     Document Type: Article

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