-
1
-
-
0003593740
-
Aminothiazoles and their derivatives
-
Metzger, J. V., Ed.; Wiley: New York
-
Barone, R.; Chanon, M.; Gallo, R. Aminothiazoles and their derivatives. In: The Chemistry of Heterocyclic Compounds, Part 2; Metzger, J. V., Ed.; Wiley: New York, 1979; Vol. 34, pp. 9-368.
-
(1979)
The Chemistry of Heterocyclic Compounds Part 2
, vol.34
, pp. 9-368
-
-
Barone, R.1
Chanon, M.2
Gallo, R.3
-
2
-
-
67651047153
-
Progress in the development of nonpeptidometic BACE 1 inhibitors for Alzheimer's disease
-
Huang, W.H.; Sheng, R.; Hu, Y.Z. Progress in the development of nonpeptidometic BACE 1 inhibitors for Alzheimer's disease. Curr. Med. Chem., 2009, 16(14), 1806-1820.
-
(2009)
Curr. Med. Chem.
, vol.16
, Issue.14
, pp. 1806-1820
-
-
Huang, W.H.1
Sheng, R.2
Hu, Y.Z.3
-
3
-
-
66449112479
-
Voltage-gated sodium channel blockers for the treatment of chronic pain
-
Matulenko, M.A.; Scanio, M.J.C.; Kort, M.E. Voltage-gated sodium channel blockers for the treatment of chronic pain. Curr. Top. Med. Chem., 2009, 9(4), 362-376.
-
(2009)
Curr. Top. Med. Chem.
, vol.9
, Issue.4
, pp. 362-376
-
-
Matulenko, M.A.1
Scanio, M.J.C.2
Kort, M.E.3
-
4
-
-
52049097040
-
Progress in the evaluation of CDK inhibitors as antitumor agents
-
McInnes, C. Progress in the evaluation of CDK inhibitors as antitumor agents. Drug Discov. Today, 2008, 13(19-20), 875-881.
-
(2008)
Drug Discov. Today
, vol.13
, Issue.19-20
, pp. 875-881
-
-
McInnes, C.1
-
5
-
-
51049090179
-
Drug discovery and development for Huntington's disease - An orphan indication with high medical need
-
Heitz, F.; La Rosa, S.; Gonzalez-Couto, E.; Gaviraghi, G.; Terstappen, G.C. Drug discovery and development for Huntington's disease - An orphan indication with high medical need. IDrugs, 2008, 11(9), 653-660.
-
(2008)
IDrugs
, vol.11
, Issue.9
, pp. 653-660
-
-
Heitz, F.1
La Rosa, S.2
Gonzalez-Couto, E.3
Gaviraghi, G.4
Terstappen, G.C.5
-
7
-
-
33746317072
-
Aminothiazole derivatives as neuropeptide Y5 receptor ligands: Finding the balance between affinity and physicochemical properties
-
DOI 10.1002/cmdc.200500022
-
Nettekoven, M.; Guba, W.; Neidhart, W.; Mattei, P.; Pflieger, P.; Plancher, J.M.; Taylor, S. Aminothiazole derivatives as neuropeptide Y5 receptor ligands: finding the balance between affinity and physicochemical properties. ChemMedChem, 2006, 1(1), 45-48. (Pubitemid 44104974)
-
(2006)
ChemMedChem
, vol.1
, Issue.1
, pp. 45-48
-
-
Nettekoven, M.1
Guba, W.2
Neidhart, W.3
Mattei, P.4
Pflieger, P.5
Plancher, J.-M.6
Taylor, S.7
-
8
-
-
21144443385
-
3 selective antagonists, through solution-phase parallel synthesis
-
DOI 10.1248/cpb.53.437
-
Sagara, Y.; Mitsuya, M.; Uchiyama, M.; Ogino, Y.; Kjmura, T.; Ohtake, N.; Mase, T. Discovery of 2-aminothiazole-4- carboxamides, a novel class of muscarinic M3 selective antagonists, through solution-phase parallel synthesis. Chem. Pharm. Bull., 2005, 53(4), 437-440. (Pubitemid 40879887)
-
(2005)
Chemical and Pharmaceutical Bulletin
, vol.53
, Issue.4
, pp. 437-440
-
-
Sagara, Y.1
Mitsuya, M.2
Uchiyama, M.3
Ogino, Y.4
Kjmura, T.5
Ohtake, N.6
Mase, T.7
-
9
-
-
18244391461
-
Solution-phase synthesis of a combinatorial library of 3-[4-(coumarin-3-yl) -1,3-thiazol-2-ylcarbamoyl]propanoic acid amides
-
Zhuravel, I.O.; Kovalenko, S.M.; Vlasov, S.V.; Chernykh, V.P. Solution-phase synthesis of a combinatorial library of 3-[4-(coumarin-3-yl)-1,3- thiazol-2- ylcarbamoyl]propanoic acid amides. Molecules, 2005, 10(2)444-456. (Pubitemid 40632787)
-
(2005)
Molecules
, vol.10
, Issue.2
, pp. 444-456
-
-
Zhuravel, I.O.1
Kovalenko, S.M.2
Vlasov, S.V.3
Chernykh, V.P.4
-
10
-
-
0030008667
-
A convenient procedure for the solution phase preparation of 2-aminothiazole combinatorial libraries
-
Bailey, N.; Dean, A.W.; Judd, D.B.; Middlemiss, D.; Storer, R.; Watson, S.P. A convenient procedure for the solution phase preparation of 2-aminothiazole combinatorial libraries. Bioorg. Med. Chem. Lett., 1996, 6(12), 1409-1414.
-
(1996)
Bioorg. Med. Chem. Lett.
, vol.6
, Issue.12
, pp. 1409-1414
-
-
Bailey, N.1
Dean, A.W.2
Judd, D.B.3
Middlemiss, D.4
Storer, R.5
Watson, S.P.6
-
11
-
-
0000196260
-
Clean synthesis of α-bromo ketones and their utilisation in the synthesis of 2-alkoxy-2,3-dihydro-2-aryl-1,4- benzodioxanes, 2-amino-4-aryl-1,3-thiazoles and piperidino-2- amino-1,3-thiazoles using polymer-supported reagents
-
Habermann, J.; Ley, S.V.; Scicinski, J.J.; Scott, J.S.; Smits, R.; Thomas, A.W. Clean synthesis of α-bromo ketones and their utilisation in the synthesis of 2-alkoxy-2,3-dihydro-2-aryl-1,4- benzodioxanes, 2-amino-4-aryl-1,3-thiazoles and piperidino-2- amino-1,3-thiazoles using polymer-supported reagents. J. Chem. Soc. Perkin Trans., 1999, 1, 2425-2427.
-
(1999)
J. Chem. Soc. Perkin Trans.
, vol.1
, pp. 2425-2427
-
-
Habermann, J.1
Ley, S.V.2
Scicinski, J.J.3
Scott, J.S.4
Smits, R.5
Thomas, A.W.6
-
12
-
-
0033980150
-
Streamlined synthesis of substituted 2-aminothiazoles using tandem precipitative and polymer-assisted reactions
-
DOI 10.1002/(SICI)1097-0290(200024)71:1<9::AID-BIT3>3.0.CO;2-#
-
Yun, Y.K.; Leung, S.S.W. ; Porco Jr., J.A. Streamlined synthesis of substituted 2-aminothiazoles using tandem precipitative and polymer-assisted reactions. Biotechnol. Bioeng., 2000, 71(1), 9-18. (Pubitemid 30077812)
-
(2000)
Biotechnology and Bioengineering
, vol.71
, Issue.1
, pp. 9-18
-
-
Yun, Y.K.1
Leung, S.S.W.2
Porco Jr., J.A.3
-
13
-
-
33744991792
-
Microwave promoted synthesis of functionalized 2-aminothiazoles
-
DOI 10.1016/j.tetlet.2006.05.053, PII S0040403906009786
-
Kabalka, G.W., Mereddy, A.R. Microwave promoted synthesis of functionalized 2-aminothiazoles. Tetrahedron Lett., 2006, 47(29), 5171-5172. (Pubitemid 43867606)
-
(2006)
Tetrahedron Letters
, vol.47
, Issue.29
, pp. 5171-5172
-
-
Kabalka, G.W.1
Mereddy, A.R.2
-
14
-
-
79751480257
-
-
www.chemspeed.com
-
-
-
-
15
-
-
0030767571
-
Polymer supported bases in combinatorial chemistry: Synthesis of aryl ethers from phenols and alkyl halides and aryl halides
-
DOI 10.1016/S0040-4039(97)01782-6, PII S0040403997017826
-
Xu, W.; Mohan, R.; Morrissey, M.M. Polymer supported bases in combinatorial chemistry: Synthesis of aryl ethers from phenols and alkyl halides and aryl halides. Tetrahedron Lett., 1997, 38(42), 7337-7340. (Pubitemid 27435124)
-
(1997)
Tetrahedron Letters
, vol.38
, Issue.42
, pp. 7337-7340
-
-
Xu, W.1
Mohan, R.2
Morrissey, M.M.3
|