Development of the route of manufacture of an oral H1-H 3 antagonist

Organic Process Research and Development

Volumn 15, Issue 1, 2011, Pages 112-122

  Bret, Guillaume ^a   Harling, Sandra J ^a   Herbal, Karim ^a   Langlade, Nathalie ^a   Loft, Mike ^a   Negus, Alan ^a   Sanganee, Mahesh ^a   Shanahan, Steve ^a   Strachan, John B ^a   Turner, Peter G ^a   Whiting, Matthew P ^a  

^a GLAXOSMITHKLINE   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

COST-OF-GOODS;

EID: 79251520296     PISSN: 10836160     EISSN: 1520586X     Source Type: Journal    
DOI: 10.1021/op1002598     Document Type: Article

References (10)

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4. Krasovskiy, A.; Knochel, P. Angew. Chem. Int. Ed 2004, 43, 3333 and references therein
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9. For related observations: Boros, E. E.; Burova, S. A.; Erickson, G. A.; Johns, B. A.; Koble, C. S.; Kurose, N.; Sharp, M. J.; Tabet, E. A.; Thompson, J. B.; Toczko, M. A. Org. Process Res. Dev. 2007, 11, 899-902
10. Krasovskiy, A.; Straub, B.; Knochel, P. Angew. Chem., Int. Ed. 2006, 45, 159