Decoding powder tabletability: Roles of particle adhesion and plasticity

Journal of Adhesion Science and Technology

Volumn 25, Issue 4-5, 2011, Pages 483-499

  Sun, Changquan Calvin ^a  

^a UNIVERSITY OF MINNESOTA   (United States)

Author keywords

adhesion; bonding area; bonding strength; plastic deformation; Powder compaction; surface energy; tabletability

Indexed keywords

BONDING STRENGTH; CHEMICAL NATURE; DEFORMATION MECHANISM; HIGH QUALITY; INTERFACIAL ADHESIONS; MANUFACTURING PROCESS; MECHANICAL AND PHYSICAL PROPERTIES; MECHANICAL STRENGTH; PARTICLE ADHESION; PARTICLE SIZE AND SHAPE; PHARMACEUTICAL INDUSTRY; POWDER COMPACTION; POWDER COMPACTIONS; QUALITATIVE MODEL; SURFACE ENERGY; TABLETABILITY;

ADHESION; CHEMICAL ANALYSIS; COMPACTION; DIFFUSION BONDING; INTERFACIAL ENERGY; MANUFACTURE; MECHANICAL PROPERTIES; PLASTIC DEFORMATION; PRODUCT DEVELOPMENT; SURFACE CHEMISTRY;

IMPACT STRENGTH;

EID: 78751665525     PISSN: 01694243     EISSN: 15685616     Source Type: Journal    
DOI: 10.1163/016942410X525678     Document Type: Article

References (62)

1. B. B. Sheth, F. J. Bandelin and R. F. Shangraw, in: Pharmaceutical Dosage Forms: Tablets, H. A. Lieberman and L. Lachman (Eds), pp. 109-185. Marcel Dekker, New York, NY (1980).
2. H. Leuenberger and M. Lanz, Advanced Powder Technol. 16, 3-25 (2005).
3. FDA Report, Critical path opportunities for generic drugs, http://www.fda.gov/oc/initiatives/ criticalpath/reports/generic.html (2007).
4. C. C. Sun, J. Pharm. Sci. 98, 1671-1687 (2009).
5. E. Joiris, P. Di Martine, C. Berneron, A. M. Guyot-Hermann and J. C. Guyot, Pharm. Res. 15, 1122-1130 (1998).
6. C. C. Sun and D. J. W. Grant, Pharm. Res. 18, 274-280 (2001).
7. C. K. Tye, C. C. Sun and G. E. Amidon, J. Pharm. Sci. 94, 465-472 (2005).
8. A. C. Shah and A. R. Mlodozeniec, J. Pharm. Sci. 66, 1377-1382 (1977).
9. F. Khan, N. Pilpel and S. Ingram, Powder Technol. 54, 161-164 (1988).
10. G. E. Amidon and M. E. Houghton, Pharm. Res. 12, 923-929 (1995).
11. A. Gupta, G. E. Peck, R. W. Miller and K. R. Morris, J. Pharm. Sci. 94, 2301-2313 (2005).
12. C. C. Sun, Int. J. Pharm. 346, 93-101 (2008).
13. H. G. Ibrahim, F. Pisano and A. Bruno, J. Pharm. Sci. 66, 669-673 (1977).
14. A. Burger, J.-O. Henck, S. Hetz, J. M. Rollinger, A. A. Weissnicht and H. Stöttner, J. Pharm. Sci. 89, 457-468 (2000).
15. J. A. Hersey, G. Bayraktar and E. Shotton, J. Pharm. Pharmacol. 19 (Suppl.), 24S-30S (1967).
16. C. C. Sun and D. J. W. Grant, Int. J. Pharm. 215, 221-228 (2001).
17. H. Nicklasson and F. Podczeck, Chem. Pharm. Bull. 55, 29-33 (2007).
18. C. C. Sun and M. W. Himmelspach, J. Pharm. Sci. 95, 200-206 (2006).
19. G. Alderborn and C. Nyström, Acta Pharm. Suec. 19, 381-390 (1982).
20. S. J. Wu and C. C. Sun, J. Pharm. Sci. 96, 1445-1450 (2007).
21. C. C. Sun, H. Hou, P. Gao, C. Ma, C. Medina and P. Alvarez, J. Pharm. Sci. 98, 239-247 (2009).
22. T. Higuchi, A. N. Rao, L. W. Busse and J. V. Swintosky, J. Am. Pharm. Assoc. (Sci. Ed.) 42, 194-200 (1953).
23. T. Higuchi, T. Shimamoto, S. P. Eriksen and I. Yashiki, J. Pharm. Sci. 54, 111-118 (1965).
24. S. W. Hoag and E. G. Rippie, J. Pharm. Sci. 83, 903-908 (1994).
25. D. V. Moe and E. G. Rippie, J. Pharm. Sci. 86, 26-32 (1997).
26. E. Nelson, W. Bussel and T. Higuchi, J. Am. Pharm. Assoc. (Sci. Ed.) 44, 223-225 (1955).
27. E. N. Hiestand, Int. J. Pharm. 67, 217-229 (1991).
28. C. Nyström and P.-G. Karehill, in: Pharmaceutical Powder Compaction Technology, G. Alderborn and C. Nyström (Eds), pp. 17-53. Marcel Dekker, New York, NY (1996).
29. E. N. Hiestand, J. Pharm. Sci. 74, 768-770 (1985).
30. K. Kendall, Science 263, 1720-1725 (1994).
31. P. E. Wray, Drug Dev. Ind. Pharm. 18, 627-657 (1992).
32. W. Flugge, Viscoelasticity, 2nd ed. Springer-Verlag, New York, NY (1975).
33. J. T. Fell and J. M. Newton, J. Pharm. Sci. 59, 688-691 (1970).
34. Y. Urahama, J. Adhesion 31, 47-58 (1989).
35. A. A. Griffith, Philosophical Trans. Royal Society (London) A221, 163-198 (1920).
36. D. Farkas, MRS Bulletin 25, 35-38 (2000).
37. J. M. Newton, G. Rowley, J. T. Fell, D. G. Peacock and K. Ridgway, J. Pharm. Pharmacol. 23 (Suppl.), 195S-201S (1971).
38. J. M. Newton, G. Rowley and J. T. Fell, J. Pharm. Pharmacol. 24, 503-504 (1972).
39. K. G. Pitt, J. M. Newton, R. Richardson and P. Stanley, J. Pharm. Pharmacol. 41, 289-292 (1989).
40. P. Stanley and J. M. Newton, J. Pharm. Pharmacol. 32, 852-854 (1980).
41. E. N. Hiestand and D. P. Smith, Powder Technol. 38, 145-159 (1984).
42. A. J. Durelli and W. F. Riley, Introduction to Photomechanics. Prentice-Hall, Englewood Cliffs, NJ (1965).
43. C. C. Sun, J. Pharm. Sci. 94, 2132-2334 (2005).
44. E. N. Hiestand, J. Pharm. Sci. 86, 985-990 (1997).
45. J. N. Coleman, U. Khan, W. J. Blau and Y. K. Gun'ko, Carbon 44, 1624-1652 (2006).
46. C. C. Sun, Int. J. Pharm. 347, 171-172 (2008).
47. E. Ryshkewitch, J. Am. Ceram. Soc. 36, 65-68 (1953).
48. C. C. Sun, J. Pharm. Sci. 94, 2061-2068 (2005).
49. C. C. Sun and D. J. W. Grant, Pharm. Res. 21, 382-386 (2004).
50. S. Malkowska and K. A. Khan, Drug Dev. Ind. Pharm. 9, 331-347 (1983).
51. W. A. Strickland, E. Nelson, L.W. Busse and T. Higuchi, J. Am. Pharm. Assoc. Sci. Ed. 45, 51-55 (1956).
52. A. H. De Boer, G. K. Bolhuis and C. F. Lerk, Powder Technol. 20, 75-82 (1978).
53. H. Vromans and C. F. Lerk, Int. J. Pharm. 46, 183-192 (1988).
54. C. C. Sun and D. J. W. Grant, Pharm. Res. 18, 281-286 (2001).
55. W. C. Oliver and G. M. Pharr, J. Mater. Res. 7, 1564-1583 (1992).
56. X. Liao and T. S. Wiedmann, J. Pharm. Sci. 94, 79-92 (2005).
57. V. M. Masterson and X. Cao, Int. J. Pharm. 362, 163-171 (2008).
58. C. C. Sun, Int. J. Pharm. 326, 94-99 (2006).
59. C. C. Sun and H. Hou, Crystal Growth & Design 8, 1575-1579 (2008).
60. S. Karki, T. Friščíc, L. Fábián, P. R. Laity, G. M. Day and W. Jones, Adv. Mater. 21, 3905-3909 (2009).
61. E. Joiris, P. Di Martino, L. Malaj, R. Censi, C. Barthelemy and P. Odou, European J. Pharmaceutics Biopharmaceutics 70, 345-356 (2008).
62. L. Shi and C. C. Sun, J. Pharm. Sci., DOI: 10.1002/jps.22172 (2010).