Synthesis and characterization of [3H]-SN56, a novel radioligand for the σ1 receptor

European Journal of Pharmacology

Volumn 653, Issue 1-3, 2011, Pages 1-7

  Fishback, James A ^a,b   Mesangeau, Christophe ^b   Poupaert, Jacques H ^c   McCurdy, Christopher R ^b   Matsumoto, Rae R ^a,b  

^a WEST VIRGINIA UNIVERSITY   (United States)

^b UNIVERSITY OF MISSISSIPPI   (United States)

^c UNIVERSITÉ CATHOLIQUE DE LOUVAIN   (Belgium)

Author keywords

Receptor; Radioligand binding assay

Indexed keywords

PENTAZOCINE; RADIOLIGAND; SIGMA 1 OPIATE RECEPTOR; TRITIUM 3 [2 (AZEPAN 1 YL)ETHYL] 6 PROPYLBENZO[D]THIAZOL 2(3H)ONE; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; BINDING ASSAY; BINDING COMPETITION; BINDING KINETICS; BINDING SITE; CONTROLLED STUDY; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; IN VITRO STUDY; MALE; NONHUMAN; PRIORITY JOURNAL; RAT;

ANIMALS; AZEPINES; BENZOTHIAZOLES; BINDING SITES; BRAIN; MALE; PENTAZOCINE; PROTEIN BINDING; RADIOLIGAND ASSAY; RADIOPHARMACEUTICALS; RATS; RATS, SPRAGUE-DAWLEY; RECEPTORS, SIGMA;

EID: 78651515142     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.ejphar.2010.10.099     Document Type: Article

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