A Novel 3-(8-Chloro-6-(trifluoromethyl)imidazo[1,2-a]pyridine-2-yl)phenyl acetate skeleton and pharmacophore model as glucagon-like peptide 1 receptor agonists

Bulletin of the Korean Chemical Society

Volumn 31, Issue 12, 2010, Pages 3760-3764

  Gong, Young Dae ^a   Cheon, Hyae Gyeong ^b   Lee, Taeho ^c   Kang, Nam Sook ^c  

^a Dongguk University   (South Korea)

^b Gachon University College of Medicine   (South Korea)

^c Korea Research Institute of Chemical Technology   (South Korea)

Author keywords

Druglike ore skeleton; Glucagon like peptide 1 receptor (GLP 1R); Imidazo 1,2 a pyridine 2 yl phenyl acetate; Pharmacophore

Indexed keywords

MOLECULES; MUSCULOSKELETAL SYSTEM; PEPTIDES; PHARMACODYNAMICS;

DRUGLIKE ORE SKELETON; GLUCAGON-LIKE PEPTIDE-1; IMIDAZO[1 ,2-A]PYRIDINE; PHARMACOPHORE MODELING; PHARMACOPHORES; PHENYL ACETATE; THERAPEUTIC POTENTIALS; TRIFLUOROMETHYL;

PYRIDINE;

EID: 78650399197     PISSN: 02532964     EISSN: 12295949     Source Type: Journal    
DOI: 10.5012/bkcs.2010.31.12.3755     Document Type: Article

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