Anti-leishmanial and anti-trypanosomal activities of 1,4-dihydropyridines: In vitro evaluation and structure-activity relationship study

Bioorganic and Medicinal Chemistry

Volumn 18, Issue 22, 2010, Pages 8044-8053

  Reimão, Juliana Q ^a   Scotti, Marcus T ^b   Tempone, André G ^a  

^a INSTITUTO ADOLFO LUTZ   (Brazil)

^b FEDERAL UNIVERSITY OF PARAÍBA   (Brazil)

Author keywords

1,4 Dihydropyridines; Leishmania; QSAR; Trypanosoma cruzi

Indexed keywords

AMLODIPINE; AZELNIDIPINE; CALCIUM CHANNEL BLOCKING AGENT; CILNIDIPINE; LERCANIDIPINE; NICARDIPINE; NIFEDIPINE; NIMODIPINE; NITRENDIPINE;

ANTIPROTOZOAL ACTIVITY; ARTICLE; CHAGAS DISEASE; CYTOTOXICITY; IC 50; IN VITRO STUDY; LEISHMANIA; LEISHMANIA BRAZILIENSIS; LEISHMANIA CHAGASI; LEISHMANIA MAJOR; LEISHMANIASIS; NONHUMAN; PROMASTIGOTE; QUANTITATIVE STRUCTURE ACTIVITY RELATION; TRYPANOSOMA CRUZI;

ANIMALS; ANTIPROTOZOAL AGENTS; CELL LINE; CRICETINAE; DIHYDROPYRIDINES; ERYTHROCYTES; LEISHMANIA; MACACA MULATTA; MICE; PARASITIC SENSITIVITY TESTS; QUANTITATIVE STRUCTURE-ACTIVITY RELATIONSHIP; STRUCTURE-ACTIVITY RELATIONSHIP; TRYPANOCIDAL AGENTS; TRYPANOSOMA CRUZI;

LEISHMANIA AMAZONENSIS; LEISHMANIA BRAZILIENSIS; LEISHMANIA DONOVANI CHAGASI; LEISHMANIA MAJOR; MAMMALIA; PROTOZOA; TRYPANOSOMA CRUZI;

EID: 78449241052     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2010.09.015     Document Type: Article

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