-
1
-
-
0023929951
-
Structure-activity profile of a series of novel triazoloquinazoline adenosine antagonists
-
Francis, J.E.; Cash, W.D.; Psychoyos, S.; Ghai, G.; Wenk, P.; Friedmann, R.C.; Atkins, C.; Warren, V.; Furness, P.; Hyun, T.L.; Stone, G.A.; Desai, M.; Williams, M. Structure-activity profile of a series of novel triazoloquinazoline adenosine antagonists. J. Med. Chem. 1988, 31, 1014-1020.
-
(1988)
J. Med. Chem.
, vol.31
, pp. 1014-1020
-
-
Francis, J.E.1
Cash, W.D.2
Psychoyos, S.3
Ghai, G.4
Wenk, P.5
Friedmann, R.C.6
Atkins, C.7
Warren, V.8
Furness, P.9
Hyun, T.L.10
Stone, G.A.11
Desai, M.12
Williams, M.13
-
2
-
-
0031824990
-
Derivatives of the triazoloquinazoline adenosine antagonist (CGS15943) having high potency at the human A2B and A3 receptor subtypes
-
Kim, Y.C.; Zwart, M.De; Chang, L.; Moro, S.; Kuenzel, J.; Melman, N.; Jzerman, A.P.; Jacobson, K.A. Derivatives of the triazoloquinazoline adenosine antagonist (CGS15943) having high potency at the human A2B and A3 receptor subtypes. J. Med. Chem. 1998, 41, 2835-2845.
-
(1998)
J. Med. Chem.
, vol.41
, pp. 2835-2845
-
-
Kim, Y.C.1
Zwart, M.D.2
Chang, L.3
Moro, S.4
Kuenzel, J.5
Melman, N.6
Jzerman, A.P.7
Jacobson, K.A.8
-
3
-
-
0025979697
-
Synthesis and benzodiazepine binding activity of a series of novel [1,2,4]triazolo[1,5-c]quinazolin-5(6H)-ones
-
Francis, J.E.; Cash, W.D.; Barbaz, B.S.; Bernard, P.S.; Lovell, R.A.; Mazzenga, G.C.; Friedmann, R.C.; Hyun, J.L.; Braunwalder, A.F.; Loo, P.S.; Bennett, D.A. Synthesis and benzodiazepine binding activity of a series of novel [1,2,4]triazolo[1,5-c]quinazolin-5(6H)-ones. J. Med. Chem. 1991, 34, 281-290.
-
(1991)
J. Med. Chem.
, vol.34
, pp. 281-290
-
-
Francis, J.E.1
Cash, W.D.2
Barbaz, B.S.3
Bernard, P.S.4
Lovell, R.A.5
Mazzenga, G.C.6
Friedmann, R.C.7
Hyun, J.L.8
Braunwalder, A.F.9
Loo, P.S.10
Bennett, D.A.11
-
4
-
-
34247554190
-
Synthesis and pharmacological investigation of novel 4-benzyl-1- substituted-4H-[1,2,4]triazolo[4,3-a]quinazolin-5-ones as new class of H1- antihistaminic agents
-
Alagarsamy, V.; Solomon, V.R.; Murugan, M. Synthesis and pharmacological investigation of novel 4-benzyl-1-substituted-4H-[1,2,4]triazolo[4,3-a] quinazolin-5-ones as new class of H1- antihistaminic agents. Bioorg. Med. Chem. 2007, 15, 4009-4015.
-
(2007)
Bioorg. Med. Chem.
, vol.15
, pp. 4009-4015
-
-
Alagarsamy, V.1
Solomon, V.R.2
Murugan, M.3
-
5
-
-
15044350987
-
Synthesis and pharmacological investigation of novel 1-substituted-4- phenyl-1,2,4-triazolo[4,3-a]quinazolin-5(4H)-ones as a new class of H1-antihistaminic agents
-
Alagarsamy, V.; Giridhar, R.; Yadav, M.R. Synthesis and pharmacological investigation of novel 1-substituted-4-phenyl-1,2,4-triazolo[4,3-a]quinazolin- 5(4H)-ones as a new class of H1-antihistaminic agents. Bioorg. Med. Chem. Lett. 2005, 15, 1877-1880.
-
(2005)
Bioorg. Med. Chem. Lett.
, vol.15
, pp. 1877-1880
-
-
Alagarsamy, V.1
Giridhar, R.2
Yadav, M.R.3
-
6
-
-
78149425235
-
Diaminotriazoles useful as inhibitors of protein kinases WO
-
2004046120
-
Albert, C.P.; Michael, A.; Robert, J.D.; Cornelia, J.F.; Vincent, G.; Ronald, G.; Mark, L.; Shi-kai, T.; Jinwang, X.; Hayley, B.; Brian, L.; David, M.; Suganthi, N.; Andrew, J. Diaminotriazoles useful as inhibitors of protein kinases. WO 2004046120; [Chem. Abstr. 2004, 141, 23537].
-
(2004)
Chem. Abstr.
, vol.141
, pp. 23537
-
-
Albert, C.P.1
Michael, A.2
Robert, J.D.3
Cornelia, J.F.4
Vincent, G.5
Ronald, G.6
Mark, L.7
Shi-kai, T.8
Jinwang, X.9
Hayley, B.10
Brian, L.11
David, M.12
Suganthi, N.13
Andrew, J.14
-
7
-
-
78149439571
-
Novel synthesis of 2-Alkoxy(aralkoxy)-5-chloro[1,2,4]triazolo-[1,5-a] quinazolines and their derivatives
-
Al-salahi, R.; Geffken, D. Novel synthesis of 2-Alkoxy(aralkoxy)-5- chloro[1,2,4]triazolo-[1,5- a]quinazolines and their derivatives. Heterocycles 2010, 81, 1843-1859.
-
(2010)
Heterocycles
, vol.81
, pp. 1843-1859
-
-
Al-salahi, R.1
Geffken, D.2
-
8
-
-
79957452383
-
Preparation of dialkyl-N-cyanoimidocarbonates EP
-
519868
-
Michael, A.O.; Ward, H.O. Preparation of dialkyl-N-cyanoimidocarbonates. EP 519868; [Chem. Abstr. 1992, 118, 168717].
-
(1992)
Chem. Abstr.
, vol.118
, pp. 168717
-
-
Michael, A.O.1
Ward, H.O.2
-
9
-
-
84971056139
-
Constitution of the so-called dithiocyanic acid and perthiocyanic acid
-
Hantzsch, A.; Wolvekamp. M. Constitution of the so-called dithiocyanic acid and perthiocyanic acid. Annalen der Chemie 1904, 331, 265-297.
-
(1904)
Annalen der Chemie
, vol.331
, pp. 265-297
-
-
Hantzsch, A.1
Wolvekamp, M.2
-
10
-
-
78149441538
-
4,5-dihydro-5-oxopyrazolo[1,5-a]qiunazoline-3-carboxylic acid derivatives US Pat.
-
4105766
-
Alexander, J.E. 4,5-dihydro-5-oxopyrazolo[1,5-a]qiunazoline-3-carboxylic acid derivatives. US Pat. 4105766; [Chem.Abstr. 1978, 77, 140065].
-
(1978)
Chem.Abstr.
, vol.77
, pp. 140065
-
-
Alexander, J.E.1
-
11
-
-
0002235515
-
Synthesis and structure elucidation of 3-methoxy-1-methyl-1H-1,2,4- triazol-5-amine and 5-methoxy-1-methyl-1H-1,2,4-triazol-3-amine
-
Selby, T.P.; Lepone, G.E. Synthesis and structure elucidation of 3-methoxy-1-methyl-1H-1,2,4- triazol-5-amine and 5-methoxy-1-methyl-1H-1,2,4- triazol-3-amine. J. Heterocycl. Chem. 1984, 21, 61-64
-
(1984)
J. Heterocycl. Chem.
, vol.21
, pp. 61-64
-
-
Selby, T.P.1
Lepone, G.E.2
-
12
-
-
84986513731
-
Diphenyl cyanocarbonimidate. A versatile synthon for the construction of heterocyclic systems
-
Webb, L.R.; Labaw, C.S. Diphenyl cyanocarbonimidate. A versatile synthon for the construction of heterocyclic systems. J. Heterocycl. Chem. 1982, 19, 1205-1206.
-
(1982)
J. Heterocycl. Chem.
, vol.19
, pp. 1205-1206
-
-
Webb, L.R.1
Labaw, C.S.2
-
13
-
-
84985155014
-
Heterocyclic amine precursors to sulfonylurea herbicides
-
Kristinsson, H.; Winkler, T. Heterocyclic amine precursors to sulfonylurea herbicides. Helv. Chim. Acta 1983, 66, 1129-1136.
-
(1983)
Helv. Chim. Acta
, vol.66
, pp. 1129-1136
-
-
Kristinsson, H.1
Winkler, T.2
-
14
-
-
84985156392
-
Synthesis of [1,2,4.triazolo]1,5-a]quinazolines. Effect of substituent orientation on carbon-13 chemical shift. Part III. Deduction of the conformation of substituents by carbon-13-NMR spectroscopy
-
Heckendorn, R.; Winkler, T. Synthesis of [1,2,4.triazolo]1,5-a] quinazolines. Effect of substituent orientation on carbon-13 chemical shift. Part III. Deduction of the conformation of substituents by carbon-13-NMR spectroscopy. Helv. Chim. Acta 1980, 63, 1-9.
-
(1980)
Helv. Chim. Acta
, vol.63
, pp. 1-9
-
-
Heckendorn, R.1
Winkler, T.2
-
15
-
-
0001512391
-
A-Lactams. VIII. O-Alkylation of a-lactams
-
Sheehan, J.C.; Nafissi-V, M.M. a-Lactams. VIII. O-Alkylation of a-lactams. J. Org. Chem. 1970, 12, 4246-4248.
-
(1970)
J. Org. Chem.
, vol.12
, pp. 4246-4248
-
-
Sheehan, J.C.1
Nafissi-V, M.M.2
-
16
-
-
0141843275
-
N-alkylation of lactams with phase transfer catalyst
-
Takahata, H.; Hashizume, T.; Yamazaki, T. N-alkylation of lactams with phase transfer catalyst. Heterocycles 1979, 12, 1449-1451.
-
(1979)
Heterocycles
, vol.12
, pp. 1449-1451
-
-
Takahata, H.1
Hashizume, T.2
Yamazaki, T.3
-
17
-
-
31644449084
-
Alkylation of N-substituted 2-phenylacetamides
-
Muin, D.Z.; Misic-V, M.M.; Petrovic, S.D. Alkylation of N-substituted 2-phenylacetamides. J. Serb. Chem. Soc. 2004, 69, 711-736.
-
(2004)
J. Serb. Chem. Soc.
, vol.69
, pp. 711-736
-
-
Muin, D.Z.1
Misic-V, M.M.2
Petrovic, S.D.3
-
18
-
-
0016808785
-
Chemistry of 2H-3,1-benzoxazine-2,4(1H)-dione (isatoic anhydrides). Synthesis of N-substituted 2H-3,1-benzoxazine-2,4(1H)-diones
-
Hardtman, G.E.; Koleter, G.; Pfister, O.R. Chemistry of 2H-3,1-benzoxazine-2,4(1H)-dione (isatoic anhydrides). Synthesis of N-substituted 2H-3,1-benzoxazine-2,4(1H)-diones. J. Heterocycl. Chem. 1975, 12, 565-572.
-
(1975)
J. Heterocycl. Chem.
, vol.12
, pp. 565-572
-
-
Hardtman, G.E.1
Koleter, G.2
Pfister, O.R.3
-
19
-
-
78149438509
-
Verfahren zur herstellung N-substituiertrer lactame DE
-
2338257
-
Luessi, H.; Berther, C.; Studinka, J. Verfahren zur herstellung N-substituiertrer lactame. DE 2338257; [Chem. Abstr. 1974, 81 106237].
-
(1974)
Chem. Abstr.
, vol.81
, pp. 106237
-
-
Luessi, H.1
Berther, C.2
Studinka, J.3
-
21
-
-
78149430050
-
A new synthesis of phenanthridine
-
Taylor, E.C.; Martin, A.E. A new synthesis of phenanthridine. J. Chem. Soc. 1952, 11, 6295.
-
(1952)
J. Chem. Soc.
, vol.11
, pp. 6295
-
-
Taylor, E.C.1
Martin, A.E.2
-
22
-
-
0037204011
-
Structure-activity relationships for pyrido-, imidazo-, pyrazolo-, pyrazino-, and pyrrolophenazinecarboxamides as topoisomerase-targeted anticancer agents. J
-
Gamage, S.A.; Spicer, J.A.; Rewcastle, G.W.; Milton, J.; Sohal, S.; Dangerfield, W.; Mistry, P.; Vicker, N.; Charlton, P.A.; Denny, W.A. Structure-activity relationships for pyrido-, imidazo-, pyrazolo-, pyrazino-, and pyrrolophenazinecarboxamides as topoisomerase-targeted anticancer agents. J. Med. Chem. 2002, 45, 740-743
-
(2002)
Med. Chem.
, vol.45
, pp. 740-743
-
-
Gamage, S.A.1
Spicer, J.A.2
Rewcastle, G.W.3
Milton, J.4
Sohal, S.5
Dangerfield, W.6
Mistry, P.7
Vicker, N.8
Charlton, P.A.9
Denny, W.A.10
-
23
-
-
0032785834
-
Synthesis and reactivity of 1,2,4-triazolo[1,5-c]quinazolines
-
Pfeiffer, W.D.; Hetzheim, A.; Pazdera, P.; Bodtke, A.; Muecke, J. Synthesis and reactivity of 1,2,4-triazolo[1,5-c]quinazolines. J. Heterocycl. Chem. 1999, 36, 1327-1336.
-
(1999)
J Heterocycl. Chem.
, vol.36
, pp. 1327-1336
-
-
Pfeiffer, W.D.1
Hetzheim, A.2
Pazdera, P.3
Bodtke, A.4
Muecke, J.5
-
24
-
-
84985257133
-
Reaction of 4-aryl-1,2,4-triazines with hydrazine. J. Heterocycl
-
Badawy, M.A.; Abdel-Hady, S.A.; Ibrahim, Y.A. Reaction of 4-aryl-1,2,4-triazines with hydrazine. J. Heterocycl. Chem. 1981, 18, 953-956.
-
(1981)
Chem.
, vol.18
, pp. 953-956
-
-
Badawy, M.A.1
Abdel-Hady, S.A.2
Ibrahim, Y.A.3
-
25
-
-
0347087388
-
Synthesis and reactions of 3-amino-2- methyl-3H-[1,2,4]triazolo[5,1-b]- quinazolin-9-one and 2-hydrazino-3-phenylamino-3H-quinazolin- 4-one
-
Saleh, M.A.; Hafez, Y.A.; Abdel-Hay, F.E.; Gad, W.I. Synthesis and reactions of 3-amino-2- methyl-3H-[1,2,4]triazolo[5,1-b]-quinazolin-9-one and 2-hydrazino-3-phenylamino-3H-quinazolin- 4-one. J. Heterocycl. Chem. 2003, 40, 973-978.
-
(2003)
J. Heterocycl Chem.
, vol.40
, pp. 973-978
-
-
Saleh, M.A.1
Hafez, Y.A.2
Abdel-Hay, F.E.3
Gad, W.I.4
-
26
-
-
0017929934
-
4-aryl-5-thioxo-1,2,4,5-tetrahydro-s-triazolo [4,3-a]quinazolines and derivatives, synthesis of compounds with aminoguanidine structutres
-
Kottke, K.; Kuehmstedt, H. 4-aryl-5-thioxo-1,2,4,5-tetrahydro-s-triazolo [4,3-a]quinazolines and derivatives, synthesis of compounds with aminoguanidine structutres. Pharmazie 1978, 33, 124-125.
-
(1978)
Pharmazie
, vol.33
, pp. 124-125
-
-
Kottke, K.1
Kuehmstedt, H.2
-
27
-
-
0018380855
-
1,2,4-triazolo- and 1,2,5-triazino[4,3-d][1,4]benzodiazepinone ring systems: Synthesis and barrier to ring inversion
-
Wade, P.C.; Vogt, B.R.; Toeplitz, B.; Puan, M.S. 1,2,4-triazolo- and 1,2,5-triazino[4,3- d][1,4]benzodiazepinone ring systems: Synthesis and barrier to ring inversion. J. Org. Chem. 1979, 44, 88-99.
-
(1979)
J. Org. Chem.
, vol.44
, pp. 88-99
-
-
Wade, P.C.1
Vogt, B.R.2
Toeplitz, B.3
Puan, M.S.4
-
28
-
-
12344327758
-
Unexpected hydrazinolysis behaviour of 1-chloro-4-methyl-5H-pyridazino[4, 5-b]indole and a convenient synthesis of new [1,2,4]- triazolo[4',3':1,6] pyridazino[4,5-b]indoles
-
Hussein, E.; Abdlrahman, A. H.; Norbert H.; Andrea, W. Unexpected hydrazinolysis behaviour of 1-chloro-4-methyl-5H-pyridazino[4,5-b]indole and a convenient synthesis of new [1,2,4]- triazolo[4',3':1,6]pyridazino[4,5-b] indoles. Molecules 2004, 9, 849-859.
-
(2004)
Molecules
, vol.9
, pp. 849-859
-
-
Hussein, E.1
Abdlrahman, A.H.2
Norbert, H.3
Andrea, W.4
-
29
-
-
78149442977
-
Preparation of tetrazoloquinoline derivatives as inhibitors of HCV WO Pat
-
2005030774
-
Sambaiah, T.; Ankush, A.; Rajinder, S.; Henry, H.L.; Peiyong, H. Preparation of tetrazoloquinoline derivatives as inhibitors of HCV. WO Pat. 2005030774; [Chem. Abstr. 2005, 142, 373704].
-
(2005)
Chem. Abstr.
, vol.142
, pp. 373704
-
-
Sambaiah, T.1
Ankush, A.2
Rajinder, S.3
Henry, H.L.4
Peiyong, H.5
|