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Volumn 31, Issue 12, 2010, Pages 2318-2321

Structure-activity studies on novel polymyxin derivatives that carry only three positive charges

Author keywords

[No Author keywords available]

Indexed keywords

ANTIINFECTIVE AGENT; CATION; FATTY ACID; NAB 7061; NAB 739; NAB 750; NAB 751; NAB 771; NAB 781; NAB 782; PEPTIDE; POLYMYXIN DERIVATIVE; RIFAMPICIN; SERINE; UNCLASSIFIED DRUG;

EID: 78049464981     PISSN: 01969781     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.peptides.2010.09.010     Document Type: Article
Times cited : (24)

References (20)
  • 1
    • 73949154997 scopus 로고    scopus 로고
    • Pharmacokinetics of novel antimicrobial cationic peptides NAB7061 and NAB739 in rats following intravenous administration
    • F.E. Ali, G. Cao, A. Poydal, T. Vaara, R.L. Nation, and M. Vaara Pharmacokinetics of novel antimicrobial cationic peptides NAB7061 and NAB739 in rats following intravenous administration J Antimicrob Chemother 64 2009 1067 1070
    • (2009) J Antimicrob Chemother , vol.64 , pp. 1067-1070
    • Ali, F.E.1    Cao, G.2    Poydal, A.3    Vaara, T.4    Nation, R.L.5    Vaara, M.6
  • 2
    • 59449088862 scopus 로고    scopus 로고
    • Antibiotic-resistant bugs in the 21st century - A clinical super-challenge
    • C.A. Arias, and B.E. Murray Antibiotic-resistant bugs in the 21st century - a clinical super-challenge New Engl J Med 360 2009 439 443
    • (2009) New Engl J Med , vol.360 , pp. 439-443
    • Arias, C.A.1    Murray, B.E.2
  • 6
    • 65349101100 scopus 로고    scopus 로고
    • Development of des-fatty acyl-polymyxin B decapeptide analogs with Pseudomonas aeruginosa-specific antimicrobial activity
    • N. Katsuma, Y. Sato, K. Ohki, K. Okimura, K. Ohnishi, and N. Sakura Development of des-fatty acyl-polymyxin B decapeptide analogs with Pseudomonas aeruginosa-specific antimicrobial activity Chem Pharm Bull 57 2009 332 336
    • (2009) Chem Pharm Bull , vol.57 , pp. 332-336
    • Katsuma, N.1    Sato, Y.2    Ohki, K.3    Okimura, K.4    Ohnishi, K.5    Sakura, N.6
  • 8
    • 69949174478 scopus 로고    scopus 로고
    • Has the era of untreatable infections arrived?
    • D. Livermore Has the era of untreatable infections arrived? J Antimicrob Chemother 64 Suppl 1 2009 i29 i36
    • (2009) J Antimicrob Chemother , vol.64 , Issue.SUPPL. 1
    • Livermore, D.1
  • 9
    • 70350528719 scopus 로고    scopus 로고
    • Colistin in the 21st century
    • R.L. Nation, and J. Li Colistin in the 21st century Curr Opin Infect Dis 22 2009 535 543
    • (2009) Curr Opin Infect Dis , vol.22 , pp. 535-543
    • Nation, R.L.1    Li, J.2
  • 11
    • 0034817854 scopus 로고    scopus 로고
    • N-terminal modifications of polymyxin B nonapeptide and their effect on antibacterial activity
    • H. Tsubery, I. Ofek, S. Cohen, and M. Fridkin N-terminal modifications of polymyxin B nonapeptide and their effect on antibacterial activity Peptides 22 2001 1675 1681
    • (2001) Peptides , vol.22 , pp. 1675-1681
    • Tsubery, H.1    Ofek, I.2    Cohen, S.3    Fridkin, M.4
  • 12
    • 76649119425 scopus 로고    scopus 로고
    • Structure-activity relationships of bacterial outer-membrane permeabilizers based on polymyxin B heptapeptides
    • H. Urakawa, K. Yamada, K. Komagoe, S. Ando, H. Oku, and T. Katsu Structure-activity relationships of bacterial outer-membrane permeabilizers based on polymyxin B heptapeptides Bioorg Med Chem Lett 20 2010 1771 1775
    • (2010) Bioorg Med Chem Lett , vol.20 , pp. 1771-1775
    • Urakawa, H.1    Yamada, K.2    Komagoe, K.3    Ando, S.4    Oku, H.5    Katsu, T.6
  • 13
    • 0026802197 scopus 로고
    • Agents that increase the permeability of the outer membrane
    • M. Vaara Agents that increase the permeability of the outer membrane Microbiol Rev 56 1992 395 411
    • (1992) Microbiol Rev , vol.56 , pp. 395-411
    • Vaara, M.1
  • 14
    • 70349496543 scopus 로고    scopus 로고
    • New approaches in peptide antibiotics
    • M. Vaara New approaches in peptide antibiotics Curr Opin Pharmacol 9 2009 571 576
    • (2009) Curr Opin Pharmacol , vol.9 , pp. 571-576
    • Vaara, M.1
  • 15
    • 50949130838 scopus 로고    scopus 로고
    • Novel polymyxin derivatives carrying only three positive charges are effective antibacterial agents
    • M. Vaara, J. Fox, G. Loidl, O. Siikanen, J. Apajalahti, and F. Hansen Novel polymyxin derivatives carrying only three positive charges are effective antibacterial agents Antimicrob Agents Chemother 52 2008 3229 3236
    • (2008) Antimicrob Agents Chemother , vol.52 , pp. 3229-3236
    • Vaara, M.1    Fox, J.2    Loidl, G.3    Siikanen, O.4    Apajalahti, J.5    Hansen, F.6
  • 16
    • 77955345521 scopus 로고    scopus 로고
    • A novel polymyxin derivative that lacks the fatty acid tail and carries only three positive charges has strong synergism with agents excluded by the intact outer membrane
    • M. Vaara, O. Siikanen, J. Apajalahti, J. Fox, N. Frimodt-Møller, and H. He A novel polymyxin derivative that lacks the fatty acid tail and carries only three positive charges has strong synergism with agents excluded by the intact outer membrane Antimicrob Agents Chemother 54 2010 3341 3346
    • (2010) Antimicrob Agents Chemother , vol.54 , pp. 3341-3346
    • Vaara, M.1    Siikanen, O.2    Apajalahti, J.3    Fox, J.4    Frimodt-Møller, N.5    He, H.6
  • 17
    • 77953706297 scopus 로고    scopus 로고
    • Susceptibility of carbapenemase-producing strains of Klebsiella pneumoniae and Escherichia coli to the direct antibacterial activity of NAB739 and to the synergistic activity of NAB7061 with rifampin and clarithromycin
    • M. Vaara, O. Siikanen, J. Apajalahti, N. Frimodt-Møller, and T. Vaara Susceptibility of carbapenemase-producing strains of Klebsiella pneumoniae and Escherichia coli to the direct antibacterial activity of NAB739 and to the synergistic activity of NAB7061 with rifampin and clarithromycin J Antimicrob Chemother 65 2010 942 945
    • (2010) J Antimicrob Chemother , vol.65 , pp. 942-945
    • Vaara, M.1    Siikanen, O.2    Apajalahti, J.3    Frimodt-Møller, N.4    Vaara, T.5
  • 18
    • 77949346087 scopus 로고    scopus 로고
    • Structure-activity relationships of polymyxin antibiotics
    • T. Velkov, P.E. Thompson, R.L. Nation, and J. Li Structure-activity relationships of polymyxin antibiotics J Med Chem 53 2010 1898 1916
    • (2010) J Med Chem , vol.53 , pp. 1898-1916
    • Velkov, T.1    Thompson, P.E.2    Nation, R.L.3    Li, J.4
  • 19
    • 0021257420 scopus 로고
    • Susceptibility of Gram-negative bacteria to polymyxin B nonapeptide
    • P. Viljanen, and M. Vaara Susceptibility of Gram-negative bacteria to polymyxin B nonapeptide Antimicrob Agents Chemother 25 1984 701 705
    • (1984) Antimicrob Agents Chemother , vol.25 , pp. 701-705
    • Viljanen, P.1    Vaara, M.2
  • 20
    • 77953707737 scopus 로고    scopus 로고
    • Novel polymyxin derivatives are effective in treating experimental Escherichia coli peritoneal infection in mice
    • C. Vingsbo Lundberg, T. Vaara, N. Frimodt-Møller, and M. Vaara Novel polymyxin derivatives are effective in treating experimental Escherichia coli peritoneal infection in mice J Antimicrob Chemother 65 2010 981 985
    • (2010) J Antimicrob Chemother , vol.65 , pp. 981-985
    • Vingsbo Lundberg, C.1    Vaara, T.2    Frimodt-Møller, N.3    Vaara, M.4


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.