Contribution of each amino acid residue in polymyxin b3 to antimicrobial and lipopolysaccharide binding activity

Chemical and Pharmaceutical Bulletin

Volumn 57, Issue 3, 2009, Pages 240-244

  Kanazawa, Kazushi ^a,b   Sato, Yuki ^a   Ohki, Kazuhiro ^a   Okimura, Keiko ^a   Uchida, Yoshiki ^b   Shindo, Mitsuno ^b   Sakura, Naoki ^a  

^a HOKURIKU UNIVERSITY   (Japan)

^b OSAKA SHOIN WOMEN'S UNIVERSITY   (Japan)

Author keywords

Alanine scanning; Antimicrobial activity; Diaminobutyric acid; Lipopolysaccharide binding activity; Polymyxin B

Indexed keywords

ALANINE DERIVATIVE; AMINO ACID; CYCLOPEPTIDE; LIPOPOLYSACCHARIDE; POLYMYXIN B; POLYMYXIN B3 DERIVATIVE; POLYPEPTIDE ANTIBIOTIC AGENT; UNCLASSIFIED DRUG;

ANTIBACTERIAL ACTIVITY; ANTIMICROBIAL ACTIVITY; ARTICLE; BACTERICIDAL ACTIVITY; BINDING ASSAY; CONFORMATIONAL TRANSITION; DRUG BINDING; DRUG POTENCY; DRUG STRUCTURE; DRUG SYNTHESIS; ESCHERICHIA COLI; HYDROPHOBICITY; MINIMUM INHIBITORY CONCENTRATION; NONHUMAN; PSEUDOMONAS AERUGINOSA; SALMONELLA TYPHIMURIUM; STRUCTURE ACTIVITY RELATION; STRUCTURE ANALYSIS;

ALANINE; AMINO ACID SEQUENCE; ANTI-BACTERIAL AGENTS; HYDROPHOBICITY; LIPOPOLYSACCHARIDES; MICROBIAL SENSITIVITY TESTS; POLYMYXIN B; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 62549141514     PISSN: 00092363     EISSN: 13475223     Source Type: Journal    
DOI: 10.1248/cpb.57.240     Document Type: Article

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