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Bioorganic and Medicinal Chemistry Letters

Volumn 20, Issue 22, 2010, Pages 6653-6656

Design, synthesis and biological evaluation of quinoline amide derivatives as novel VEGFR-2 inhibitors

(6) Yang, Ying a Shi, Lei a Zhou, Yang a Li, Huan Qiu a Zhu, Zhen Wei a Zhu, Hai Liang a

a NANJING UNIVERSITY (China)

Author keywords

Docking; Quinoline amide; SAR; VEGFR 2 inhibitor

Indexed keywords

5 CHLORO 2 HYDROXY N (QUINOLIN 8 YL)BENZAMIDE; AMIDE; QUINOLINE DERIVATIVE; UNCLASSIFIED DRUG; VASCULOTROPIN RECEPTOR 2;

ARTICLE; BINDING SITE; CANCER THERAPY; DRUG INHIBITION; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS; ENDOTHELIUM CELL; HUMAN; HUMAN CELL; IC 50; IN VITRO SELECTION; MOLECULAR DOCKING; PHARMACOPHORE; UMBILICAL VEIN;

AMIDES; CELLS, CULTURED; DRUG DESIGN; HUMANS; INHIBITORY CONCENTRATION 50; MODELS, MOLECULAR; QUINOLINES; VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR-2;

EID: 77958064279 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/j.bmcl.2010.09.014 Document Type: Article

Times cited : (55)

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