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Volumn 1359, Issue , 2010, Pages 67-74

Mechanism of Kv2.1 channel inhibition by a selective COX-2 inhibitor SC-791-modification of gating

Author keywords

COX 2 inhibitor; Potassium channel; SC 791

Indexed keywords

CYCLOOXYGENASE 2 INHIBITOR; POTASSIUM CHANNEL KV2.1; SC 791; UNCLASSIFIED DRUG; VOLTAGE GATED POTASSIUM CHANNEL;

EID: 77957977131     PISSN: 00068993     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.brainres.2010.08.062     Document Type: Article
Times cited : (8)

References (34)
  • 1
    • 0033179040 scopus 로고    scopus 로고
    • Delayed rectifier currents in rat globus pallidus neurons are attributable to Kv2.1 and Kv3.1/3.2 K(+) channels
    • G. Baranauskas, T. Tkatch, and D.J. Surmeier Delayed rectifier currents in rat globus pallidus neurons are attributable to Kv2.1 and Kv3.1/3.2 K(+) channels J. Neurosci. 19 1999 6394 6404
    • (1999) J. Neurosci. , vol.19 , pp. 6394-6404
    • Baranauskas, G.1    Tkatch, T.2    Surmeier, D.J.3
  • 3
    • 0029586384 scopus 로고
    • Closed- and open-state binding of 4-aminopyridine to the cloned human potassium channel Kv1.5
    • R. Bouchard, and D. Fedida Closed- and open-state binding of 4-aminopyridine to the cloned human potassium channel Kv1.5 J. Pharmacol. Exp. Ther. 275 1995 864 876
    • (1995) J. Pharmacol. Exp. Ther. , vol.275 , pp. 864-876
    • Bouchard, R.1    Fedida, D.2
  • 4
    • 70350452558 scopus 로고    scopus 로고
    • Differential effects of selective cyclooxygenase-2 inhibitors on vascular smooth muscle ion channels may account for differences in cardiovascular risk profiles
    • L.I. Brueggemann, A.R. Mackie, B.K. Mani, L.L. Cribbs, and K.L. Byron Differential effects of selective cyclooxygenase-2 inhibitors on vascular smooth muscle ion channels may account for differences in cardiovascular risk profiles Mol. Pharmacol. 76 2009 1053 1061
    • (2009) Mol. Pharmacol. , vol.76 , pp. 1053-1061
    • Brueggemann, L.I.1    MacKie, A.R.2    Mani, B.K.3    Cribbs, L.L.4    Byron, K.L.5
  • 6
    • 0037364161 scopus 로고    scopus 로고
    • The development of COX2 inhibitors
    • R.J. Flower The development of COX2 inhibitors Nat. Rev. Drug Discov. 2 2003 179 191
    • (2003) Nat. Rev. Drug Discov. , vol.2 , pp. 179-191
    • Flower, R.J.1
  • 7
    • 38349110209 scopus 로고    scopus 로고
    • Inhibition of delayed rectifier potassium channels and induction of arrhythmia: A novel effect of celecoxib and the mechanism underlying it
    • R.V. Frolov, I.G. Berim, and S. Singh Inhibition of delayed rectifier potassium channels and induction of arrhythmia: a novel effect of celecoxib and the mechanism underlying it J. Biol. Chem. 283 2008 1518 1524
    • (2008) J. Biol. Chem. , vol.283 , pp. 1518-1524
    • Frolov, R.V.1    Berim, I.G.2    Singh, S.3
  • 8
    • 45849112870 scopus 로고    scopus 로고
    • Effects of celecoxib on ionic currents and spontaneous firing in rat retinal neurons
    • R.V. Frolov, M.M. Slaughter, and S. Singh Effects of celecoxib on ionic currents and spontaneous firing in rat retinal neurons Neuroscience 154 2008 1525 1532
    • (2008) Neuroscience , vol.154 , pp. 1525-1532
    • Frolov, R.V.1    Slaughter, M.M.2    Singh, S.3
  • 9
    • 75649132167 scopus 로고    scopus 로고
    • Mechanisms of Kv2.1 channel inhibition by celecoxib-modification of gating and channel block
    • R.V. Frolov, V.E. Bondarenko, and S. Singh Mechanisms of Kv2.1 channel inhibition by celecoxib-modification of gating and channel block Br. J. Pharmacol. 159 2010 405 418
    • (2010) Br. J. Pharmacol. , vol.159 , pp. 405-418
    • Frolov, R.V.1    Bondarenko, V.E.2    Singh, S.3
  • 10
    • 28244447363 scopus 로고    scopus 로고
    • Screening new drugs for immunotoxic potential: III. Assessment of the effects of selective and nonselective COX-2 inhibitors on T-cell-dependent antibody and natural killer cell responses in the rat
    • S.M. Furst, K.N. Khan, W.J. Komocsar, and J. Mennear Screening new drugs for immunotoxic potential: III. Assessment of the effects of selective and nonselective COX-2 inhibitors on T-cell-dependent antibody and natural killer cell responses in the rat J. Immunotoxicol. 2 2005 161 170
    • (2005) J. Immunotoxicol. , vol.2 , pp. 161-170
    • Furst, S.M.1    Khan, K.N.2    Komocsar, W.J.3    Mennear, J.4
  • 12
    • 33745238704 scopus 로고    scopus 로고
    • Cyclooxygenase-2 (COX-2)-independent anticarcinogenic effects of selective COX-2 inhibitors
    • S. Grosch, T.J. Maier, S. Schiffmann, and G. Geisslinger Cyclooxygenase-2 (COX-2)-independent anticarcinogenic effects of selective COX-2 inhibitors J. Natl Cancer Inst. 98 2006 736 747
    • (2006) J. Natl Cancer Inst. , vol.98 , pp. 736-747
    • Grosch, S.1    Maier, T.J.2    Schiffmann, S.3    Geisslinger, G.4
  • 14
    • 34548315729 scopus 로고    scopus 로고
    • The cytotoxicity of celecoxib towards cardiac myocytes is cyclooxygenase-2 independent
    • B.B. Hasinoff, D. Patel, and X. Wu The cytotoxicity of celecoxib towards cardiac myocytes is cyclooxygenase-2 independent Cardiovasc. Toxicol. 7 2007 19 27
    • (2007) Cardiovasc. Toxicol. , vol.7 , pp. 19-27
    • Hasinoff, B.B.1    Patel, D.2    Wu, X.3
  • 15
    • 77950080219 scopus 로고    scopus 로고
    • Protective effect of rebamipide against celecoxib-induced gastric mucosal cell apoptosis
    • T. Ishihara, K. Tanaka, S. Tashiro, K. Yoshida, and T. Mizushima Protective effect of rebamipide against celecoxib-induced gastric mucosal cell apoptosis Biochem. Pharmacol. 79 2010 1622 1633
    • (2010) Biochem. Pharmacol. , vol.79 , pp. 1622-1633
    • Ishihara, T.1    Tanaka, K.2    Tashiro, S.3    Yoshida, K.4    Mizushima, T.5
  • 16
    • 0036896925 scopus 로고    scopus 로고
    • Delayed rectifier K + currents, IK, are encoded by Kv2 alpha-subunits and regulate tonic firing in mammalian sympathetic neurons
    • S.A. Malin, and J.M. Nerbonne Delayed rectifier K + currents, IK, are encoded by Kv2 alpha-subunits and regulate tonic firing in mammalian sympathetic neurons J. Neurosci. 22 2002 10094 10105
    • (2002) J. Neurosci. , vol.22 , pp. 10094-10105
    • Malin, S.A.1    Nerbonne, J.M.2
  • 17
    • 0038643828 scopus 로고    scopus 로고
    • Preferential closed channel blockade of HERG potassium currents by chemically synthesised BeKm-1 scorpion toxin
    • J.T. Milnes, C.E. Dempsey, J.M. Ridley, O. Crociani, A. Arcangeli, J.C. Hancox, and H.J. Witchel Preferential closed channel blockade of HERG potassium currents by chemically synthesised BeKm-1 scorpion toxin FEBS Lett. 547 2003 20 26
    • (2003) FEBS Lett. , vol.547 , pp. 20-26
    • Milnes, J.T.1    Dempsey, C.E.2    Ridley, J.M.3    Crociani, O.4    Arcangeli, A.5    Hancox, J.C.6    Witchel, H.J.7
  • 19
    • 0033103708 scopus 로고    scopus 로고
    • Identification of the Kv2.1 K + channel as a major component of the delayed rectifier K + current in rat hippocampal neurons
    • H. Murakoshi, and J.S. Trimmer Identification of the Kv2.1 K + channel as a major component of the delayed rectifier K + current in rat hippocampal neurons J. Neurosci. 19 1999 1728 1735
    • (1999) J. Neurosci. , vol.19 , pp. 1728-1735
    • Murakoshi, H.1    Trimmer, J.S.2
  • 20
    • 21044449616 scopus 로고    scopus 로고
    • Targeting of voltage-gated potassium channel isoforms to distinct cell surface microdomains
    • K.M. O'Connell, and M.M. Tamkun Targeting of voltage-gated potassium channel isoforms to distinct cell surface microdomains J. Cell Sci. 118 2005 2155 2166
    • (2005) J. Cell Sci. , vol.118 , pp. 2155-2166
    • O'Connell, K.M.1    Tamkun, M.M.2
  • 23
    • 0030859539 scopus 로고    scopus 로고
    • Kv2.1/Kv9.3, a novel ATP-dependent delayed-rectifier K + channel in oxygen-sensitive pulmonary artery myocytes
    • A.J. Patel, M. Lazdunski, and E. Honore Kv2.1/Kv9.3, a novel ATP-dependent delayed-rectifier K + channel in oxygen-sensitive pulmonary artery myocytes EMBO J. 16 1997 6615 6625
    • (1997) EMBO J. , vol.16 , pp. 6615-6625
    • Patel, A.J.1    Lazdunski, M.2    Honore, E.3
  • 24
    • 0032052936 scopus 로고    scopus 로고
    • Localization of potassium channels in the retina
    • L.H. Pinto, and D.J. Klumpp Localization of potassium channels in the retina Prog. Retin. Eye Res. 17 1998 207 230
    • (1998) Prog. Retin. Eye Res. , vol.17 , pp. 207-230
    • Pinto, L.H.1    Klumpp, D.J.2
  • 27
    • 0141887470 scopus 로고    scopus 로고
    • Epidermal COX-2 induction following ultraviolet irradiation: Suggested mechanism for the role of COX-2 inhibition in photoprotection
    • C.S. Tripp, E.A. Blomme, K.S. Chinn, M.M. Hardy, P. LaCelle, and A.P. Pentland Epidermal COX-2 induction following ultraviolet irradiation: suggested mechanism for the role of COX-2 inhibition in photoprotection J. Invest. Dermatol. 121 2003 853 861
    • (2003) J. Invest. Dermatol. , vol.121 , pp. 853-861
    • Tripp, C.S.1    Blomme, E.A.2    Chinn, K.S.3    Hardy, M.M.4    Lacelle, P.5    Pentland, A.P.6
  • 28
    • 0036949973 scopus 로고    scopus 로고
    • KV2.1 K + channels underlie major voltage-gated K + outward current in H9c2 myoblasts
    • W. Wang, N. Hino, H. Yamasaki, T. Aoki, and R. Ochi KV2.1 K + channels underlie major voltage-gated K + outward current in H9c2 myoblasts Jpn J. Physiol. 52 2002 507 514
    • (2002) Jpn J. Physiol. , vol.52 , pp. 507-514
    • Wang, W.1    Hino, N.2    Yamasaki, H.3    Aoki, T.4    Ochi, R.5
  • 30
    • 0037440022 scopus 로고    scopus 로고
    • Kv1.4 channel block by quinidine: Evidence for a drug-induced allosteric effect
    • S. Wang, M.J. Morales, Y.J. Qu, G.C. Bett, H.C. Strauss, and R.L. Rasmusson Kv1.4 channel block by quinidine: evidence for a drug-induced allosteric effect J. Physiol. 546 2003 387 401
    • (2003) J. Physiol. , vol.546 , pp. 387-401
    • Wang, S.1    Morales, M.J.2    Qu, Y.J.3    Bett, G.C.4    Strauss, H.C.5    Rasmusson, R.L.6
  • 32
    • 1642540579 scopus 로고    scopus 로고
    • Unexpected nanomolar inhibition of carbonic anhydrase by COX-2-selective celecoxib: New pharmacological opportunities due to related binding site recognition
    • A. Weber, A. Casini, A. Heine, D. Kuhn, C.T. Supuran, A. Scozzafava, and G. Klebe Unexpected nanomolar inhibition of carbonic anhydrase by COX-2-selective celecoxib: new pharmacological opportunities due to related binding site recognition J. Med. Chem. 47 2004 550 557
    • (2004) J. Med. Chem. , vol.47 , pp. 550-557
    • Weber, A.1    Casini, A.2    Heine, A.3    Kuhn, D.4    Supuran, C.T.5    Scozzafava, A.6    Klebe, G.7
  • 34
    • 34548260898 scopus 로고    scopus 로고
    • Effects of celecoxib on voltage-gated calcium channel currents in rat pheochromocytoma (PC12) cells
    • Y. Zhang, J. Tao, H. Huang, G. Ding, Y. Cheng, and W. Sun Effects of celecoxib on voltage-gated calcium channel currents in rat pheochromocytoma (PC12) cells Pharmacol. Res. 56 2007 267 274
    • (2007) Pharmacol. Res. , vol.56 , pp. 267-274
    • Zhang, Y.1    Tao, J.2    Huang, H.3    Ding, G.4    Cheng, Y.5    Sun, W.6


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.