'Click' assembly of selective inhibitors for MAO-A

Bioorganic and Medicinal Chemistry Letters

Volumn 20, Issue 21, 2010, Pages 6222-6225

  Jia, Zhao ^a   Zhu, Qing ^a  

^a ZHEJIANG UNIVERSITY OF TECHNOLOGY   (China)

Author keywords

Click chemistry; Docking study; Monoamine oxidase; Selective inhibitors

Indexed keywords

AMINE OXIDASE (FLAVIN CONTAINING) ISOENZYME A; AMINE OXIDASE (FLAVIN CONTAINING) ISOENZYME B; MONOAMINE OXIDASE A INHIBITOR; MONOAMINE OXIDASE B INHIBITOR; TYROSINE;

ARTICLE; CHEMICAL REACTION; CLICK CHEMISTRY; CYCLOADDITION; DRUG BINDING; DRUG SYNTHESIS; ENZYME INHIBITION; IC 50; MOLECULAR DOCKING;

CATALYTIC DOMAIN; HYDROGEN BONDING; MODELS, MOLECULAR; MONOAMINE OXIDASE; MONOAMINE OXIDASE INHIBITORS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 77957888281     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2010.08.104     Document Type: Article

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