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Volumn 5, Issue 10, 2010, Pages 1717-1725

Synthesis and evaluation of bombesin analogues conjugated to two different triazolyl-derived chelators for 99mTc labeling

(7) Brans, Luc a García Garayoa, Elisa b Schweinsberg, Christian b Maes, Veronique a Struthers, Harriet c Schibli, Roger b,c Tourwé, Dirk a

a VRIJE UNIVERSITEIT BRUSSEL (Belgium)

b PAUL SCHERRER INSTITUTE (Switzerland)

c ETH ZURICH (Switzerland)

Author keywords

Bombesin; Chelators; Click chemistry; Radiochemistry; Triazolyl; Tumor targeting

Indexed keywords

BOMBESIN DERIVATIVE; CHELATING AGENT; GASTRIN RELEASING PEPTIDE RECEPTOR; N ALPHA CARBOXYMETHYLHISTIDINE; TECHNETIUM 99M; TRIAZOLE DERIVATIVE; UNCLASSIFIED DRUG;

AMINO ACID SEQUENCE; ANIMAL EXPERIMENT; ANIMAL MODEL; ARTICLE; BINDING AFFINITY; COMPUTER ASSISTED TOMOGRAPHY; CYCLOADDITION; DRUG CONJUGATION; DRUG DISTRIBUTION; DRUG EXCRETION; DRUG RECEPTOR BINDING; DRUG STRUCTURE; DRUG SYNTHESIS; DRUG UPTAKE; HUMAN; HUMAN CELL; ISOTOPE LABELING; MOUSE; NONHUMAN; PRIORITY JOURNAL; SINGLE PHOTON EMISSION COMPUTER TOMOGRAPHY;

ANIMALS; BOMBESIN; CATALYSIS; CELL LINE, TUMOR; CHELATING AGENTS; COPPER; HUMANS; ISOTOPE LABELING; MICE; MICE, NUDE; RECEPTORS, BOMBESIN; TECHNETIUM; TOMOGRAPHY, EMISSION-COMPUTED, SINGLE-PHOTON; TRIAZOLES; XENOGRAFT MODEL ANTITUMOR ASSAYS;

EID: 77957689595 PISSN: 18607179 EISSN: 18607187 Source Type: Journal
DOI: 10.1002/cmdc.201000191 Document Type: Article

Times cited : (16)

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