Optimization of physical characterization, skin permeation of naproxen from glycofurol-based topical gel

Asian Journal of Pharmaceutics

Volumn 4, Issue 2, 2010, Pages 154-162

  Barakat, Nahla S ^a  

^a KING SAUD UNIVERSITY   (Saudi Arabia)

Author keywords

Glycofurol; naproxen; permeation coefficient; physical stability; skin irritation test; topical delivery

Indexed keywords

CARBOPOL 974P; DIETHYLENE GLYCOL MONOETHYL ETHER; GANTREZ COPOLYMER; GELLING AGENT; GLYCOFUROL; GLYCOL; NAPROXEN; POLY(MALEIC ANHYDRIDE METHYL VINYL ETHER); POVIDONE; UNCLASSIFIED DRUG;

ADHESION; ANTIINFLAMMATORY ACTIVITY; ARTICLE; DRUG DIFFUSION; DRUG FORMULATION; DRUG PENETRATION; DRUG SAFETY; DRUG SCREENING; DRUG SOLUBILITY; DRUG STABILITY; DRUG TOLERABILITY; GEL; GELATION; NONHUMAN; PARAMETER; PH; RAT; SKIN IRRITATION; SKIN PENETRATION; SKIN PERMEABILITY; SKIN TEST; STEADY STATE; TRANSDERMAL DRUG ADMINISTRATION; VISCOSITY;

EID: 77956256435     PISSN: 09738398     EISSN: 1998409X     Source Type: Journal    
DOI: 10.4103/0973-8398.68468     Document Type: Article

References (41)

1. Mitchell JA, Warner TD. Cyclooxygenase-2: Pharmacology, physiology, biochemistry and relevance to NSAID therapy. Br J Pharmacol 1999;128:1121-1132
2. Vaile JH, Davis P. Topical NSAIDs for musculoskeletal conditions: A review of the literature. Drugs 1998;56:783-799
3. Burnham R, Gregg R, Healy P. The effectiveness of topical diclofenac for lateral epicondylitis. Clin J Sports Med 1998;8:78-81.
4. Moore RA, Tramer MR, Carroll D. Quantitive systematic review of topically applied non-steroidal anti-inflammatory drugs. Br Med J 1998;316:333-338
5. Monteiro-Riviere NA, Inman AD, Riviere JE, McNeill SC, Francoeur ML. Topical penetration of piroxicam is dependent on the distribution of the local cutaneous vasculature. Pharm Res 1993;10:1326-1331
6. Huang YB, Wu PC, Ko HM, Tsai YH. Cardamon oil as a skin permeation enhancer for indomethacin, piroxicam and diclofenac. Int J Pharm 1995;126:111-117
7. Yokomozo Y, Sagitani H. Effects of phospholipids on the percutaneous penetration of indomethacin through the dorsal skin of guinea pig in vitro. J Control Release 1996;38:267-274
8. Singh P, Roberts MS. Skin permeability and local tissue concentration of nonsteroidal anti-inflammatory drugs after topical application. J Pharmacol Exp Ther 1994;268:44-151.
9. Sioufi A, Pammer F, Boschet F. Percutaneous absorption of diclofenac in healthy volunteers after single and repeated topical application of diclofenac emugel. Biopharm Drug Dispos 1994;15:441-449
10. Giuliano F, Warner TD. Ex vivo assay to determine the cyclooxygenase selectivity of non-steroidal anti-inflammatory drugs. Br J Pharmacol 1999;12:1824-1830
11. Bonina F P, Puglia C, Barbuzzi T, De Caprariis P, Palagiano F, Rimoli MG, et al. In vitro and in vivo evaluation of polyoxyethylene esters as dermal prodrugs of ketoprofen, naproxen and diclofenac. Eur J Pharm Sci 2001;14:123-134
12. Glavas-Dodov M, Goracinova K, Mladenovska K, Fredro-Kumbaradzi E. Release profile of lidocaine HCl from topical liposomal gel formulation. Int J Pharm 2002;242:381-384
13. Pabla D, Zia H. A comparative permeation/release study of different testosterone gel formulations. Drug Deliv 2007;14:389-396
14. Sharma NC, Galustians HJ, Qaquish J, Galustians A, Rustogi KN, Petrone ME, et al. The clinical effectiveness of a dentifrice containing triclosan and a copolymer for controlling breath odor measured organoleptically twelve hours after tooth brushing. J Clin Dent 1999;10:131-134
15. Arbos P, Wirth M, Arangoa MA, Gabor F, Irache JM. Gantrez AN as a new polymer for the preparation of ligand-nanoparticle conjugates. J Control Release 2002;83:321-330
16. Shin SC, Cho CW, Choi HK. Permeation of piroxicam from the poloxamer gels. Drug Dev Ind Pharm 1999;25:273-278
17. Bonacucina G, Martelli S, Palmieri G F. Rheological, mucoadhesive and release properties of carbopol gels in hydrophilic cosolvents. Int J Pharm 2004;282:115-130
18. Shin SC, Lee J W, Yang KH, Chi H, Lee CH. Preparation and evaluation of bioadhesive benzocaine gels for enhanced local anesthetic effects. Int J Pharm 2003;260:77-81.
19. Lardy F, Vennat B, Pouget P, Pourrat A. Functionalization of hydrocolloids: Principal component analysis applied to the study of correlations between parameters describing the consistency of hydrogels. Drug Dev Ind Pharm 2000;26:715-721
20. Contreras MD, Sanchez M. Application of a factorial design to the study of the flow behavior, spreadability, transparency of Carbopol ETD 2020 gel. Part II. Int J Pharm 2002;234:149-157
21. Kleck CM. Gels and jellies. In: Swarbrick J, Boyland JC, editors. Encyclopedia of Pharmaceutical Technology. Vol.6. New York: Mercel Dekker; 1992. p. 415-439
22. Provost C, Herbost H, Kinget R. Transparent oil-water gels: Study of some physico-chemical and biopharmaceutical characteristics. Part 3: Viscosity and conductivity measurements. Pharm Ind. 1988;50:1190-1195
23. Martin AN, Banker GS, Chun AH. Rheology. In: Bean HS, Beckett AH, Carless JE, editors. Advances in Pharmaceutical Sciences. Vol.1. New York: Academic Press; 1967. p. 1-85.
24. Prentice JH. Measurements in the rheology of foodstuffs. London: Elsevier; 1984.
25. Balzer D, Varwig S, Weihrauch M. Viscoelasticity of personal care products. Coll Surf A Phys Eng Aspects 1995;99:233-246
26. Fang JY, Fang CL, Hong CT, Chen HY, Lin TY, Wei HM. Capsaicin and nonivamide as novel skin permeation enhancers for indomethacin. Eur J Pharm Sci 2001;12:195-203.
27. Suwanpidokkul N, Thongnopnua P, Umprayn K. Transdermal delivery of zidovudine (azt): The effects of vehicles, enhancers, and polymer membranes on permeation across cadaver pig skin. AAPS PharmSciTech 2004;5:e48.
28. Meidan VM, Al-Khallil M, Michniak BB. Enhanced iontophoretic delivery of buspirone hydrochloride across human skin using chemical enhancers. Int J Pharm 2003;264:73-83.
29. Patel SR, Zhong H, Sharma A, Kalia YN. In vitro and in vivo evaluation of the transdermal iontophoretic delivery of sumatriptan succinate. Eur J Pharm Biopharm 2007;66:296-301.
30. Tas C, Ozkan Y, Savaser A, Baykara T. In vitro release studies of chlorpheniramine maleate from gels prepared by different cellulose derivatives. Farmaco 2003;58:605-611
31. Namdeo A, Jain NK. Liquid crystalline pharmacogel based enhanced transdermal delivery of propranolo hydrochloride. J Control Release 2002;82:223-236
32. Mutalik S, Udupa N. Glibenclamide transdermal patches: Physicochemical, pharmacodynamic, and pharmacokinetic evaluations. J Pharm Sci 2004;3:1577-1594
33. Ugweke MI, Verbeke N, Kinget R. The biopharmaceutical aspects of nasal mucoadhesive drug delivery. J Pharm Pharmacol 2001;53:3-22.
34. Ho HO, Huang FC, Sokoloski TD, Sheu MT. The influence of cosolvents on the in vitro percutaneous penetration of diclofenac sodium from gel system. J Pharm Pharmacol 1994;46:636-642
35. Barry BW. Properties that influence percutaneous absorption, Chapter 4. In: Barry BW (Edt), Dermatological Formulations. Percutaneous Absorption. Vol.18, New York: Dekker; 1983. p. 127-233.
36. Takahashi A, Suzuki S, Kawasaki N, Kubo W, Miyazaki S, Loebenberg R, et al. Percutaneous absorption of non-steroidal anti-inflammatory drugs from in situ gelling xyloglucan formulations in rats. Int J Pharm 2002;246:179-186
37. Chow DS, Kaka I, Wang TI. Concentration dependent enhancement of 1-dodecylazacycloheptan-2-one on the percutaneous penetration kinetics of triamcinolone acetonide. J Pharm Sci 1984;73:1794-1799
38. Williams AC, Barry B W. Skin absorption enhancers. Crit Rev Ther Drug Carrier Syst 1992;9:305-353
39. Forslind B, Engstrom S, Enghlom J, Norlen L. A novel approach to the understanding of human skin function. J Dermatol Sci 1997;14: 115-125
40. Mura P, Faucci MT, Bramanti G, Corti P. Evaluation of transcutol as a clonazepam transdermal permeation enhancer from hydrophilic gel formulations. Eur J Pharm Sci 2000;9:365-372
41. Draize JH, Woodward G, Calvery HO. Methods for the study of irritation and toxicity of substances applied topically to the shin and mucous membranes. J Pharmacol Exp Ther 1944;82:377-379