Characterization of the biological effects of a novel protein kinase D inhibitor in endothelial cells

Biochemical Journal

Volumn 429, Issue 3, 2010, Pages 565-572

  Evans, Ian M ^a   Bagherzadeh, Azadeh ^b   Charles, Mark ^b   Raynham, Tony ^b   Ireson, Chris ^b   Boakes, Alexandra ^b   Kelland, Lloyd ^b   Zachary, Ian C ^a  

^a UNIVERSITY COLLEGE LONDON   (United Kingdom)

^b UNIVERSITY COLLEGE LONDON   (United Kingdom)

Author keywords

Angiogenesis; CRT5 inhibitor; Endothelium; Protein kinase C (PKC); Protein kinase D (PKD); Vascular endothelial growth factor (VEGF)

Indexed keywords

ANGIOGENESIS; CRT5 INHIBITOR; ENDOTHELIUM; PROTEIN KINASE C; PROTEIN KINASE D (PKD); VASCULAR ENDOTHELIAL GROWTH FACTOR;

AMIDES; FETAL MONITORING; PEPTIDES; PHOSPHORYLATION; RNA; SELF ASSEMBLY;

ENDOTHELIAL CELLS;

CRT5; CRT6; CYCLIC AMP RESPONSIVE ELEMENT BINDING PROTEIN; HEAT SHOCK PROTEIN 27; HISTONE DEACETYLASE 5; MITOGEN ACTIVATED PROTEIN KINASE; PROTEIN KINASE D; PROTEIN KINASE INHIBITOR; SMALL INTERFERING RNA; UNCLASSIFIED DRUG; VASCULOTROPIN; PROTEIN KINASE C; VASCULOTROPIN A; VASCULOTROPIN RECEPTOR 2;

ANGIOGENESIS; ARTICLE; CELL MIGRATION; CELL PROLIFERATION; CONTROLLED STUDY; ENDOTHELIUM CELL; GENETIC TRANSFECTION; HUMAN; HUMAN CELL; IN VITRO STUDY; PRIORITY JOURNAL; PROTEIN PHOSPHORYLATION; SIGNAL TRANSDUCTION; STATISTICAL SIGNIFICANCE; STIMULATION; UMBILICAL VEIN; CELL CULTURE; CELL MOTION; CYTOLOGY; DRUG ANTAGONISM; DRUG EFFECT; ENZYME SPECIFICITY; ENZYMOLOGY; METABOLISM; PHOSPHORYLATION; VASCULAR ENDOTHELIUM;

CELL MOVEMENT; CELL PROLIFERATION; CELLS, CULTURED; ENDOTHELIUM, VASCULAR; HUMANS; NEOVASCULARIZATION, PHYSIOLOGIC; PHOSPHORYLATION; PROTEIN KINASE C; PROTEIN KINASE INHIBITORS; SUBSTRATE SPECIFICITY; VASCULAR ENDOTHELIAL GROWTH FACTOR A; VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR-2;

EID: 77955071352     PISSN: 02646021     EISSN: 14708728     Source Type: Journal    
DOI: 10.1042/BJ20100578     Document Type: Article

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