Preparation and evaluation of sustained release matrix tablets of tramadol hydrochloride using glyceryl palmitostearate

Tropical Journal of Pharmaceutical Research

Volumn 9, Issue 3, 2010, Pages 275-281

  Deore, Rakesh K ^a   Kavitha, Kunchu ^a   Tamizhmani, Theetha G ^a  

^a BHARATHI COLLEGE OF PHARMACY   (India)

Author keywords

Direct compression; Glyceryl palmitostearate; Melt granulation; Sustained release; Tramadol hydrochloride

Indexed keywords

GLYCEROL PALMITOSTEARATE; TRAMADOL;

ARTICLE; COMPARATIVE STUDY; COMPRESSION; CONCENTRATION (PARAMETERS); CONTROLLED STUDY; DIFFUSION; DISSOLUTION; DRUG INTERACTION; DRUG RELEASE; INFRARED SPECTROSCOPY; KINETICS; RELEASE KINETICS; SUSTAINED RELEASE PREPARATION; TABLET HARDNESS;

EID: 77954159649     PISSN: 15965996     EISSN: 15969827     Source Type: Journal    
DOI: 10.4314/tjpr.v9i3.56289     Document Type: Article

References (22)

1. Gudsoorkar VR, Rambhau D. Influence variable of process one standard drug release from disintegrating sustained release Ibuprofen beads. The Eastern Pharmacist, 1997; 40: 111-113.
2. Wise DL. In Handbook of Pharmaceutical Controlled Release Technology. Marcel Dekker, New York and Basel; 2005. p. 435-440.
3. Bodmeier RA, Swarbrick J, Boylan JC. Eds. Encyclopedia of pharmaceutical technology. 2nd ed. Vol. III, New York Marcel Dekkerlnc; 1998. p. 2988-3000.
4. Hamdani J, Moes AJ, Amighi K. Physical & thermal characterization of Precirol & Compritol as lipophilic glycerides used for the preparation of controlled release matrix pellets. Int J Pharm, 2003; 260: 47-57.
5. Zang YE, Schwartz JB. Melt granulation and heat treatment for wax matrix-controlled drug release. Drug Dev Ind Pharm, 2003; 29: 131-138.
6. Hamdani J, Moes AJ, Amighi K. Development and evaluation of prolonged release pellets obtained by melt pelletization process. Int J Pharm, 2002; 245: 167-177.
7. Lloanusi NO, Schwartz JB. The effect of wax on compaction of microcrystalline cellulose beads made by extrusion and spheronization. Drug Dev Ind Pharm, 1998; 24: 37-44.
8. Barthelemy P, Laforet JP, Farah N, Joachim J. Compritol 888 ATO: an innovative hot melt coating agent for prolonged release drug formulations. Eur J Pharm Biopharm, 1999; 47: 87-90.
9. Chaudhari PD. Melt Granulation Technique: A Review, 2006 [cited 2006 Jan 8]. Available from Http://www.pharmainfo. net./exclusive/reviews.
10. Mahaparale PR, Kasture PV, Deshmukh SS, Kuchekar BS. Sustained release matrices of Metoprolol succinate using Compritol 888 ATO and Precirol ATO 05. J Pharm Res, 2006; 5: 10-14.
11. Liu J, Zhang F, McGinity JW. Properties of lipophilic matrix tablets containing Phenylpropanolamine HCL prepared by hot-melt extrusion. Eur J Pharm Biopharm, 2001; 52: 181-190.
12. Lehmann KA. Tramadol in acute pain. Drugs, 1997; 53: 25-33.
13. Rxlist. Tramadol hydrochloride-drug [cited 2009 Aug 25]. Available from http:// www.rxlist.com
14. Tiwari SB, Murthy TK, Pai MR, Mehta PR, Chowdhary PB. Controlled Release formulation of Tramadol Hydrochloride using Hydrophilic & Hydrophobic Matrix system. AAPS PharmsciTech, 2003; 4: 110-116.
15. Obaidat AA, Obaidat RM. Controlled release of Tramadol hydrochloride from matrices prepared using glyceryl behenate. Eur J Pharm Biopharm, 2001; 52: 231-235.
16. Malonne H, Fontaine J, Moes A. In vitro/in vivo characterization of a Tramadol Hydrochloride depote system composed of monoolein and water. Biol Pharm Bull, 2000; 23: 627-631.
17. Zhang ZY, Ping QN, Xiao B. Microencapsulation and characterization of Tramadol-resin complexes. J Control Rel, 2000; 66: 107-113.
18. Patel NM, Soniwala MM. Influence of release enhancer on release of Venlafaxine HCL from Glyceryl Behenate matrix tablet. Indian Drugs, 2008; 45: 98-104.
19. Harland R, Dubernet C, Benoit JP, Peppas N. A model of dissolution-controlled, release from non-swellable polymeric microspheres. J Control Rel, 2003; 6: 282-291.
20. Higuchi T. Mechanism of sustained action medication. Theoratical analysis of rate release of solid drugs dispersed in solid matrices. J Pharm Sci, 1963; 52: 1145-1149.
21. Korsmeyer RW, Gurny R, Doelker E, Buri P, Peppas NA. Mechanisms of solute release from porous hydrophilic polymers. Int J Pharm, 1983; 15: 25-35.
22. Reza MS, Quadir MA, Haider SS. Comparative evaluation of plastic, hydrophobic and hydrophilic polymers as matrices for controlled release drug delivery. J Pharm Pharmac Sci, 2003; 6: 282 -291.