Effect of limonene on permeation enhancement of ketoprofen in palm oil esters nanoemulsion

Journal of Oleo Science

Volumn 59, Issue 7, 2010, Pages 395-400

  Sakeena, M H F ^a   Elrashid, S M ^a   Muthanna, F A ^a   Ghassan, Z A ^a   Kanakal, M M ^a   Laila, Lia ^a   Munavvar, A S ^a   Azmin, M N ^a  

^a SCHOOL OF PHARMACEUTICAL SCIENCES   (Malaysia)

Author keywords

Ketoprofen; Palm oil esters; Permeation enhancement

Indexed keywords

CYCLOHEXENE DERIVATIVE; EMULSION; ESTER; KETOPROFEN; LIMONENE; NANOPARTICLE; PALM OIL; TERPENE; VEGETABLE OIL;

ANIMAL; DOSE RESPONSE; DRUG EFFECTS; EMULSION; IN VITRO STUDY; MALE; METABOLISM; PERMEABILITY; RAT; SKIN; SKIN ABSORPTION; SPRAGUE DAWLEY RAT; STIMULATION;

ANIMALS; CYCLOHEXENES; DOSE-RESPONSE RELATIONSHIP, DRUG; EMULSIONS; ESTERS; IN VITRO TECHNIQUES; KETOPROFEN; MALE; NANOPARTICLES; PERMEABILITY; PLANT OILS; RATS; RATS, SPRAGUE-DAWLEY; SKIN; SKIN ABSORPTION; STIMULATION, CHEMICAL; TERPENES;

EID: 77953521552     PISSN: 13458957     EISSN: 13473352     Source Type: Journal    
DOI: 10.5650/jos.59.395     Document Type: Article

References (25)

1. Kantor, T. G. Ketoprofen: A review of its pharmacologic and clinical properties. Pharmacotherapy 6, 93-103 (1986).
2. Cho, Y.J.; Choi, H. K. Enhancement of percutaneous absorption of ketoprofen: Effect of vehicles and adhesive matrix. Int. J. Pharm. 169, 95-104 (1998).
3. Cordero, J. A.; Alarcon, L.; Escribano, E.; Obach, R.; Domenech, J. A comparative study of the transdermal penetration of a series of NSAIDs drug. J. Pharm. Sci. 86, 503-508 (1997).
4. Dos Anjos, J. L. V.; Alonso, A. Terpenes increase the portioning and molecular dynamics of an amphipathic spin label in stratum corneum membranes. Int.J. Pharma. 350, 103-112 (2008).
5. Bouwstra, J. A.; Honeywell-Nguyen, P. L. Skin structure and mode of actions of vehicles. Adv. Drug Deliv. Rev. 54, S41-S55 (2002).
6. Rhee, Y. S.; Choi, J. G.; Park, E. S.; Chi, S. C. Transdermal delivery of ketoprofen using microemulsions. Int. J. Pharm. 228, 161-170 (2001).
7. Femenia'-Fonta, A.; Balaguer-Fernandez, C.; Merino, V.; Rodilla, V.; Lapez-Castellano, A. Effect of chemical enhancers on the in vitro percutaneous absorption of sumatriptan succinate. Eur. J. Pharm. Biopharm. 61, 50-55 (2005).
8. Barry, B. W. Lipid-protein-partitioning theory of skin penetration enhancement. J. Control. Res. 15, 237-248 (1991).
9. Vaddi, H. K.; Ho, P. C.; Chan, Y. W.; Chan, S. Y. Terpenes in propylene glycol as skin-penetration enhancers: Permeation and partition of haloperidol, Fourier transform infraredspectroscopy and differential scanning calorimetry. J. Pharm. Sci. 91, 1639-1651 (2002).
10. Aqil, M.; Ahad, A.; Sultana, Y.; Ali, A. Status of terpenes as skin penetration enhancers. Drug Discovery Today 12, 23/24 (1061-1067).
11. Koyama, Y.; Bando, H.; Yamashita, F.; Takakura, Y.; Sezaki, H.; Hashida, M. Comparative analysis of percutaneous absorption enhancement by D-limonene and oleic acid based on a skin diffusion model. Pharm. Res. 11, 377-383 (1994).
12. Tadros, T.; Izquierdo, P.; Esquena, J.; Solans, C. Formation and stability of nanoemulsions. Adv. Colloid Interface Sci. 108 (109), 303-318 (2004).
13. Keng, P. S.; Basri, M.; Zakaria, M. R. S.; Abdul Rahman, M. B.; Ariff, A. B.; Abbdul Rahman, R. N. Z.; Salleh, A. B. Newly synthesized palm esters for cosmetics industry. Indust. Crops & Products 29 (1), 37-44 (2009).
14. Gunawan, E. R.; Basri, M.; Abdulrahman, M. B.; Saleh, A. B.; Abdulrahman, R. N. Z. Lipase-catalyzed synthesis of Palmbased wax esters. J. Oleo. Sci. 53 (10), 471-477 (2004).
15. Keng, P. S., Basri, M., Abdul Rahman, M. B.; Salleh, A. B.; Abdul Rahman, R. N. Z.; Ariff, A. B. Optimization of palm-based wax esters production using statistical experiment design. J. Oleo. Sci. 54 (10), 519-528 (2005).
16. Basri, M.; Zakaria, M. R. S.; Huong, C. K.; Ismail, I.; Misran, M.; Kassim, A.; Salleh, A. B.; Abdul Rahman, R. N. Z.; Abdul Rahman, M. B. Formation and stability of new palm based nanoemulsions. Abstracts/J. Biotechnology 136S, S144-146 (2008).
17. Abdulrahman, M. B.; Huan, Q-Y.; Tejo, B. A.; Basri, M.; Salleh, A. B.;Rahman, R. N. Z. A. Self-assembly formation of palm-based esters nano-emulsion: A molecular dynamics study. Chem. Phys. Lett. 480, 220-224 (2009).
18. Sakeena, M. H. F.; Muthanna, F. A.; Ghassan, Z. A.; Kanakal, M. M.; Elrashid, S. M.; Munavvar, A. S.; Azmin, M. N. Formulation and in vitro evaluation of ketoprofen in palm oil esters nanoemulsion for topical delivery. J. Oleo Sci. 59 (4), 223-228 (2010).
19. Sakeena, M. H. F.; Kanakal, M. M.; Abdulkarim, M. F.; Abdullah, G. Z.; Akram, J.; Munavvar Zubaid, A. S.; Azmin, M. N. Development and validation of ketoprofen analysis by high performance liquid chromatography. Malaysian J. Pharm. 1 (7), 61 (2009).
20. Okabe, H.; Obata, Y.; Takayama, K.; Nagai, T. Percutaneous absorption enhancing effect and skin irritation of monocyclic monoterpenes. Drug Design & Delivery 6, 229-238 (1990).
21. Okabe, H.; Takayama, K.; Nagai, T. Percutaneous absorption of ketoprofen from acrylic gel patches containing d-loimonene and ethanol as absorption enhancers. Chem. Pharm. Bulletin 40, 1906-1910 (1992).
22. Gupta, P.; Garg, S. Recent advances in semisolid dosage forms for dermatological application. Pharm. Technol. 26, 144-161 (2002).
23. Williams, A. C.; Barry, B. W. Penetration enhancers. Adv. Drug Deliv. Rev. 56, 603-618 (2004).
24. Cornwell, P. A.; Barry, B. W.; Bouwstra, J. A.; Gooris, G. S. Modes of action of terpene penetration enhancers in human skin: Differential scanning calorimetry, small-angle X-ray diffraction and enhancer uptake studies. Int. J. Pharm. 127, 9-26 (1996).
25. Yamane, M. A.; Williams, A. C.; Barry, B. W. Effects of terpenes and oleic acid as skin penetration enhancers towards 5-fluorouracil as assessed with time: Permeation, partitioning and differential scanning calorimetry. Int. J. Pharm. 116, 237-251 (1995).