Development of colon targeted multiparticulate pulsatile drug delivery system for treating nocturnal asthma

Drug Delivery

Volumn 17, Issue 5, 2010, Pages 343-351

  Kadam, Vinayak D ^a   Gattani, Surendra G ^a  

^a R C PATEL INSTITUTE OF PHARMACEUTICAL EDUCATION AND RESEARCH   (India)

Author keywords

Colon targeted; Factorial design; Multiparticulate; Nocturnal asthma; Pulsatile drug delivery

Indexed keywords

EUDRAGIT; THEOPHYLLINE;

ANIMAL EXPERIMENT; ARTICLE; CONTROLLED STUDY; DRUG ABSORPTION; DRUG BLOOD LEVEL; DRUG COATING; DRUG DELIVERY SYSTEM; DRUG FORMULATION; DRUG PELLET; DRUG SOLUBILITY; INTESTINE FLUID; MALE; MAXIMUM PLASMA CONCENTRATION; NOCTURNAL ASTHMA; NONHUMAN; PH; PRIORITY JOURNAL; PULSATILE DRUG RELEASE; RABBIT; STOMACH JUICE; STOMACH PH; TIME TO MAXIMUM PLASMA CONCENTRATION;

ACRYLIC RESINS; ANIMALS; ASTHMA; BRONCHODILATOR AGENTS; COLON; DELAYED-ACTION PREPARATIONS; DRUG CHRONOTHERAPY; DRUG DELIVERY SYSTEMS; EXCIPIENTS; HYDROGEN-ION CONCENTRATION; MALE; POLYMETHACRYLIC ACIDS; RABBITS; SOLUBILITY; THEOPHYLLINE; TIME FACTORS;

EID: 77953262236     PISSN: 10717544     EISSN: 15210464     Source Type: Journal    
DOI: 10.3109/10717541003762821     Document Type: Article

References (34)

1. Akhgari, A., Farahmand, F., Garekani, H.A., Sadeghi, F., Vandamme, T.F. (2006). Permeability and swelling studies on free films containing inulin in combination with different polymethacrylates aimed for colonic drug delivery. Eur J Pharm S. 28:307-314
2. Akhgari, A., Garekani, H.A., Sadeghi, F., Azimaie, M. (2005). Statistical optimization of indomethacin pellets coated with pH-dependent methacrylic polymers for possible colonic drug delivery. Int J Pharm. 305:22-30.
3. Ashford, M., Fell, J.J., Sharma, D., Woathead, H. (1993). An evaluation of pectin as a carrier for drug targeting to the colon. J Contr Rel. 26:213-220
4. Bose, B., Cater, J.Z., Clark, R.A. (1987). A once daily theophylline preparation in prevention of nocturnal symptoms in childhood asthma. Eur J Pediatr. 146:524-527
5. Bussermar, T., Otto, L., Bodmier, R. (2001). Pulsatile drug delivery system. Crit. Rev Ther Drug Carrier System. 18:433-458
6. Chaudhari, S.P., Chauradhi, P.D., Mistry, C.J., Patil, M.J. (2007). The effect of core and coating composition on drug release from directly compressed time controlled release tablets. Pharm Tech. 31:132-144
7. Chourasia, N.K., Jain, N.K. (2003). Pharmaceutical approaches to the colon targeted drug delivery system. J Pharm Pharm Sci. 1:33-66.
8. Fukui, E., Miyamura, N., Uemura, K., Kobayashi, M. (2000). Preparation of enteric coated timed-release press-coated tablets and evaluation of their function by in vitro and in vivo tests for colon targeting. Int J Pharm. 204:7-15.
9. Gang, C., Feng, A., Mei-Juan, Z., Jin, S. (2004). Time and pH-dependent colon-specific drug delivery for orally administered diclofenac sodium and 5-amino salicylic acid. World J Gastroenterol. 10:1769-1774.
10. Gupta, K., Beckert, E., Price, C. (2001). A novel pH- and time based multiunit potential colonic drug delivery system. I. Development. Int J Pharm. 213:93-102.
11. Gupta, V.K., Beckent, T.E., Price, J.C. (1993). A novel pH and time based multi unit potential colonic drug delivery system. I. development. Int J Pharm. 3:83-91.
12. Hui, C., Shang, T., Su-Lan, H., Ping-Ping, W., Pei-Dawn, C. (2001). Effect of curcumin on theophylline pharmacokinetics in rabbits. J Chin Med. 12:51-59
13. Ibekwe, V.C., Khela, M.K., Evans, D.F., Basit, A.W. (2008). A new concept in colonic targeting: a combined pH-responsive and bacterially-triggered drug delivery technology. Aliment Pharmacol Ther. 28:911-916
14. Illet, K.F., Tee, L.B.G., Reeves, P.T., Minchin, R.F. (1990). Metabolism of drugs and other xenobiotics in the gut lumen and wall. Pharmacol Ther. 46:67-93.
15. Kadam, V.D., Gattani, S.G. (2009). Formulation and evaluation of a pulsatile drug delivery system using time- and pH-dependant polymers. Pharm Dev Tech. 15:57-63.
16. Kararli, T.T. (1995). Comparison of the gastrointestinal anatomy, physiology, and biochemistry of humans and commonly used laboratory animals. Biopharm D Dispo. 16:351-380
17. Keir, S., Page, C. (2008). The rabbit as a model to study asthma and other lung diseases. Pulmon Pharmacol Therap. 21:721-730
18. Kramer, J., Blume, H. (1994). Biopharmaceutical aspects of multiparticulates. In: Ghebre-Sellassie, ed. Multiparticulate oral drug delivery. 1st ed. New York: Marcel Dekker, 307-332
19. Lemmer, B. (1992). Why are so many biological system periodic? Proceedings of apv course. Pulsatile drug delivery. Currents Approaches and Future Trends, 20-22.
20. Mastiholimath, V.S., Dandagi, P.M., Jain, S.S., Gadad, A.P., Kulkarni, A.R. (2007). Time and pH dependent colon specific, pulsatile delivery of theophylline for nocturnal asthma. Int J Pharm. 328:49-56.
21. Nykanen, P., Lempaa, S., Aaltonen, M.L., Jurjenson, H., Veski, P., Marvola, M. (2001). Citric acid as excipient in multiple-unit enteric-coated pellets for targeting drugs on the colon. Int J Pharm. 229:155-162
22. Paola, M., Francesca, M., Marzia, C., Rodr, L.G., Guez M, Antonio, M.R.A. (2003). Development of enteric-coated pectin-based matrix tablets for colonic delivery of theophylline. J Drug Target. 11:365-371
23. Qi, M., Wang, P., Wu, D. (2003). A novel pH- and time-dependent system for colonic drug delivery. Drug Dev Ind Pharm. 29:661-667
24. Rane, A.B., Gattani, S.G., Kadam, V.D., Tekade, A.R. (2009). Formulation and evaluation of press coated tablets for pulsatile drug delivery using hydrophilic and hydrophobic polymers. Chem Pharm Bull. 57:1213-1217
25. Rao, K.P., Patil, C.C. (2007). Formulation and evaluation of colon targeted oral tablets of naproxen. Ind J Pharm Educ Res. 146-149
26. Schellekens, R.C.A., Stellaard, F., Mitrovic, D., Stuurman, F.E., Kosterinka, J.G.W., Frijlink, H.W. (2008). Pulsatile drug delivery to ileo-colonic segments by structured incorporation of disintegrants in pH-responsive polymer coatings. J Contr Rel. 132:91-98
27. Siepmann, F., Muschert, S., Leclercq, B., Carlin, B., Siepmann, J. (2008). How to improve the storage stability of aqueous polymeric film coatings. J Contr Rel. 126:26-33.
28. Smith, H.W. (1965). Observations of the flora of the alimentary tract of animals and factors affecting its composition. J Pathol Bacteriol. 89:95-122.
29. Staib, A.H., Loew, D., Harder, S., Graul, E.H., Pfab, R. (1986). Measurement of theophylline absorption from different regions of the gastro-intestinal tract using a remote controlled drug delivery device. Eur J Clin Pharmacol. 30:691-697
30. Sutherland, E.U., Nalson, H.S. (1996). Nocturnal asthma. J Allergy Clin Immunol. 1179-1186
31. Tekade, A.R., Gattani, S.G. (2009). Development and evaluation of pulsatile drug delivery system using novel polymer. Pharm Dev Tech. 14:380-387.
32. Watts, P.J., Illum, L. (1997). Colonic drug delivery. Drug Dev Ind Pharm. 23:893-913.
33. Youan, B.C. (2004). Chronopharmaceutics, gimmick or clinically relevant approach to drug delivery. J Contr Rel. 98:337-353
34. Zahirul, K., Zeljko, M.I.P., Nevenka, K. (1999). A pH-dependent colon targeted oral drug delivery system using methacrylic acid copolymers. I. Manipulation of drug release using Eudragit® L100-55 and Eudragit® ; S100 combinations. J Contr Rel. 58:215-222