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Volumn 54, Issue 6, 2010, Pages 2379-2384

Semimechanistic pharmacokinetic-pharmacodynamic model with adaptation development for time-kill experiments of ciprofloxacin against Pseudomonas aeruginosa

Author keywords

[No Author keywords available]

Indexed keywords

AMIDE; CARRIER PROTEIN; CIPROFLOXACIN; DRUG CARRIER; MEX PROTEIN; PHENYLARGININE BETA NAPHTHYLAMIDE; UNCLASSIFIED DRUG;

EID: 77952597327     PISSN: 00664804     EISSN: 10986596     Source Type: Journal    
DOI: 10.1128/AAC.01478-08     Document Type: Article
Times cited : (21)

References (38)
  • 1
    • 0345466364 scopus 로고    scopus 로고
    • Involvement of an active efflux system in the natural resistance of Pseudomonas aeruginosa to aminoglycosides
    • Aires, J. R., T. Kohler, H. Nikaido, and P. Plesiat. 1999. Involvement of an active efflux system in the natural resistance of Pseudomonas aeruginosa to aminoglycosides. Antimicrob. Agents Chemother. 43:2624-2628.
    • (1999) Antimicrob. Agents Chemother. , vol.43 , pp. 2624-2628
    • Aires, J.R.1    Kohler, T.2    Nikaido, H.3    Plesiat, P.4
  • 2
    • 0034924146 scopus 로고    scopus 로고
    • Type II topoisomerase mutations in fluoroquinolone-resistant clinical strains of Pseudomonas aeruginosa isolated in 1998 and 1999: Role of target enzyme in mechanism of fluoroquinolone resistance
    • Akasaka, T., M. Tanaka, A. Yamaguchi, and K. Sato. 2001. Type II topoisomerase mutations in fluoroquinolone-resistant clinical strains of Pseudomonas aeruginosa isolated in 1998 and 1999: role of target enzyme in mechanism of fluoroquinolone resistance. Antimicrob. Agents Chemother. 45: 2263-2268.
    • (2001) Antimicrob. Agents Chemother. , vol.45 , pp. 2263-2268
    • Akasaka, T.1    Tanaka, M.2    Yamaguchi, A.3    Sato, K.4
  • 3
    • 0032839484 scopus 로고    scopus 로고
    • Stability of antibiotics used for antibiotic-lock treatment of infections of implantable venous devices (ports)
    • Anthony, T. U., and L. G. Rubin. 1999. Stability of antibiotics used for antibiotic-lock treatment of infections of implantable venous devices (ports). Antimicrob. Agents Chemother. 43:2074-2076.
    • (1999) Antimicrob. Agents Chemother. , vol.43 , pp. 2074-2076
    • Anthony, T.U.1    Rubin, L.G.2
  • 5
    • 0023176033 scopus 로고
    • Comparative study with enoxacin and netilmicin in a pharmacodynamic model to determine importance of ratio of antibiotic peak concentration to MIC for bactericidal activity and emergence of resistance
    • Blaser, J., B. B. Stone, M. C. Groner, and S. H. Zinner. 1987. Comparative study with enoxacin and netilmicin in a pharmacodynamic model to determine importance of ratio of antibiotic peak concentration to MIC for bactericidal activity and emergence of resistance. Antimicrob. Agents Chemother. 31:1054-1060.
    • (1987) Antimicrob. Agents Chemother. , vol.31 , pp. 1054-1060
    • Blaser, J.1    Stone, B.B.2    Groner, M.C.3    Zinner, S.H.4
  • 6
    • 59749102442 scopus 로고    scopus 로고
    • Development and qualification of a pharmacodynamic model for the pronounced inoculum effect of ceftazidime against Pseudomonas aeruginosa
    • Bulitta, J. B., N. S. Ly, J. C. Yang, A. Forrest, W. J. Jusko, and B. T. Tsuji. 2009. Development and qualification of a pharmacodynamic model for the pronounced inoculum effect of ceftazidime against Pseudomonas aeruginosa. Antimicrob. Agents Chemother. 53:46-56.
    • (2009) Antimicrob. Agents Chemother. , vol.53 , pp. 46-56
    • Bulitta, J.B.1    Ly, N.S.2    Yang, J.C.3    Forrest, A.4    Jusko, W.J.5    Tsuji, B.T.6
  • 7
    • 33748677949 scopus 로고    scopus 로고
    • Mechanism-based pharmacodynamic models of fluoroquinolone resistance in Staphylococcus aureus
    • Chung, P., P. J. McNamara, J. J. Campion, and M. E. Evans. 2006. Mechanism- based pharmacodynamic models of fluoroquinolone resistance in Staphylococcus aureus. Antimicrob. Agents Chemother. 50:2957-2965.
    • (2006) Antimicrob. Agents Chemother. , vol.50 , pp. 2957-2965
    • Chung, P.1    McNamara, P.J.2    Campion, J.J.3    Evans, M.E.4
  • 8
    • 0031407768 scopus 로고    scopus 로고
    • DNA gyrase, topoisomerase IV, and the 4-quinolones
    • Drlica, K., and X. Zhao. 1997. DNA gyrase, topoisomerase IV, and the 4-quinolones. Microbiol. Mol. Biol. Rev. 61:377-392.
    • (1997) Microbiol. Mol. Biol. Rev. , vol.61 , pp. 377-392
    • Drlica, K.1    Zhao, X.2
  • 9
    • 0025734363 scopus 로고
    • Ionic binding, adaptive resistance and post-antibiotic effect of netilmicin and ciprofloxacin
    • Gould, I. M., K. Milne, G. Harvey, and C. Jason. 1991. Ionic binding, adaptive resistance and post-antibiotic effect of netilmicin and ciprofloxacin. J. Antimicrob. Chemother. 27:741-748.
    • (1991) J. Antimicrob. Chemother. , vol.27 , pp. 741-748
    • Gould, I.M.1    Milne, K.2    Harvey, G.3    Jason, C.4
  • 12
    • 0033081949 scopus 로고    scopus 로고
    • Mechanisms of fluoroquinolone resistance
    • Hooper, D. C. 1999. Mechanisms of fluoroquinolone resistance. Drug Resist. Updat. 2:38-55.
    • (1999) Drug Resist. Updat. , vol.2 , pp. 38-55
    • Hooper, D.C.1
  • 13
    • 21844477302 scopus 로고    scopus 로고
    • Mechanisms of resistance to quinolones
    • Jacoby, G. A. 2005. Mechanisms of resistance to quinolones. Clin. Infect. Dis. 41:S120-S126.
    • (2005) Clin. Infect. Dis. , vol.41
    • Jacoby, G.A.1
  • 15
    • 43249096035 scopus 로고    scopus 로고
    • Pharmacokinetic-pharmacodynamic modeling and simulation for in vivo bactericidal effect in murine infection model
    • Katsube, T., Y. Yamano, and Y. Yano. 2008. Pharmacokinetic- pharmacodynamic modeling and simulation for in vivo bactericidal effect in murine infection model. J. Pharm. Sci. 97:1606-1614.
    • (2008) J. Pharm. Sci. , vol.97 , pp. 1606-1614
    • Katsube, T.1    Yamano, Y.2    Yano, Y.3
  • 16
    • 12944249381 scopus 로고    scopus 로고
    • Use of an efflux pump inhibitor to determine the prevalence of efflux pump-mediated fluoroquinolone resistance and multidrug resistance in Pseudomonas aeruginosa
    • Kriengkauykiat, J., E. Porter, O. Lomovskaya, and A. Wong-Beringer. 2005. Use of an efflux pump inhibitor to determine the prevalence of efflux pump-mediated fluoroquinolone resistance and multidrug resistance in Pseudomonas aeruginosa. Antimicrob. Agents Chemother. 49:565-570.
    • (2005) Antimicrob. Agents Chemother. , vol.49 , pp. 565-570
    • Kriengkauykiat, J.1    Porter, E.2    Lomovskaya, O.3    Wong-Beringer, A.4
  • 17
    • 0029129966 scopus 로고
    • Role of mexA-mexB-oprM in antibiotic efflux in Pseudomonas aeruginosa
    • Li, X. Z., H. Nikaido, and K. Poole. 1995. Role of mexA-mexB-oprM in antibiotic efflux in Pseudomonas aeruginosa. Antimicrob. Agents Chemother. 39:1948-1953.
    • (1995) Antimicrob. Agents Chemother. , vol.39 , pp. 1948-1953
    • Li, X.Z.1    Nikaido, H.2    Poole, K.3
  • 18
    • 33644656533 scopus 로고    scopus 로고
    • Efficacy and potential for resistance selection of antipseudomonal treatments in a mouse model of lung infection by hypermutable Pseudomonas aeruginosa
    • Macia, M. D., N. Borrell, M. Segura, C. Gomez, J. L. Perez, and A. Oliver. 2006. Efficacy and potential for resistance selection of antipseudomonal treatments in a mouse model of lung infection by hypermutable Pseudomonas aeruginosa. Antimicrob. Agents Chemother. 50:975-983.
    • (2006) Antimicrob. Agents Chemother. , vol.50 , pp. 975-983
    • Macia, M.D.1    Borrell, N.2    Segura, M.3    Gomez, C.4    Perez, J.L.5    Oliver, A.6
  • 19
    • 0037403960 scopus 로고    scopus 로고
    • Diversity of mechanism-based pharmacodynamic models
    • Mager, D. E., E. Wyska, and W. J. Jusko. 2003. Diversity of mechanism-based pharmacodynamic models. Drug Metab. Dispos. 31:510-518.
    • (2003) Drug Metab. Dispos. , vol.31 , pp. 510-518
    • Mager, D.E.1    Wyska, E.2    Jusko, W.J.3
  • 20
    • 27644575196 scopus 로고    scopus 로고
    • Bacterial efflux systems and efflux pumps inhibitors
    • Marquez, B. 2005. Bacterial efflux systems and efflux pumps inhibitors. Biochimie 87:1137-1147 .
    • (2005) Biochimie , vol.87 , pp. 1137-1147
    • Marquez, B.1
  • 22
    • 18844452358 scopus 로고    scopus 로고
    • Standardization of pharmacokinetic/pharmacodynamic (PK/PD) terminology for anti-infective drugs: An update
    • Mouton, J. W., M. N. Dudley, O. Cars, H. Derendorf, and G. L. Drusano. 2005. Standardization of pharmacokinetic/pharmacodynamic (PK/PD) terminology for anti-infective drugs: an update. J. Antimicrob. Chemother. 55:601-607.
    • (2005) J. Antimicrob. Chemother. , vol.55 , pp. 601-607
    • Mouton, J.W.1    Dudley, M.N.2    Cars, O.3    Derendorf, H.4    Drusano, G.L.5
  • 23
    • 13244281964 scopus 로고    scopus 로고
    • Pharmacokinetic/pharmacodynamic modelling of antibacterials in vitro and in vivo using bacterial growth and kill kinetics: The minimum inhibitory concentration versus stationary concentration
    • Mouton, J. W., and A. A. Vinks. 2005. Pharmacokinetic/pharmacodynamic modelling of antibacterials in vitro and in vivo using bacterial growth and kill kinetics: the minimum inhibitory concentration versus stationary concentration. Clin. Pharmacokinet. 44:201-210.
    • (2005) Clin. Pharmacokinet. , vol.44 , pp. 201-210
    • Mouton, J.W.1    Vinks, A.A.2
  • 24
    • 0030985564 scopus 로고    scopus 로고
    • Pharmacokinetic-pharmacodynamic modeling of activity of ceftazidime during continuous and intermittent infusion
    • Mouton, J. W., A. A. Vinks, and N. C. Punt. 1997. Pharmacokinetic- pharmacodynamic modeling of activity of ceftazidime during continuous and intermittent infusion. Antimicrob. Agents Chemother. 41:733-738.
    • (1997) Antimicrob. Agents Chemother. , vol.41 , pp. 733-738
    • Mouton, J.W.1    Vinks, A.A.2    Punt, N.C.3
  • 25
    • 33846024399 scopus 로고    scopus 로고
    • Semimechanistic pharmacokinetic/pharmacodynamic model for assessment of activity of antibacterial agents from time-kill curve experiments
    • Nielsen, E. I., A. Viberg, E. Lowdin, O. Cars, M. O. Karlsson, and M. Sandstrom. 2007. Semimechanistic pharmacokinetic/pharmacodynamic model for assessment of activity of antibacterial agents from time-kill curve experiments. Antimicrob. Agents Chemother. 51:128-136.
    • (2007) Antimicrob. Agents Chemother. , vol.51 , pp. 128-136
    • Nielsen, E.I.1    Viberg, A.2    Lowdin, E.3    Cars, O.4    Karlsson, M.O.5    Sandstrom, M.6
  • 26
    • 13344270397 scopus 로고    scopus 로고
    • Determination of free extracellular concentrations of piperacillin by microdialysis
    • Nolting, A., T. D. Costa, R. Vistelle, K. H. Rand, and H. Derendorf. 1996. Determination of free extracellular concentrations of piperacillin by microdialysis. J. Pharm. Sci. 85:369-372.
    • (1996) J. Pharm. Sci. , vol.85 , pp. 369-372
    • Nolting, A.1    Costa, T.D.2    Vistelle, R.3    Rand, K.H.4    Derendorf, H.5
  • 27
    • 26044458858 scopus 로고    scopus 로고
    • Nosocomial infections due to multidrug-resistant Pseudomonas aeruginosa: Epidemiology and treatment options
    • DOI 10.1592/phco.2005.25.10.1353
    • Obritsch, M. D., D. N. Fish, R. MacLaren, and R. Jung. 2005. Nosocomial infections due to multidrug-resistant Pseudomonas aeruginosa: epidemiology and treatment options. Pharmacotherapy 25:1353-1364. (Pubitemid 41407633)
    • (2005) Pharmacotherapy , vol.25 , Issue.10 I , pp. 1353-1364
    • Obritsch, M.D.1    Fish, D.N.2    MacLaren, R.3    Jung, R.4
  • 28
    • 33845879085 scopus 로고    scopus 로고
    • Mutant prevention concentration of ciprofloxacin and enrofloxacin against Escherichia coli, Salmonella Typhimurium and Pseudomonas aeruginosa
    • Pasquali, F., and G. Manfreda. 2007. Mutant prevention concentration of ciprofloxacin and enrofloxacin against Escherichia coli, Salmonella Typhimurium and Pseudomonas aeruginosa. Vet. Microbiol. 119:304-310.
    • (2007) Vet. Microbiol. , vol.119 , pp. 304-310
    • Pasquali, F.1    Manfreda, G.2
  • 29
    • 34447271963 scopus 로고    scopus 로고
    • Influence of high mutation rates on the mechanisms and dynamics of in vitro and in vivo resistance development to single or combined antipseudomonal agents
    • Plasencia, V., N. Borrell, M. D. Macia, B. Moya, J. L. Perez, and A. Oliver. 2007. Influence of high mutation rates on the mechanisms and dynamics of in vitro and in vivo resistance development to single or combined antipseudomonal agents. Antimicrob. Agents Chemother. 51:2574-2581.
    • (2007) Antimicrob. Agents Chemother. , vol.51 , pp. 2574-2581
    • Plasencia, V.1    Borrell, N.2    Macia, M.D.3    Moya, B.4    Perez, J.L.5    Oliver, A.6
  • 30
    • 0038440791 scopus 로고    scopus 로고
    • Mechanisms of resistance to quinolones: Target alterations, decreased accumulation and DNA gyrase protection
    • Ruiz, J. 2003. Mechanisms of resistance to quinolones: target alterations, decreased accumulation and DNA gyrase protection. J. Antimicrob. Chemother. 51:1109-1117.
    • (2003) J. Antimicrob. Chemother. , vol.51 , pp. 1109-1117
    • Ruiz, J.1
  • 31
    • 71249107458 scopus 로고    scopus 로고
    • Pharmacokinetic-pharmacodynamic modeling of the in vitro activities of oxazolidinone antimicrobial agents against methicillin-resistant Staphylococcus aureus
    • Schmidt, S., S. N. Sabarinath, A. Barbour, D. Abbanat, P. Manitpisitkul, S. Sha, and H. Derendorf. 2009. Pharmacokinetic-pharmacodynamic modeling of the in vitro activities of oxazolidinone antimicrobial agents against methicillin-resistant Staphylococcus aureus. Antimicrob. Agents Chemother. 53:5039-5045.
    • (2009) Antimicrob. Agents Chemother. , vol.53 , pp. 5039-5045
    • Schmidt, S.1    Sabarinath, S.N.2    Barbour, A.3    Abbanat, D.4    Manitpisitkul, P.5    Sha, S.6    Derendorf, H.7
  • 32
    • 31444440959 scopus 로고    scopus 로고
    • Pharmacokinetic/ pharmacodynamic (PK/PD) evaluation of a once-daily treatment using ciprofloxacin in an extended-release dosage form
    • Schuck, E. L., A. Dalhoff, H. Stass, and H. Derendorf. 2005. Pharmacokinetic/ pharmacodynamic (PK/PD) evaluation of a once-daily treatment using ciprofloxacin in an extended-release dosage form. Infection 33(Suppl. 2):22-28.
    • (2005) Infection , vol.33 , Issue.SUPPL. 2 , pp. 22-28
    • Schuck, E.L.1    Dalhoff, A.2    Stass, H.3    Derendorf, H.4
  • 33
    • 0346694551 scopus 로고    scopus 로고
    • Efflux as a mechanism of resistance to antimicrobials in Pseudomonas aeruginosa and related bacteria: Unanswered questions
    • Schweizer, H. P. 2003. Efflux as a mechanism of resistance to antimicrobials in Pseudomonas aeruginosa and related bacteria: unanswered questions. Genet. Mol. Res. 2:48-62.
    • (2003) Genet. Mol. Res. , vol.2 , pp. 48-62
    • Schweizer, H.P.1
  • 34
    • 18844410491 scopus 로고    scopus 로고
    • Modelling time-kill studies to discern the pharmacodynamics of meropenem
    • Tam, V. H., A. N. Schilling, and M. Nikolaou. 2005. Modelling time-kill studies to discern the pharmacodynamics of meropenem. J. Antimicrob. Chemother. 55:699-706.
    • (2005) J. Antimicrob. Chemother. , vol.55 , pp. 699-706
    • Tam, V.H.1    Schilling, A.N.2    Nikolaou, M.3
  • 35
    • 0032708146 scopus 로고    scopus 로고
    • Pharmacokinetics and pharmacodynamics of fluoroquinolones
    • Turnidge, J. 1999. Pharmacokinetics and pharmacodynamics of fluoroquinolones. Drugs 58(Suppl. 2):29-36.
    • (1999) Drugs , vol.58 , Issue.SUPPL. 2 , pp. 29-36
    • Turnidge, J.1
  • 36
    • 0038323939 scopus 로고    scopus 로고
    • Antibiotic efflux pumps in eukaryotic cells: Occurrence and impact on antibiotic cellular pharmacokinetics, pharmacodynamics and toxicodynamics
    • Van Bambeke, F., J. M. Michot, and P. M. Tulkens. 2003. Antibiotic efflux pumps in eukaryotic cells: occurrence and impact on antibiotic cellular pharmacokinetics, pharmacodynamics and toxicodynamics. J. Antimicrob. Chemother. 51:1067-1077.
    • (2003) J. Antimicrob. Chemother. , vol.51 , pp. 1067-1077
    • Van Bambeke, F.1    Michot, J.M.2    Tulkens, P.M.3
  • 37
    • 40549127440 scopus 로고    scopus 로고
    • Mechanism-based pharmacokinetic-pharmacodynamic models of in vitro fungistatic and fungicidal effects against Candida albicans
    • Venisse, N., N. Gregoire, M. Marliat, and W. Couet. 2008. Mechanism-based pharmacokinetic-pharmacodynamic models of in vitro fungistatic and fungicidal effects against Candida albicans. Antimicrob. Agents Chemother. 52: 937-943.
    • (2008) Antimicrob. Agents Chemother. , vol.52 , pp. 937-943
    • Venisse, N.1    Gregoire, N.2    Marliat, M.3    Couet, W.4
  • 38
    • 8844283457 scopus 로고    scopus 로고
    • Role of efflux mechanisms on fluoroquinolone resistance in Streptococcus pneumoniae and Pseudomonas aeruginosa
    • Zhanel, G. G., D. J. Hoban, K. Schurek, and J. A. Karlowsky. 2004. Role of efflux mechanisms on fluoroquinolone resistance in Streptococcus pneumoniae and Pseudomonas aeruginosa. Int. J. Antimicrob. Agents 24:529-535.
    • (2004) Int. J. Antimicrob. Agents , vol.24 , pp. 529-535
    • Zhanel, G.G.1    Hoban, D.J.2    Schurek, K.3    Karlowsky, J.A.4


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